JP2021532087A5 - - Google Patents

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Publication number
JP2021532087A5
JP2021532087A5 JP2021500846A JP2021500846A JP2021532087A5 JP 2021532087 A5 JP2021532087 A5 JP 2021532087A5 JP 2021500846 A JP2021500846 A JP 2021500846A JP 2021500846 A JP2021500846 A JP 2021500846A JP 2021532087 A5 JP2021532087 A5 JP 2021532087A5
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JP
Japan
Prior art keywords
linker
compound according
compound
bone
quinolone
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Granted
Application number
JP2021500846A
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English (en)
Japanese (ja)
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JP2021532087A (ja
JP7501960B2 (ja
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Priority claimed from PCT/US2019/041063 external-priority patent/WO2020014269A1/en
Publication of JP2021532087A publication Critical patent/JP2021532087A/ja
Publication of JP2021532087A5 publication Critical patent/JP2021532087A5/ja
Application granted granted Critical
Publication of JP7501960B2 publication Critical patent/JP7501960B2/ja
Active legal-status Critical Current
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JP2021500846A 2018-07-09 2019-07-09 ビスホスホネート・キノロン複合体及びそれらの用途 Active JP7501960B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862695583P 2018-07-09 2018-07-09
US62/695,583 2018-07-09
PCT/US2019/041063 WO2020014269A1 (en) 2018-07-09 2019-07-09 Bisphosphonate quinolone conjugates and uses thereof

Publications (3)

Publication Number Publication Date
JP2021532087A JP2021532087A (ja) 2021-11-25
JP2021532087A5 true JP2021532087A5 (https=) 2022-06-10
JP7501960B2 JP7501960B2 (ja) 2024-06-18

Family

ID=69142455

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021500846A Active JP7501960B2 (ja) 2018-07-09 2019-07-09 ビスホスホネート・キノロン複合体及びそれらの用途

Country Status (5)

Country Link
EP (1) EP3820565A4 (https=)
JP (1) JP7501960B2 (https=)
CN (1) CN112672787A (https=)
CA (1) CA3105829A1 (https=)
WO (1) WO2020014269A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12285489B2 (en) * 2018-06-26 2025-04-29 Frank Hallock Ebetino Bone targeted antimicrobial oxazolidinone related compounds, formulations thereof, and uses thereof
WO2025019691A1 (en) * 2023-07-19 2025-01-23 Zymeron Corporation Drug conjugates for bone marrow protection

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5087240A (en) 1983-08-18 1992-02-11 Drug Delivery Systems Inc. Transdermal drug patch with conductive fibers
US4921475A (en) 1983-08-18 1990-05-01 Drug Delivery Systems Inc. Transdermal drug patch with microtubes
US5163899A (en) 1987-03-20 1992-11-17 Drug Delivery Systems Inc. Transdermal drug delivery system
US5312325A (en) 1987-05-28 1994-05-17 Drug Delivery Systems Inc Pulsating transdermal drug delivery system
GB8804164D0 (en) 1988-02-23 1988-03-23 Tucker J M Bandage for administering physiologically active compound
US5008110A (en) 1988-11-10 1991-04-16 The Procter & Gamble Company Storage-stable transdermal patch
US5088977A (en) 1988-12-21 1992-02-18 Drug Delivery Systems Inc. Electrical transdermal drug applicator with counteractor and method of drug delivery
DK0431519T3 (da) 1989-12-04 1994-07-04 Searle & Co System til transdermal indgivelse af albuterol
US5352456A (en) 1991-10-10 1994-10-04 Cygnus Therapeutic Systems Device for administering drug transdermally which provides an initial pulse of drug
DE69228827T2 (de) 1991-12-18 1999-10-21 Minnesota Mining And Mfg. Co., Saint Paul Mehrschichtige sperrstrukturen
ATE132381T1 (de) 1992-01-29 1996-01-15 Voelkl Franz Ski Ballspielschläger, insbesondere tennisschläger
US6333424B1 (en) * 1996-10-09 2001-12-25 Eliza Nor Biopharmaceuticals, Inc. Therapeutic derivatives of diphosphonates
EP1881974A4 (en) * 2005-04-21 2011-03-16 Targanta Therapeutics Inc PHOSPHONE FLUOROQUINOLONES, THEIR ANTIBACTERIAL ANALOGUES, AND METHODS FOR PREVENTING AND TREATING BONE AND JOINT INFECTIONS
EP1928890B1 (en) * 2005-08-11 2013-04-03 Targanta Therapeutics Inc. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
WO2007138381A2 (en) 2005-10-14 2007-12-06 Targanta Therapeutics Inc. Phosphonated oxazolidinones and uses thereof for the prevention and treatment of bone and joint infections

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