JP2021533143A5 - - Google Patents
Info
- Publication number
- JP2021533143A5 JP2021533143A5 JP2021505964A JP2021505964A JP2021533143A5 JP 2021533143 A5 JP2021533143 A5 JP 2021533143A5 JP 2021505964 A JP2021505964 A JP 2021505964A JP 2021505964 A JP2021505964 A JP 2021505964A JP 2021533143 A5 JP2021533143 A5 JP 2021533143A5
- Authority
- JP
- Japan
- Prior art keywords
- unsubstituted
- substituted
- substituents
- alkyl
- pyrazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2018128415A RU2761824C2 (ru) | 2018-08-03 | 2018-08-03 | Ингибиторы CDK8/19 |
| RU2018128415 | 2018-08-03 | ||
| PCT/RU2019/050123 WO2020027704A1 (ru) | 2018-08-03 | 2019-07-31 | Ингибиторы cdk8/19 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021533143A JP2021533143A (ja) | 2021-12-02 |
| JP2021533143A5 true JP2021533143A5 (https=) | 2022-08-09 |
| JP7365396B2 JP7365396B2 (ja) | 2023-10-19 |
Family
ID=69231230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021505964A Active JP7365396B2 (ja) | 2018-08-03 | 2019-07-31 | Cdk8/19阻害薬 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US11840531B2 (https=) |
| EP (1) | EP3831829A4 (https=) |
| JP (1) | JP7365396B2 (https=) |
| KR (1) | KR102926889B1 (https=) |
| CN (1) | CN113166140B (https=) |
| AR (1) | AR115898A1 (https=) |
| AU (1) | AU2019313199B2 (https=) |
| BR (1) | BR112021001939A2 (https=) |
| CA (1) | CA3108298A1 (https=) |
| CL (1) | CL2021000282A1 (https=) |
| CO (1) | CO2021001174A2 (https=) |
| EA (1) | EA202190452A1 (https=) |
| MA (1) | MA52375B2 (https=) |
| MX (1) | MX2021001335A (https=) |
| PE (1) | PE20210416A1 (https=) |
| PH (1) | PH12021550258A1 (https=) |
| RU (1) | RU2761824C2 (https=) |
| TW (1) | TWI839374B (https=) |
| WO (1) | WO2020027704A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023533016A (ja) | 2020-07-11 | 2023-08-01 | ファイザー・インク | 抗ウイルス性ヘテロアリールケトン誘導体 |
| US11351149B2 (en) | 2020-09-03 | 2022-06-07 | Pfizer Inc. | Nitrile-containing antiviral compounds |
| WO2024109660A1 (zh) * | 2022-11-21 | 2024-05-30 | 上海齐鲁制药研究中心有限公司 | Cdk抑制剂 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR060358A1 (es) * | 2006-04-06 | 2008-06-11 | Novartis Vaccines & Diagnostic | Quinazolinas para la inhibicion de pdk 1 |
| MX2010006244A (es) * | 2007-12-06 | 2010-12-02 | Schering Corp | Moduladores de gamma secretasa. |
| CN103249721B (zh) * | 2010-10-18 | 2016-10-12 | 拉夸里亚创药株式会社 | 作为ttx-s阻滞剂的芳胺衍生物 |
| TWI529171B (zh) * | 2013-07-29 | 2016-04-11 | 赫孚孟拉羅股份公司 | 1,7-萘啶衍生物 |
| JP2017522324A (ja) | 2014-07-17 | 2017-08-10 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung | 新規ナフチリジン及びイソキノリンならびにcdk8/19阻害剤としてのその使用 |
| EP3383875B1 (en) * | 2015-11-30 | 2022-02-09 | Council Of Scientific & Industrial Research | 3-pyrimidinyl pyrrolo [2,3-b] pyridine as anticancer agents and the process for the preparation thereof |
| US11213520B2 (en) * | 2016-05-23 | 2022-01-04 | Boehringer Ingelheim International Gmbh | Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors |
-
2018
- 2018-08-03 RU RU2018128415A patent/RU2761824C2/ru active
-
2019
- 2019-07-31 MA MA52375A patent/MA52375B2/fr unknown
- 2019-07-31 PE PE2021000162A patent/PE20210416A1/es unknown
- 2019-07-31 US US17/264,670 patent/US11840531B2/en active Active
- 2019-07-31 MX MX2021001335A patent/MX2021001335A/es unknown
- 2019-07-31 AU AU2019313199A patent/AU2019313199B2/en active Active
- 2019-07-31 WO PCT/RU2019/050123 patent/WO2020027704A1/ru not_active Ceased
- 2019-07-31 KR KR1020217006527A patent/KR102926889B1/ko active Active
- 2019-07-31 EP EP19844331.9A patent/EP3831829A4/en active Pending
- 2019-07-31 JP JP2021505964A patent/JP7365396B2/ja active Active
- 2019-07-31 CA CA3108298A patent/CA3108298A1/en active Pending
- 2019-07-31 CN CN201980065665.1A patent/CN113166140B/zh active Active
- 2019-07-31 BR BR112021001939-1A patent/BR112021001939A2/pt unknown
- 2019-07-31 EA EA202190452A patent/EA202190452A1/ru unknown
- 2019-08-02 TW TW108127569A patent/TWI839374B/zh active
- 2019-08-02 AR ARP190102200A patent/AR115898A1/es unknown
-
2021
- 2021-02-02 CL CL2021000282A patent/CL2021000282A1/es unknown
- 2021-02-02 CO CONC2021/0001174A patent/CO2021001174A2/es unknown
- 2021-02-03 PH PH12021550258A patent/PH12021550258A1/en unknown
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