JP2022509965A5 - - Google Patents

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Publication number
JP2022509965A5
JP2022509965A5 JP2021529329A JP2021529329A JP2022509965A5 JP 2022509965 A5 JP2022509965 A5 JP 2022509965A5 JP 2021529329 A JP2021529329 A JP 2021529329A JP 2021529329 A JP2021529329 A JP 2021529329A JP 2022509965 A5 JP2022509965 A5 JP 2022509965A5
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JP
Japan
Prior art keywords
methyl
acid
inden
dihydro
chloro
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JP2021529329A
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English (en)
Japanese (ja)
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JP2022509965A (ja
JP7583719B2 (ja
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Priority claimed from PCT/EP2019/082715 external-priority patent/WO2020114853A1/en
Publication of JP2022509965A publication Critical patent/JP2022509965A/ja
Publication of JP2022509965A5 publication Critical patent/JP2022509965A5/ja
Application granted granted Critical
Publication of JP7583719B2 publication Critical patent/JP7583719B2/ja
Active legal-status Critical Current
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JP2021529329A 2018-12-03 2019-11-27 4-((1R,3S)-6-クロロ-3-フェニル-2,3-ジヒドロ-1H-インデン-1-イル)-1,2,2-トリメチルピペラジン及び4-((1R,3S)-6-クロロ-3-(フェニル-d5)-2,3-ジヒドロ-1H-インデン-1-イル)-2,2-ジメチル-1-(メチル-d3)ピペラジンのプロドラッグ Active JP7583719B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA201800947 2018-12-03
DKPA201800947 2018-12-03
PCT/EP2019/082715 WO2020114853A1 (en) 2018-12-03 2019-11-27 Prodrugs of 4-((1r,3s)-6-chloro-3-phenyl-2,3-dihydro-1h-inden-1-yl)-1,2,2-trimethylpiperazine and 4-((1/r,3s)-6-chloro-3-(phenyl-d5)-2,3-dihydro-1h-inden-1-yl)-2,2-dimethy-1-(methyl-d3)piperazine

Publications (3)

Publication Number Publication Date
JP2022509965A JP2022509965A (ja) 2022-01-25
JP2022509965A5 true JP2022509965A5 (https=) 2022-12-02
JP7583719B2 JP7583719B2 (ja) 2024-11-14

Family

ID=69061245

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021529329A Active JP7583719B2 (ja) 2018-12-03 2019-11-27 4-((1R,3S)-6-クロロ-3-フェニル-2,3-ジヒドロ-1H-インデン-1-イル)-1,2,2-トリメチルピペラジン及び4-((1R,3S)-6-クロロ-3-(フェニル-d5)-2,3-ジヒドロ-1H-インデン-1-イル)-2,2-ジメチル-1-(メチル-d3)ピペラジンのプロドラッグ

Country Status (5)

Country Link
US (2) US11535600B2 (https=)
EP (1) EP3891134A1 (https=)
JP (1) JP7583719B2 (https=)
CN (1) CN113056457B (https=)
WO (1) WO2020114853A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020114853A1 (en) 2018-12-03 2020-06-11 H. Lundbeck A/S Prodrugs of 4-((1r,3s)-6-chloro-3-phenyl-2,3-dihydro-1h-inden-1-yl)-1,2,2-trimethylpiperazine and 4-((1/r,3s)-6-chloro-3-(phenyl-d5)-2,3-dihydro-1h-inden-1-yl)-2,2-dimethy-1-(methyl-d3)piperazine

Family Cites Families (44)

* Cited by examiner, † Cited by third party
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WO2020089147A1 (en) 2018-10-29 2020-05-07 H. Lundbeck A/S Amorphous compounds of formula (i) and amorphous compounds of formula (i) salts
WO2020114853A1 (en) 2018-12-03 2020-06-11 H. Lundbeck A/S Prodrugs of 4-((1r,3s)-6-chloro-3-phenyl-2,3-dihydro-1h-inden-1-yl)-1,2,2-trimethylpiperazine and 4-((1/r,3s)-6-chloro-3-(phenyl-d5)-2,3-dihydro-1h-inden-1-yl)-2,2-dimethy-1-(methyl-d3)piperazine

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