JP2022525926A - 胃内滞留剤形用のカプセル及びカプセルコーティング - Google Patents

胃内滞留剤形用のカプセル及びカプセルコーティング Download PDF

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JP2022525926A
JP2022525926A JP2021556484A JP2021556484A JP2022525926A JP 2022525926 A JP2022525926 A JP 2022525926A JP 2021556484 A JP2021556484 A JP 2021556484A JP 2021556484 A JP2021556484 A JP 2021556484A JP 2022525926 A JP2022525926 A JP 2022525926A
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gastric retention
coating
retention system
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Japanese (ja)
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JP2022525926A5 (enExample
Inventor
ビース ヌプラ
オルトルーター デイビッド
ピーク エリック
シュワルツ マーリーン
ビショフ ミーガン
ホラー ソニア
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リンドラ セラピューティクス， インコーポレイティド
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Publication of JP2022525926A publication Critical patent/JP2022525926A/ja
Publication of JP2022525926A5 publication Critical patent/JP2022525926A5/ja
Priority to JP2025005892A priority Critical patent/JP2025066761A/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4891—Coated capsules; Multilayered drug free capsule shells
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
    • A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
    • A61J3/005—Coating of tablets or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
    • A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
    • A61J3/07—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms into the form of capsules or similar small containers for oral use
    • A61J3/071—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms into the form of capsules or similar small containers for oral use into the form of telescopically engaged two-piece capsules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/485—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)
JP2021556484A 2019-03-20 2020-03-19 胃内滞留剤形用のカプセル及びカプセルコーティング Pending JP2022525926A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025005892A JP2025066761A (ja) 2019-03-20 2025-01-16 胃内滞留剤形用のカプセル及びカプセルコーティング

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962821352P 2019-03-20 2019-03-20
US62/821,352 2019-03-20
PCT/US2020/023704 WO2020191229A1 (en) 2019-03-20 2020-03-19 Capsules and capsule coatings for gastric residence dosage forms

Related Child Applications (1)

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JP2025005892A Division JP2025066761A (ja) 2019-03-20 2025-01-16 胃内滞留剤形用のカプセル及びカプセルコーティング

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JP2022525926A true JP2022525926A (ja) 2022-05-20
JP2022525926A5 JP2022525926A5 (enExample) 2024-07-31

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JP2021556484A Pending JP2022525926A (ja) 2019-03-20 2020-03-19 胃内滞留剤形用のカプセル及びカプセルコーティング
JP2025005892A Pending JP2025066761A (ja) 2019-03-20 2025-01-16 胃内滞留剤形用のカプセル及びカプセルコーティング

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US (2) US12447130B2 (enExample)
EP (1) EP3941445A4 (enExample)
JP (2) JP2022525926A (enExample)
CN (2) CN119033720A (enExample)
AU (1) AU2020240108B2 (enExample)
BR (1) BR112021018496A2 (enExample)
CA (1) CA3134049A1 (enExample)
IL (1) IL286512B2 (enExample)
MX (2) MX2021011314A (enExample)
WO (1) WO2020191229A1 (enExample)

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WO2020117855A1 (en) 2018-12-03 2020-06-11 Lyndra, Inc. Stomach simulating device
BR112021018496A2 (pt) 2019-03-20 2021-11-30 Lyndra Therapeutics Inc Cápsulas e revestimento de cápsula para formas de dosagem de residência gástrica
AU2020242062B2 (en) 2019-03-20 2025-12-11 Nortiva Bio, Inc. Coatings for gastric residence dosage forms
JP7847119B2 (ja) 2020-07-29 2026-04-16 ザ・セカント・グループ・エルエルシー 架橋ポリ（セバシン酸グリセロール）を含む構造を含む形状誘導型制御放出および保持
CN120091832A (zh) * 2022-08-03 2025-06-03 林德拉治疗公司 用于胃驻留系统的金属芯部

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JP2012510987A (ja) * 2008-12-04 2012-05-17 インテック ファーマ リミテッド ザレプロン胃内滞留性薬剤送達システム
WO2011048494A2 (en) * 2009-10-19 2011-04-28 Intec Pharma Ltd. Novel gastroretentive dosage forms of poorly soluble drugs
JP2017518308A (ja) * 2014-06-02 2017-07-06 テバ ファーマシューティカル インダストリーズ リミティド 膨張性胃内滞留型剤形
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Publication number Publication date
CA3134049A1 (en) 2020-09-24
CN119033720A (zh) 2024-11-29
IL286512B1 (en) 2025-11-01
EP3941445A1 (en) 2022-01-26
IL286512B2 (en) 2026-03-01
US20250332111A1 (en) 2025-10-30
AU2020240108B2 (en) 2025-12-04
MX2021011314A (es) 2021-12-10
EP3941445A4 (en) 2023-08-02
WO2020191229A1 (en) 2020-09-24
BR112021018496A2 (pt) 2021-11-30
US12447130B2 (en) 2025-10-21
IL286512A (en) 2021-10-31
CN113966216A (zh) 2022-01-21
AU2020240108A1 (en) 2021-11-11
US20220160642A1 (en) 2022-05-26
MX2025012985A (es) 2025-12-01
JP2025066761A (ja) 2025-04-23

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