JP2021525738A5 - - Google Patents

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Publication number
JP2021525738A5
JP2021525738A5 JP2020566706A JP2020566706A JP2021525738A5 JP 2021525738 A5 JP2021525738 A5 JP 2021525738A5 JP 2020566706 A JP2020566706 A JP 2020566706A JP 2020566706 A JP2020566706 A JP 2020566706A JP 2021525738 A5 JP2021525738 A5 JP 2021525738A5
Authority
JP
Japan
Prior art keywords
imidazo
pyrazine
pyrido
bromo
methylpiperazine
Prior art date
Application number
JP2020566706A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2019231270A5 (https=
JP2021525738A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/KR2019/006553 external-priority patent/WO2019231270A1/en
Publication of JP2021525738A publication Critical patent/JP2021525738A/ja
Publication of JPWO2019231270A5 publication Critical patent/JPWO2019231270A5/ja
Publication of JP2021525738A5 publication Critical patent/JP2021525738A5/ja
Withdrawn legal-status Critical Current

Links

JP2020566706A 2018-05-31 2019-05-31 複素環誘導体及びその使用 Withdrawn JP2021525738A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20180062254 2018-05-31
KR10-2018-0062254 2018-05-31
PCT/KR2019/006553 WO2019231270A1 (en) 2018-05-31 2019-05-31 Heterocyclic derivatives and use thereof

Publications (3)

Publication Number Publication Date
JP2021525738A JP2021525738A (ja) 2021-09-27
JPWO2019231270A5 JPWO2019231270A5 (https=) 2022-04-04
JP2021525738A5 true JP2021525738A5 (https=) 2022-04-04

Family

ID=68698381

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020566706A Withdrawn JP2021525738A (ja) 2018-05-31 2019-05-31 複素環誘導体及びその使用

Country Status (12)

Country Link
US (1) US20210198259A1 (https=)
EP (1) EP3807282A4 (https=)
JP (1) JP2021525738A (https=)
KR (1) KR102344295B1 (https=)
CN (1) CN112204032A (https=)
AU (1) AU2019279421A1 (https=)
BR (1) BR112020023946A2 (https=)
CA (1) CA3098825A1 (https=)
MX (1) MX2020011955A (https=)
SG (1) SG11202010985TA (https=)
TW (1) TW202021969A (https=)
WO (1) WO2019231270A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20230107927A1 (en) 2020-02-28 2023-04-06 First Wave Bio, Inc. Methods of treating iatrogenic autoimmune colitis
IL298760A (en) 2020-06-05 2023-02-01 Kinnate Biopharma Inc Fibroblast growth factor receptor kinase inhibitors
EP4067357A1 (en) * 2021-03-30 2022-10-05 JW Pharmaceutical Corporation Novel crystalline form of 1-(8-bromopyrido[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-4-yl)-n-methylazetidin-3-amine hydrogen sulfate monohydrate
CN113929634A (zh) * 2021-11-22 2022-01-14 山西永津集团有限公司 一种2,3-二溴喹喔啉的合成方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE358395B (https=) * 1967-09-27 1973-07-30 Siegfried Ag
BRPI0407926A (pt) * 2003-03-27 2006-02-21 Pfizer Prod Inc 4-amino[1,2,4]triazol[4,3-a]quinoxalinas substituìdas
TW201024297A (en) * 2008-09-10 2010-07-01 Kalypsys Inc Heterocyclic inhibitors of histamine receptors for the treatment of disease
TW201204727A (en) * 2010-03-10 2012-02-01 Kalypsys Inc Heterocyclic inhibitors of histamine receptors for the treatment of disease
TW201206936A (en) * 2010-07-19 2012-02-16 Alcon Res Ltd Methods and compositions for the treatment of allergy
TWI551600B (zh) * 2011-09-30 2016-10-01 C&C新藥研究所 新穎雜環衍生物及其用途
CA2904364A1 (en) * 2013-03-15 2014-09-25 Epigenetix, Inc. Oxazolo[5,4-c]quinolin-2-one compounds as bromodomain inhibitors
JP2018537450A (ja) * 2015-11-16 2018-12-20 ファンダシオン パラ ラ インベスティガシオン メディカ アプリカダFundacion Para La Investigasion Medica Aplicada Dnaメチルトランスフェラーゼ阻害剤としての新規化合物
JP7212612B2 (ja) * 2016-07-28 2023-01-25 プロメガ コーポレイション セレンテラジン類縁体

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