JP2022500416A - がんを処置するためのキットおよび方法 - Google Patents

がんを処置するためのキットおよび方法 Download PDF

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JP2022500416A
JP2022500416A JP2021513941A JP2021513941A JP2022500416A JP 2022500416 A JP2022500416 A JP 2022500416A JP 2021513941 A JP2021513941 A JP 2021513941A JP 2021513941 A JP2021513941 A JP 2021513941A JP 2022500416 A JP2022500416 A JP 2022500416A
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compound
kit
cancer
crystal
peak
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レディー,グル
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スペクトラム ファーマシューティカルズ インコーポレイテッド
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/47Quinolines; Isoquinolines
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    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
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    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
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    • A61K31/7068Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
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    • A61K31/7072Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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JP2021513941A 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法 Pending JP2022500416A (ja)

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US201862731500P 2018-09-14 2018-09-14
US62/731,500 2018-09-14
PCT/US2019/050843 WO2020056156A1 (en) 2018-09-14 2019-09-12 Kits and methods for treating cancers

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JP2021513941A Pending JP2022500416A (ja) 2018-09-14 2019-09-12 がんを処置するためのキットおよび方法
JP2021514419A Active JP7554030B2 (ja) 2018-09-14 2019-09-12 キナゾリン化合物及びその塩酸塩の結晶形

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US (2) US20220040180A1 (https=)
EP (2) EP3849557A4 (https=)
JP (2) JP2022500416A (https=)
KR (2) KR102802129B1 (https=)
CN (2) CN112770758A (https=)
AR (2) AR116669A1 (https=)
AU (2) AU2019337640A1 (https=)
BR (2) BR112021004527A2 (https=)
CA (2) CA3110369A1 (https=)
IL (2) IL281168A (https=)
MX (2) MX2021002875A (https=)
PH (2) PH12021550432A1 (https=)
PY (2) PY1976960A (https=)
SG (2) SG11202102006YA (https=)
TW (2) TW202027750A (https=)
UY (2) UY38374A (https=)
WO (2) WO2020056156A1 (https=)

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BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer
JP2023503318A (ja) 2019-11-21 2023-01-27 ファルマ、マール、ソシエダード、アノニマ ルルビネクテジン製剤で小細胞肺がんを処置する方法
CN114642728A (zh) * 2021-06-02 2022-06-21 德琪(浙江)医药科技有限公司 mTOR抑制剂的制药用途及其药物组合物

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BR112021004527A2 (pt) 2018-09-14 2021-06-08 Spectrum Pharmaceuticals, Inc. kits e métodos para tratamento contra câncer

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MX2021002876A (es) 2021-06-04
TW202027750A (zh) 2020-08-01
US20220056011A1 (en) 2022-02-24
AR116406A1 (es) 2021-05-05
TW202023562A (zh) 2020-07-01
BR112021004527A2 (pt) 2021-06-08
WO2020053816A1 (en) 2020-03-19
US20220040180A1 (en) 2022-02-10
AU2019337640A1 (en) 2021-03-11
CA3110369A1 (en) 2020-03-19
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AU2019340598A1 (en) 2021-03-18
IL281167A (en) 2021-04-29
SG11202102006YA (en) 2021-04-29
BR112021004546A2 (pt) 2021-06-08
UY38375A (es) 2020-04-30
WO2020056156A1 (en) 2020-03-19
EP3849557A1 (en) 2021-07-21
CN112823153A (zh) 2021-05-18
KR20210061371A (ko) 2021-05-27
IL281168A (en) 2021-04-29
PY1976957A (es) 2022-02-24
JP2022500456A (ja) 2022-01-04
EP3849557A4 (en) 2022-06-08
KR102802129B1 (ko) 2025-05-02
KR20210046818A (ko) 2021-04-28
JP7554030B2 (ja) 2024-09-19
MX2021002875A (es) 2021-07-15
PY1976960A (es) 2020-06-15
AR116669A1 (es) 2021-06-02
AU2019340598B2 (en) 2024-08-29
EP3849964A1 (en) 2021-07-21
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US11883402B2 (en) 2024-01-30
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