JP2022526364A5 - - Google Patents
Info
- Publication number
- JP2022526364A5 JP2022526364A5 JP2021557761A JP2021557761A JP2022526364A5 JP 2022526364 A5 JP2022526364 A5 JP 2022526364A5 JP 2021557761 A JP2021557761 A JP 2021557761A JP 2021557761 A JP2021557761 A JP 2021557761A JP 2022526364 A5 JP2022526364 A5 JP 2022526364A5
- Authority
- JP
- Japan
- Prior art keywords
- independently selected
- substituted
- pharmaceutically acceptable
- acceptable salt
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1904373.6 | 2019-03-29 | ||
| GBGB1904373.6A GB201904373D0 (en) | 2019-03-29 | 2019-03-29 | Novel compounds and pharamaceutical compositions thereof for the treatment of inflammatory disorders |
| PCT/EP2020/058064 WO2020200900A1 (en) | 2019-03-29 | 2020-03-24 | Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022526364A JP2022526364A (ja) | 2022-05-24 |
| JP2022526364A5 true JP2022526364A5 (https=) | 2023-04-03 |
Family
ID=66442982
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021557761A Pending JP2022526364A (ja) | 2019-03-29 | 2020-03-24 | 炎症性障害の治療のための新規化合物及びその医薬組成物 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US20220218679A1 (https=) |
| EP (1) | EP3947378B1 (https=) |
| JP (1) | JP2022526364A (https=) |
| KR (1) | KR20210145238A (https=) |
| CN (1) | CN113646305A (https=) |
| AR (1) | AR118521A1 (https=) |
| AU (1) | AU2020252038A1 (https=) |
| BR (1) | BR112021019055A2 (https=) |
| CA (1) | CA3134736A1 (https=) |
| CO (1) | CO2021014223A2 (https=) |
| GB (1) | GB201904373D0 (https=) |
| IL (1) | IL286677A (https=) |
| MA (1) | MA55497A (https=) |
| MX (1) | MX2021011576A (https=) |
| PH (1) | PH12021552375A1 (https=) |
| SG (1) | SG11202110644WA (https=) |
| TW (1) | TW202102501A (https=) |
| WO (1) | WO2020200900A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201904375D0 (en) * | 2019-03-29 | 2019-05-15 | Galapagos Nv | Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders |
| GB201904374D0 (en) * | 2019-03-29 | 2019-05-15 | Galapagos Nv | Novel compunds and pharmaceutical composistions thereof for the treatment of inflammatory disorders |
| CN113243338A (zh) * | 2021-05-14 | 2021-08-13 | 福州大学 | 一种小鼠缺血性卒中模型的构建与评估方法 |
| EP4434981A4 (en) * | 2021-12-23 | 2025-08-20 | Hangzhou Polymed Biopharmaceuticals Inc | FIVE- AND SIX-MEMBERED COMPOUND, ITS PREPARATION PROCESS AND PHARMACEUTICAL COMPOSITION AND ITS USE |
| WO2024133560A1 (en) * | 2022-12-21 | 2024-06-27 | Dark Blue Therapeutics Ltd | Imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine derivatives as mllt1 and mllt3 inhibitors |
| EP4389747A1 (en) * | 2022-12-21 | 2024-06-26 | Dark Blue Therapeutics Ltd | Imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrazine derivatives as mllt1 and mllt3 inhibitors |
| CN119751445B (zh) * | 2024-12-10 | 2025-11-25 | 江南大学 | 6-乙炔基吡唑并[1,5-a]吡啶的制备方法 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1657242A4 (en) * | 2003-08-15 | 2008-10-29 | Banyu Pharma Co Ltd | imidazopyridine |
| JPWO2005108399A1 (ja) * | 2004-05-10 | 2008-03-21 | 萬有製薬株式会社 | イミダゾピリジン化合物 |
| US9169260B2 (en) * | 2011-03-22 | 2015-10-27 | Merck Sharp & Dohme Corp. | Amidopyrazole inhibitors of interleukin receptor-associated kinases |
| GB201401086D0 (en) * | 2014-01-23 | 2014-03-12 | Galapagos Nv | Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders |
| JP2018524372A (ja) * | 2015-07-15 | 2018-08-30 | アウリジーン ディスカバリー テクノロジーズ リミテッド | Ｉｒａｋ−４阻害剤としてのインダゾール及びアザインダゾール化合物 |
| GB201518456D0 (en) * | 2015-10-19 | 2015-12-02 | Galapagos Nv | Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory, autoimmune and/or proliferative diseases |
| WO2018060174A1 (de) * | 2016-09-29 | 2018-04-05 | Bayer Pharma Aktiengesellschaft | Substituierte benzimidazole, pharmazeutische präparate diese enthaltend, sowie deren verwendung zur herstellung von arzneimitteln |
| WO2018060072A1 (de) * | 2016-09-29 | 2018-04-05 | Bayer Pharma Aktiengesellschaft | Neue substituierte benzimidazole, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln |
| CN109890829B (zh) * | 2016-11-02 | 2022-07-15 | 豪夫迈·罗氏有限公司 | 作为IRAK4调节剂的吡唑并[1,5a]嘧啶衍生物 |
| CN110835338A (zh) * | 2018-08-17 | 2020-02-25 | 浙江海正药业股份有限公司 | 咪唑并吡啶类衍生物及其制备方法和其在医药上的用途 |
| MA54755A (fr) * | 2019-01-18 | 2021-11-24 | Biogen Ma Inc | Dérivés d'imidazo[1,2-a]pyridinyle servant d'inhibiteurs d'irak4 |
| GB201904374D0 (en) * | 2019-03-29 | 2019-05-15 | Galapagos Nv | Novel compunds and pharmaceutical composistions thereof for the treatment of inflammatory disorders |
| GB201904375D0 (en) * | 2019-03-29 | 2019-05-15 | Galapagos Nv | Novel compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders |
-
2019
- 2019-03-29 GB GBGB1904373.6A patent/GB201904373D0/en not_active Ceased
-
2020
- 2020-03-24 US US17/599,465 patent/US20220218679A1/en not_active Abandoned
- 2020-03-24 MX MX2021011576A patent/MX2021011576A/es unknown
- 2020-03-24 MA MA055497A patent/MA55497A/fr unknown
- 2020-03-24 JP JP2021557761A patent/JP2022526364A/ja active Pending
- 2020-03-24 WO PCT/EP2020/058064 patent/WO2020200900A1/en not_active Ceased
- 2020-03-24 SG SG11202110644WA patent/SG11202110644WA/en unknown
- 2020-03-24 CN CN202080025098.XA patent/CN113646305A/zh active Pending
- 2020-03-24 AU AU2020252038A patent/AU2020252038A1/en not_active Abandoned
- 2020-03-24 BR BR112021019055A patent/BR112021019055A2/pt not_active IP Right Cessation
- 2020-03-24 CA CA3134736A patent/CA3134736A1/en active Pending
- 2020-03-24 KR KR1020217035254A patent/KR20210145238A/ko not_active Ceased
- 2020-03-24 PH PH1/2021/552375A patent/PH12021552375A1/en unknown
- 2020-03-24 EP EP20715295.0A patent/EP3947378B1/en active Active
- 2020-03-27 AR ARP200100870A patent/AR118521A1/es not_active Application Discontinuation
- 2020-03-27 TW TW109110404A patent/TW202102501A/zh unknown
-
2021
- 2021-09-26 IL IL286677A patent/IL286677A/en unknown
- 2021-10-25 CO CONC2021/0014223A patent/CO2021014223A2/es unknown
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