JP2020511457A5 - - Google Patents
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- Publication number
- JP2020511457A5 JP2020511457A5 JP2019549506A JP2019549506A JP2020511457A5 JP 2020511457 A5 JP2020511457 A5 JP 2020511457A5 JP 2019549506 A JP2019549506 A JP 2019549506A JP 2019549506 A JP2019549506 A JP 2019549506A JP 2020511457 A5 JP2020511457 A5 JP 2020511457A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- ethyl
- chloro
- methoxypiperidin
- imidazol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 CCc([n]c(C(NC(CCN(C1)c2nnc(C(C)(CO)O)[s]2)C1O*)=O)n1)c1Cl Chemical compound CCc([n]c(C(NC(CCN(C1)c2nnc(C(C)(CO)O)[s]2)C1O*)=O)n1)c1Cl 0.000 description 4
- OXPMFWCVFIRINV-UHFFFAOYSA-N CCc([nH]c(C(NC(CC1)CCN1c1nnc(C(C)(C)O)[s]1)=O)n1)c1Cl Chemical compound CCc([nH]c(C(NC(CC1)CCN1c1nnc(C(C)(C)O)[s]1)=O)n1)c1Cl OXPMFWCVFIRINV-UHFFFAOYSA-N 0.000 description 1
- ZOJOQBJHNOZVRY-VIFPVBQESA-N CCc([nH]c(C(NC(CC1)CCN1c1nnc([C@@H](C)CO)[s]1)=O)n1)c1Cl Chemical compound CCc([nH]c(C(NC(CC1)CCN1c1nnc([C@@H](C)CO)[s]1)=O)n1)c1Cl ZOJOQBJHNOZVRY-VIFPVBQESA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201711008754 | 2017-03-14 | ||
| IN201711008754 | 2017-03-14 | ||
| PCT/JP2018/010670 WO2018169092A1 (en) | 2017-03-14 | 2018-03-13 | N-phosphonoxymethyl prodrugs of hydroxyalkyl thiadiazole derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2020511457A JP2020511457A (ja) | 2020-04-16 |
| JP2020511457A5 true JP2020511457A5 (https=) | 2020-07-27 |
Family
ID=62002340
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019549506A Pending JP2020511457A (ja) | 2017-03-14 | 2018-03-13 | ヒドロキシアルキルチアジアゾール誘導体のｎ−ホスホノキシメチルプロドラッグ |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US10752647B2 (https=) |
| EP (1) | EP3596071A1 (https=) |
| JP (1) | JP2020511457A (https=) |
| CA (1) | CA3056571C (https=) |
| TW (1) | TW201840322A (https=) |
| WO (1) | WO2018169092A1 (https=) |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200526626A (en) | 2003-09-13 | 2005-08-16 | Astrazeneca Ab | Chemical compounds |
| WO2006087544A2 (en) | 2005-02-18 | 2006-08-24 | Astrazeneca Ab | Pyrrole derivatives as dna gyrase and topoisomerase inhibitors |
| NZ561613A (en) | 2005-02-18 | 2010-12-24 | Astrazeneca Ab | Antibacterial piperidine derivatives |
| CN101163674A (zh) | 2005-02-18 | 2008-04-16 | 阿斯利康(瑞典)有限公司 | 作为dna促旋酶和拓扑异构酶抑制剂的吡咯衍生物 |
| US20080269214A1 (en) | 2005-03-04 | 2008-10-30 | Astrazeneca Ab | Pyrrole Derivatives as Dna Gyrase and Topoisomerase Inhibitors |
| CN101171250A (zh) | 2005-03-04 | 2008-04-30 | 阿斯利康(瑞典)有限公司 | 具有抗菌活性的氮杂环丁烷和吡咯的三环衍生物 |
| JP2009520785A (ja) | 2005-12-23 | 2009-05-28 | アストラゼネカ アクチボラグ | 抗菌性のピロロピリジン、ピロロピリミジン、及びピロロアゼピン |
| WO2008020229A2 (en) | 2006-08-17 | 2008-02-21 | Astrazeneca Ab | Antibacterial pyrrolecarboxamides |
| WO2008020227A2 (en) | 2006-08-17 | 2008-02-21 | Astrazeneca Ab | Antibacterial pyrrolecarboxamides |
| TW200819437A (en) | 2006-08-17 | 2008-05-01 | Astrazeneca Ab | Chemical compounds |
| TW200906412A (en) | 2007-06-12 | 2009-02-16 | Astrazeneca Ab | Piperidine compounds and uses thereof |
| TWI498115B (zh) | 2007-12-27 | 2015-09-01 | Daiichi Sankyo Co Ltd | 咪唑羰基化合物 |
| US20120108565A1 (en) | 2008-07-30 | 2012-05-03 | Lalima Sharma | Pyrrole carboxylic acid derivatives as antibacterial agents |
| TW201026694A (en) | 2008-12-12 | 2010-07-16 | Astrazeneca Ab | Compound 468 |
| TW201026695A (en) | 2008-12-12 | 2010-07-16 | Astrazeneca Ab | Piperidine compounds and uses thereof-596 |
| JP2011026305A (ja) * | 2009-06-24 | 2011-02-10 | Daiichi Sankyo Co Ltd | イミダゾールカルボニル化合物を含有する医薬組成物 |
| CN103261200B (zh) * | 2010-09-13 | 2016-03-30 | 阿迪维纳斯疗法有限公司 | 作为a2b腺苷受体拮抗剂的前药的嘌呤化合物、它们的制备方法及医药用途 |
| WO2014057415A2 (en) | 2012-10-10 | 2014-04-17 | Vitas Pharma Research Pvt Ltd | Inhibitors of dna gyrase for the treatment of bacterial infections |
| KR20180054650A (ko) | 2015-09-30 | 2018-05-24 | 다이이찌 산쿄 가부시키가이샤 | 히드록시알킬 티아디아졸 유도체 |
-
2018
- 2018-03-13 EP EP18718234.0A patent/EP3596071A1/en not_active Withdrawn
- 2018-03-13 JP JP2019549506A patent/JP2020511457A/ja active Pending
- 2018-03-13 US US16/492,027 patent/US10752647B2/en active Active
- 2018-03-13 CA CA3056571A patent/CA3056571C/en active Active
- 2018-03-13 TW TW107108384A patent/TW201840322A/zh unknown
- 2018-03-13 WO PCT/JP2018/010670 patent/WO2018169092A1/en not_active Ceased
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