JP2022502393A5 - - Google Patents

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Publication number
JP2022502393A5
JP2022502393A5 JP2021516806A JP2021516806A JP2022502393A5 JP 2022502393 A5 JP2022502393 A5 JP 2022502393A5 JP 2021516806 A JP2021516806 A JP 2021516806A JP 2021516806 A JP2021516806 A JP 2021516806A JP 2022502393 A5 JP2022502393 A5 JP 2022502393A5
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JP
Japan
Prior art keywords
compound
methyl
formula
pyran
tetrahydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021516806A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022502393A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/052414 external-priority patent/WO2020068661A1/en
Publication of JP2022502393A publication Critical patent/JP2022502393A/ja
Publication of JP2022502393A5 publication Critical patent/JP2022502393A5/ja
Pending legal-status Critical Current

Links

JP2021516806A 2018-09-26 2019-09-23 Ｎ−（１−（（２−（ジメチルアミノ）エチル）アミノ）−２−メチル−１−オキソプロパン−２−イル）−４−（４−（２−メチル−５−（（２ｓ，３ｒ，４ｒ，５ｓ，６ｒ）−３，４，５−トリヒドロキシ−６−（メチルチオ）テトラヒドロ−２ｈ−ピラン−２−イル）ベンジル）フェニル）ブタンアミドの結晶形態及びそれらの合成方法 Pending JP2022502393A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862736871P 2018-09-26 2018-09-26
US62/736,871 2018-09-26
PCT/US2019/052414 WO2020068661A1 (en) 2018-09-26 2019-09-23 Crystalline forms of n-(1 -((2-(dimethylamino)ethyl)amino)-2-m ethyl-1 -oopropan-2-yl)-4-(4-(2-methyl-5- (2s,3r,4r,5s,6r)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2h-pyran-2-yl)benzyl) phenl)butanamide and methods of their synthesis

Publications (2)

Publication Number Publication Date
JP2022502393A JP2022502393A (ja) 2022-01-11
JP2022502393A5 true JP2022502393A5 (enExample) 2022-03-07

Family

ID=68165724

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021516806A Pending JP2022502393A (ja) 2018-09-26 2019-09-23 Ｎ−（１−（（２−（ジメチルアミノ）エチル）アミノ）−２−メチル−１−オキソプロパン−２−イル）−４−（４−（２−メチル−５−（（２ｓ，３ｒ，４ｒ，５ｓ，６ｒ）−３，４，５−トリヒドロキシ−６−（メチルチオ）テトラヒドロ−２ｈ−ピラン−２−イル）ベンジル）フェニル）ブタンアミドの結晶形態及びそれらの合成方法

Country Status (13)

Country Link
US (1) US10968192B2 (enExample)
EP (1) EP3856714A1 (enExample)
JP (1) JP2022502393A (enExample)
KR (1) KR20210065974A (enExample)
CN (1) CN113039176A (enExample)
AU (1) AU2019346497A1 (enExample)
BR (1) BR112021004839A2 (enExample)
CA (1) CA3113037A1 (enExample)
CO (1) CO2021005141A2 (enExample)
IL (1) IL281728A (enExample)
MX (1) MX2021003545A (enExample)
SG (1) SG11202102498UA (enExample)
WO (1) WO2020068661A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114599643B (zh) * 2020-05-15 2023-04-14 上海喆邺生物科技有限公司 一种芳基葡糖苷衍生物
EP4119550B1 (en) * 2020-05-15 2025-08-20 Shanghai Zheye Biotechnology Co., Ltd. Aryl glucoside derivative and use thereof in drug
CN117018204A (zh) * 2020-07-06 2023-11-10 诺未科技（北京）有限公司 一种治疗癌症的组合物及其应用和药物
US20250170157A1 (en) 2023-11-10 2025-05-29 Lexicon Pharmaceuticals, Inc. Methods and compositions for the treatment of hepatic encephalopathy

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