JP2021529752A5 - - Google Patents

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Publication number
JP2021529752A5
JP2021529752A5 JP2020572891A JP2020572891A JP2021529752A5 JP 2021529752 A5 JP2021529752 A5 JP 2021529752A5 JP 2020572891 A JP2020572891 A JP 2020572891A JP 2020572891 A JP2020572891 A JP 2020572891A JP 2021529752 A5 JP2021529752 A5 JP 2021529752A5
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JP
Japan
Prior art keywords
alkyl
alkoxy
group
heteroaryl
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020572891A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021529752A (ja
JP7396682B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/040121 external-priority patent/WO2020006557A1/en
Publication of JP2021529752A publication Critical patent/JP2021529752A/ja
Publication of JP2021529752A5 publication Critical patent/JP2021529752A5/ja
Application granted granted Critical
Publication of JP7396682B2 publication Critical patent/JP7396682B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020572891A 2018-06-29 2019-07-01 イタコン酸誘導体の組成物及び使用方法 Active JP7396682B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862763735P 2018-06-29 2018-06-29
US62/763,735 2018-06-29
PCT/US2019/040121 WO2020006557A1 (en) 2018-06-29 2019-07-01 Compositions and methods of using itaconic acid derivatives

Publications (3)

Publication Number Publication Date
JP2021529752A JP2021529752A (ja) 2021-11-04
JP2021529752A5 true JP2021529752A5 (https=) 2022-06-21
JP7396682B2 JP7396682B2 (ja) 2023-12-12

Family

ID=68985877

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020572891A Active JP7396682B2 (ja) 2018-06-29 2019-07-01 イタコン酸誘導体の組成物及び使用方法

Country Status (5)

Country Link
US (1) US12060310B2 (https=)
EP (1) EP3813815B1 (https=)
JP (1) JP7396682B2 (https=)
ES (1) ES3063485T3 (https=)
WO (1) WO2020006557A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2021013299A (es) 2019-04-30 2022-01-31 Sitryx Therapeutics Ltd Derivados de acido itaconico y usos de estos en el tratamiento de una enfermedad inflamatoria asociada con una respuesta inmunitaria indeseable.
EP4237404A1 (en) * 2020-10-29 2023-09-06 Sitryx Therapeutics Limited Novel compounds
WO2022223778A1 (en) 2021-04-23 2022-10-27 Helmholtz-Zentrum für Infektionsforschung GmbH Citraconic acid and derivatives thereof for use as a medicament
CN119685257B (zh) * 2024-12-16 2026-02-27 华中科技大学同济医学院附属协和医院 体外诱导t细胞免疫记忆分化的方法及应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260479A (en) 1991-12-16 1993-11-09 Merck & Co., Inc. Inhibitors of farnesyl protein transferase
EP1062954B1 (en) * 1998-10-27 2007-05-30 Suntory Limited Use of itaconic acid for regulation of glycolytic metabolism
US8293925B2 (en) 2009-09-21 2012-10-23 Chemocentryx, Inc. Pyrrolidinone carboxamide derivatives
LU91877B1 (en) 2011-09-23 2013-03-25 Univ Luxembourg Method to predict the presence of itaconic Acid, IRG1 and/or protein IRG1 in a subject and pharmaceutical composition for performing gene therapy
US8691993B2 (en) 2011-12-12 2014-04-08 Hoffmann-La Roche Inc. Piperidinyl naphthylacetic acids
EP2833877A4 (en) 2012-04-03 2015-11-25 Aposense Ltd NEW TARGETING AGENTS FOR DIAGNOSTIC AND THERAPEUTIC INDICATIONS
EP3416634A4 (en) 2016-02-15 2019-10-09 Artyomov, Maxim IMMUNOMODULATORY AGENTS AND METHOD FOR USE THEREOF

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