JP2019524720A5 - - Google Patents
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- Publication number
- JP2019524720A5 JP2019524720A5 JP2019500809A JP2019500809A JP2019524720A5 JP 2019524720 A5 JP2019524720 A5 JP 2019524720A5 JP 2019500809 A JP2019500809 A JP 2019500809A JP 2019500809 A JP2019500809 A JP 2019500809A JP 2019524720 A5 JP2019524720 A5 JP 2019524720A5
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- triazole
- alkyl
- optionally
- deoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP16179060.5 | 2016-07-12 | ||
| EP16179060 | 2016-07-12 | ||
| PCT/EP2017/067180 WO2018011093A1 (en) | 2016-07-12 | 2017-07-09 | Alpha-d-galactoside inhibitors of galectins |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019524720A JP2019524720A (ja) | 2019-09-05 |
| JP2019524720A5 true JP2019524720A5 (OSRAM) | 2021-11-04 |
| JP7038099B2 JP7038099B2 (ja) | 2022-03-17 |
Family
ID=56411454
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019500809A Expired - Fee Related JP7038099B2 (ja) | 2016-07-12 | 2017-07-09 | ガレクチンのα－Ｄ－ガラクトシド阻害剤 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US10988502B2 (OSRAM) |
| EP (1) | EP3484903A1 (OSRAM) |
| JP (1) | JP7038099B2 (OSRAM) |
| CN (1) | CN109563120B (OSRAM) |
| CA (1) | CA3025866A1 (OSRAM) |
| WO (1) | WO2018011093A1 (OSRAM) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107406478B (zh) | 2015-01-30 | 2021-07-27 | 格莱克特生物技术公司 | 半乳糖凝集素的α-D-半乳糖苷抑制剂 |
| WO2018011094A1 (en) * | 2016-07-12 | 2018-01-18 | Galecto Biotech Ab | Alpha-d-galactoside inhibitors of galectins |
| BR112020013647A2 (pt) | 2018-01-10 | 2020-12-01 | Galecto Biotech Ab | novo inibidor galactosídeo de galectinas |
| US11299485B2 (en) | 2018-01-25 | 2022-04-12 | Fujimoto Co., Ltd. | Thiophene derivative and use thereof |
| JP2021529163A (ja) | 2018-06-29 | 2021-10-28 | グリコス バイオメディカル オーワイ | コンジュゲート |
| WO2020078807A1 (en) * | 2018-10-15 | 2020-04-23 | Galecto Biotech Ab | Prodrug of galactoside inhibitors of galectins |
| CN113366007A (zh) * | 2018-10-15 | 2021-09-07 | 格莱克特生物技术公司 | 半乳糖凝集素的半乳糖苷抑制剂 |
| US11447517B2 (en) * | 2018-11-21 | 2022-09-20 | Galecto Biotech Ab | Galactoside inhibitor of galectins |
| WO2020248068A1 (en) | 2019-06-14 | 2020-12-17 | UNIVERSITé LAVAL | Synthesis of 3-azido-3-deoxy-d-galactopyranose |
| JP7674275B2 (ja) * | 2019-07-03 | 2025-05-09 | ガレクト バイオテック エービー | ガレクチンの新規なガラクトシド阻害剤 |
| WO2021001528A1 (en) * | 2019-07-03 | 2021-01-07 | Galecto Biotech Ab | Novel galactoside inhibitor of galectins |
| US20230038373A1 (en) | 2019-12-18 | 2023-02-09 | Glykos Biomedical Oy | Stabile conjugate |
| EP4081519A1 (en) * | 2019-12-24 | 2022-11-02 | GlycoMimetics, Inc. | Galectin-3 inhibiting c-glycoside ketones, ethers, and alcohols |
| CN113943330A (zh) * | 2020-07-17 | 2022-01-18 | 中国科学院上海药物研究所 | 一类含糖结构化合物、其制备方法、药物组合物和用途 |
| CA3202107A1 (en) * | 2020-12-22 | 2022-06-30 | Galecto Biotech Ab | Novel galactoside inhibitor of galectins |
| CN117043156A (zh) * | 2020-12-28 | 2023-11-10 | 格莱克特生物技术公司 | 半乳糖凝集素的新型半乳糖苷抑制剂 |
| CZ2023132A3 (cs) * | 2023-04-04 | 2024-10-16 | Ústav Chemických Procesů Av Čr, V. V. I. | Komplexy ruthenia pro inhibici galektinů, způsob jejich výroby a jejich použití |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060148712A1 (en) * | 2000-03-13 | 2006-07-06 | Fu-Tong Liu | Monocyte chemoattractant activity of galectin-3 |
| US6849607B2 (en) | 2001-05-09 | 2005-02-01 | Health Research, Inc. | Galectin recognized photosensitizers for photodynamic therapy |
| SE0401301D0 (sv) * | 2004-05-21 | 2004-05-21 | Forskarpatent I Syd Ab | Novel 3-triazolyl-galactoside inhibitors of galectins |
| SE0401300D0 (sv) | 2004-05-21 | 2004-05-21 | Forskarpatent I Syd Ab | Novel Galactoside Inhibitors of Galectins |
| US8703720B2 (en) | 2009-04-28 | 2014-04-22 | Galecto Biotech Ab | Galactoside inhibitors of galectins |
| WO2014067986A1 (en) | 2012-10-31 | 2014-05-08 | Galecto Biotech Ab | Galactoside inhibitor of galectin-3 and its use for treating pulmonary fibrosis |
| EP2620443A1 (en) * | 2012-01-25 | 2013-07-31 | Galecto Biotech AB | Novel galactoside inhibitors of galectins |
| EP2906227B1 (en) | 2012-10-10 | 2018-10-03 | Galectin Therapeutics Inc. | Galactose-pronged carbohydrate compounds for the treatment of diabetic nephropathy and associated disorders |
| JP6366598B2 (ja) * | 2012-11-15 | 2018-08-01 | タフツ ユニバーシティー | ガレクチンタンパク質阻害剤を用いて被験体の眼の血管新生または繊維症を処置し、調節し、または、予防する方法、組成物、およびキット |
| CN107406478B (zh) * | 2015-01-30 | 2021-07-27 | 格莱克特生物技术公司 | 半乳糖凝集素的α-D-半乳糖苷抑制剂 |
| WO2018011094A1 (en) * | 2016-07-12 | 2018-01-18 | Galecto Biotech Ab | Alpha-d-galactoside inhibitors of galectins |
-
2017
- 2017-07-09 EP EP17735568.2A patent/EP3484903A1/en not_active Withdrawn
- 2017-07-09 CN CN201780042826.6A patent/CN109563120B/zh not_active Expired - Fee Related
- 2017-07-09 JP JP2019500809A patent/JP7038099B2/ja not_active Expired - Fee Related
- 2017-07-09 WO PCT/EP2017/067180 patent/WO2018011093A1/en not_active Ceased
- 2017-07-09 US US16/313,625 patent/US10988502B2/en active Active
- 2017-07-09 CA CA3025866A patent/CA3025866A1/en active Pending
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