JP2021528499A5 - - Google Patents

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Publication number
JP2021528499A5
JP2021528499A5 JP2021521740A JP2021521740A JP2021528499A5 JP 2021528499 A5 JP2021528499 A5 JP 2021528499A5 JP 2021521740 A JP2021521740 A JP 2021521740A JP 2021521740 A JP2021521740 A JP 2021521740A JP 2021528499 A5 JP2021528499 A5 JP 2021528499A5
Authority
JP
Japan
Prior art keywords
group
substituted
bisphosphonate
compound
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021521740A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021528499A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/039018 external-priority patent/WO2020005964A1/en
Publication of JP2021528499A publication Critical patent/JP2021528499A/ja
Publication of JP2021528499A5 publication Critical patent/JP2021528499A5/ja
Pending legal-status Critical Current

Links

JP2021521740A 2018-06-26 2019-06-25 骨標的抗菌オキサゾリジノン関連化合物、その製剤及び用途 Pending JP2021528499A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862690053P 2018-06-26 2018-06-26
US62/690,053 2018-06-26
PCT/US2019/039018 WO2020005964A1 (en) 2018-06-26 2019-06-25 Bone targeted antimicrobial oxazolidinone related compounds, formulations thereof, and uses thereof

Publications (2)

Publication Number Publication Date
JP2021528499A JP2021528499A (ja) 2021-10-21
JP2021528499A5 true JP2021528499A5 (https=) 2022-07-05

Family

ID=68987043

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021521740A Pending JP2021528499A (ja) 2018-06-26 2019-06-25 骨標的抗菌オキサゾリジノン関連化合物、その製剤及び用途

Country Status (6)

Country Link
US (1) US12285489B2 (https=)
EP (1) EP3813840A4 (https=)
JP (1) JP2021528499A (https=)
CN (1) CN112533612A (https=)
CA (1) CA3105042A1 (https=)
WO (1) WO2020005964A1 (https=)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8586781B2 (en) 1998-04-02 2013-11-19 Mbc Pharma, Inc. Bone targeted therapeutics and methods of making and using the same
TW200410701A (en) * 2002-10-15 2004-07-01 Novartis Ag Method of administering bisphosphonates
EP1881974A4 (en) * 2005-04-21 2011-03-16 Targanta Therapeutics Inc PHOSPHONE FLUOROQUINOLONES, THEIR ANTIBACTERIAL ANALOGUES, AND METHODS FOR PREVENTING AND TREATING BONE AND JOINT INFECTIONS
WO2007138381A2 (en) 2005-10-14 2007-12-06 Targanta Therapeutics Inc. Phosphonated oxazolidinones and uses thereof for the prevention and treatment of bone and joint infections
EP2213315A1 (en) * 2009-01-30 2010-08-04 Mero S.r.L. Antibacterial hydrogel and use thereof in orthopedics
US20110124597A1 (en) * 2009-09-25 2011-05-26 Anacor Pharmaceuticals, Inc. Boron containing small molecules
WO2017210611A1 (en) * 2016-06-03 2017-12-07 Biovinc, Llc. Bisphosphonate quinolone conjugates and uses thereof
CA3105829A1 (en) * 2018-07-09 2020-01-16 Biovinc, Llc. Bisphosphonate quinolone conjugates and uses thereof

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