JP2021521132A5 - - Google Patents

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Publication number
JP2021521132A5
JP2021521132A5 JP2020555192A JP2020555192A JP2021521132A5 JP 2021521132 A5 JP2021521132 A5 JP 2021521132A5 JP 2020555192 A JP2020555192 A JP 2020555192A JP 2020555192 A JP2020555192 A JP 2020555192A JP 2021521132 A5 JP2021521132 A5 JP 2021521132A5
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JP
Japan
Prior art keywords
compound according
amino
prevention
treatment
salt
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Granted
Application number
JP2020555192A
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English (en)
Japanese (ja)
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JP2021521132A (ja
JP7333336B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2019/058398 external-priority patent/WO2019197244A1/en
Publication of JP2021521132A publication Critical patent/JP2021521132A/ja
Publication of JP2021521132A5 publication Critical patent/JP2021521132A5/ja
Application granted granted Critical
Publication of JP7333336B2 publication Critical patent/JP7333336B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020555192A 2018-04-10 2019-04-03 置換オキソピリジン誘導体 Active JP7333336B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18166490.5 2018-04-10
EP18166490 2018-04-10
PCT/EP2019/058398 WO2019197244A1 (en) 2018-04-10 2019-04-03 A substituted oxopyridine derivative

Publications (3)

Publication Number Publication Date
JP2021521132A JP2021521132A (ja) 2021-08-26
JP2021521132A5 true JP2021521132A5 (enExample) 2023-05-16
JP7333336B2 JP7333336B2 (ja) 2023-08-24

Family

ID=61965754

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020555192A Active JP7333336B2 (ja) 2018-04-10 2019-04-03 置換オキソピリジン誘導体

Country Status (17)

Country Link
US (1) US11884660B2 (enExample)
EP (1) EP3774796B1 (enExample)
JP (1) JP7333336B2 (enExample)
KR (1) KR102858566B1 (enExample)
CN (1) CN111902414B (enExample)
AU (1) AU2019251699B2 (enExample)
BR (1) BR112020018237A2 (enExample)
CA (1) CA3096480A1 (enExample)
DK (1) DK3774796T3 (enExample)
ES (1) ES2922533T3 (enExample)
IL (1) IL277811B2 (enExample)
MX (1) MX2020010635A (enExample)
PE (1) PE20210165A1 (enExample)
SA (1) SA520420308B1 (enExample)
SG (1) SG11202008352YA (enExample)
WO (1) WO2019197244A1 (enExample)
ZA (1) ZA202006963B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116874469B (zh) * 2023-09-06 2023-11-10 成都施贝康生物医药科技有限公司 一种氧代吡啶类化合物、中间体及其制备方法和用途
CN116947818B (zh) * 2023-09-18 2023-12-19 成都施贝康生物医药科技有限公司 一种氧代吡啶类化合物、中间体及其制备方法和用途

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7453002B2 (en) 2004-06-15 2008-11-18 Bristol-Myers Squibb Company Five-membered heterocycles useful as serine protease inhibitors
US7429604B2 (en) 2004-06-15 2008-09-30 Bristol Myers Squibb Company Six-membered heterocycles useful as serine protease inhibitors
GB0420722D0 (en) 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
JP5419706B2 (ja) 2006-12-20 2014-02-19 タケダ カリフォルニア インコーポレイテッド グルコキナーゼアクチベーター
US9809545B2 (en) 2013-03-27 2017-11-07 Merck Sharp & Dohme Corp. Factor XIa inhibitors
TWI633089B (zh) 2013-03-28 2018-08-21 拜耳製藥股份有限公司 經取代的酮基吡啶衍生物
US9475809B2 (en) 2013-07-23 2016-10-25 Bayer Pharma Aktiengesellschaft Substituted oxopyridine derivatives and use thereof as factor xia/plasma
WO2015063093A1 (de) 2013-10-30 2015-05-07 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
WO2015120777A1 (zh) 2014-02-14 2015-08-20 四川海思科制药有限公司 一种吡啶酮或嘧啶酮衍生物、及其制备方法和应用
WO2016046158A1 (de) 2014-09-24 2016-03-31 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
WO2016046166A1 (de) 2014-09-24 2016-03-31 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
JP6517925B2 (ja) 2014-09-24 2019-05-22 バイエル ファーマ アクチエンゲゼルシャフト 置換されたオキソピリジン誘導体
ES2716417T3 (es) 2014-09-24 2019-06-12 Bayer Pharma AG Derivados de oxopiridina sustituidos con acción antiinflamatoria y antitrombótica
WO2016046156A1 (de) 2014-09-24 2016-03-31 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
ES2712886T3 (es) 2014-09-24 2019-05-16 Bayer Pharma AG Derivados de piridobenzazepina y piridobenzazocina que inhiben el factor XIa
CA2979937A1 (en) 2015-03-19 2016-09-22 Bayer Pharma Aktiengesellschaft Oxo-pyridine-derivatives as factor xia inhibitors for the treatment of thrombosis
JO3703B1 (ar) 2015-07-09 2021-01-31 Bayer Pharma AG مشتقات أوكسوبيريدين مستبدلة
EP3344618A1 (de) 2015-09-04 2018-07-11 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate
CN113912586B (zh) 2016-08-31 2023-04-07 江苏恒瑞医药股份有限公司 氧代吡啶酰胺类衍生物、其制备方法及其在医药上的应用

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