JP2021533143A5 - - Google Patents

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Publication number
JP2021533143A5
JP2021533143A5 JP2021505964A JP2021505964A JP2021533143A5 JP 2021533143 A5 JP2021533143 A5 JP 2021533143A5 JP 2021505964 A JP2021505964 A JP 2021505964A JP 2021505964 A JP2021505964 A JP 2021505964A JP 2021533143 A5 JP2021533143 A5 JP 2021533143A5
Authority
JP
Japan
Prior art keywords
unsubstituted
substituted
substituents
alkyl
pyrazole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021505964A
Other languages
English (en)
Japanese (ja)
Other versions
JP7365396B2 (ja
JP2021533143A (ja
Filing date
Publication date
Priority claimed from RU2018128415A external-priority patent/RU2761824C2/ru
Application filed filed Critical
Publication of JP2021533143A publication Critical patent/JP2021533143A/ja
Publication of JP2021533143A5 publication Critical patent/JP2021533143A5/ja
Application granted granted Critical
Publication of JP7365396B2 publication Critical patent/JP7365396B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021505964A 2018-08-03 2019-07-31 Cdk8/19阻害薬 Active JP7365396B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
RU2018128415A RU2761824C2 (ru) 2018-08-03 2018-08-03 Ингибиторы CDK8/19
RU2018128415 2018-08-03
PCT/RU2019/050123 WO2020027704A1 (ru) 2018-08-03 2019-07-31 Ингибиторы cdk8/19

Publications (3)

Publication Number Publication Date
JP2021533143A JP2021533143A (ja) 2021-12-02
JP2021533143A5 true JP2021533143A5 (https=) 2022-08-09
JP7365396B2 JP7365396B2 (ja) 2023-10-19

Family

ID=69231230

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021505964A Active JP7365396B2 (ja) 2018-08-03 2019-07-31 Cdk8/19阻害薬

Country Status (19)

Country Link
US (1) US11840531B2 (https=)
EP (1) EP3831829A4 (https=)
JP (1) JP7365396B2 (https=)
KR (1) KR102926889B1 (https=)
CN (1) CN113166140B (https=)
AR (1) AR115898A1 (https=)
AU (1) AU2019313199B2 (https=)
BR (1) BR112021001939A2 (https=)
CA (1) CA3108298A1 (https=)
CL (1) CL2021000282A1 (https=)
CO (1) CO2021001174A2 (https=)
EA (1) EA202190452A1 (https=)
MA (1) MA52375B2 (https=)
MX (1) MX2021001335A (https=)
PE (1) PE20210416A1 (https=)
PH (1) PH12021550258A1 (https=)
RU (1) RU2761824C2 (https=)
TW (1) TWI839374B (https=)
WO (1) WO2020027704A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023533016A (ja) 2020-07-11 2023-08-01 ファイザー・インク 抗ウイルス性ヘテロアリールケトン誘導体
US11351149B2 (en) 2020-09-03 2022-06-07 Pfizer Inc. Nitrile-containing antiviral compounds
WO2024109660A1 (zh) * 2022-11-21 2024-05-30 上海齐鲁制药研究中心有限公司 Cdk抑制剂

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR060358A1 (es) * 2006-04-06 2008-06-11 Novartis Vaccines & Diagnostic Quinazolinas para la inhibicion de pdk 1
MX2010006244A (es) * 2007-12-06 2010-12-02 Schering Corp Moduladores de gamma secretasa.
CN103249721B (zh) * 2010-10-18 2016-10-12 拉夸里亚创药株式会社 作为ttx-s阻滞剂的芳胺衍生物
TWI529171B (zh) * 2013-07-29 2016-04-11 赫孚孟拉羅股份公司 1,7-萘啶衍生物
JP2017522324A (ja) 2014-07-17 2017-08-10 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung 新規ナフチリジン及びイソキノリンならびにcdk8/19阻害剤としてのその使用
EP3383875B1 (en) * 2015-11-30 2022-02-09 Council Of Scientific & Industrial Research 3-pyrimidinyl pyrrolo [2,3-b] pyridine as anticancer agents and the process for the preparation thereof
US11213520B2 (en) * 2016-05-23 2022-01-04 Boehringer Ingelheim International Gmbh Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors

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