JP2019535788A5 - - Google Patents

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Publication number
JP2019535788A5
JP2019535788A5 JP2019528512A JP2019528512A JP2019535788A5 JP 2019535788 A5 JP2019535788 A5 JP 2019535788A5 JP 2019528512 A JP2019528512 A JP 2019528512A JP 2019528512 A JP2019528512 A JP 2019528512A JP 2019535788 A5 JP2019535788 A5 JP 2019535788A5
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JP
Japan
Prior art keywords
alkyl
group
pharmaceutically acceptable
halo
substituted
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JP2019528512A
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English (en)
Japanese (ja)
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JP7114591B2 (ja
JP2019535788A (ja
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Priority claimed from PCT/US2017/063231 external-priority patent/WO2018098412A1/en
Publication of JP2019535788A publication Critical patent/JP2019535788A/ja
Publication of JP2019535788A5 publication Critical patent/JP2019535788A5/ja
Application granted granted Critical
Publication of JP7114591B2 publication Critical patent/JP7114591B2/ja
Active legal-status Critical Current
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JP2019528512A 2016-11-28 2017-11-27 Gsk-3阻害剤 Active JP7114591B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662426631P 2016-11-28 2016-11-28
US62/426,631 2016-11-28
PCT/US2017/063231 WO2018098412A1 (en) 2016-11-28 2017-11-27 Gsk-3 inhibitors

Publications (3)

Publication Number Publication Date
JP2019535788A JP2019535788A (ja) 2019-12-12
JP2019535788A5 true JP2019535788A5 (cg-RX-API-DMAC10.html) 2022-03-01
JP7114591B2 JP7114591B2 (ja) 2022-08-08

Family

ID=60655130

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019528512A Active JP7114591B2 (ja) 2016-11-28 2017-11-27 Gsk-3阻害剤

Country Status (8)

Country Link
US (1) US10752609B2 (cg-RX-API-DMAC10.html)
EP (1) EP3544613B1 (cg-RX-API-DMAC10.html)
JP (1) JP7114591B2 (cg-RX-API-DMAC10.html)
KR (1) KR102575990B1 (cg-RX-API-DMAC10.html)
CN (1) CN110545817B (cg-RX-API-DMAC10.html)
ES (1) ES2878078T3 (cg-RX-API-DMAC10.html)
MA (1) MA46889A (cg-RX-API-DMAC10.html)
WO (1) WO2018098412A1 (cg-RX-API-DMAC10.html)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110198934B (zh) * 2016-11-28 2022-07-22 百时美施贵宝公司 作为gsk-3抑制剂的嘧啶甲酰胺
MA54550A (fr) 2018-12-20 2022-03-30 Amgen Inc Inhibiteurs de kif18a
AU2019401495B2 (en) 2018-12-20 2025-06-26 Amgen Inc. Heteroaryl amides useful as KIF18A inhibitors
AU2019404576B2 (en) * 2018-12-20 2025-07-17 Amgen Inc. Heteroaryl amides useful as KIF18A inhibitors
AU2020325115B2 (en) 2019-08-02 2026-03-12 Amgen Inc. Pyridine derivatives as KIF18A inhibitors
JP7699100B2 (ja) 2019-08-02 2025-06-26 アムジエン・インコーポレーテツド Kif18a阻害剤
CN116178281B (zh) * 2023-04-27 2023-07-21 中国药科大学 一种双功能免疫抑制剂及其制备方法和应用
CN121666382A (zh) * 2023-05-10 2026-03-13 缆图药品公司 GSK3α抑制剂和其使用方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102438D0 (sv) * 2001-07-05 2001-07-05 Astrazeneca Ab New compounds
BRPI0814441A2 (pt) * 2007-07-19 2015-07-14 Schering Corp Compostos de amida heterocíclica como inibidores de proteína cinase
WO2012024179A1 (en) * 2010-08-18 2012-02-23 Merck Sharp & Dohme Corp. Substituted amide derivatives as dgat-1 inhibitors
JP2017500287A (ja) * 2013-11-06 2017-01-05 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company Gsk−3阻害剤として有用な置換ピリジン誘導体
AU2014347027A1 (en) 2013-11-06 2016-06-23 Bristol-Myers Squibb Company GSK -3 inhibitors
WO2016144792A1 (en) * 2015-03-06 2016-09-15 Alpharmagen, Llc Alpha 7 nicotinic acetylcholine receptor allosteric modulators, their derivatives and uses thereof
CN110198934B (zh) * 2016-11-28 2022-07-22 百时美施贵宝公司 作为gsk-3抑制剂的嘧啶甲酰胺

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