JP2019507745A5 - - Google Patents
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- Publication number
- JP2019507745A5 JP2019507745A5 JP2018541607A JP2018541607A JP2019507745A5 JP 2019507745 A5 JP2019507745 A5 JP 2019507745A5 JP 2018541607 A JP2018541607 A JP 2018541607A JP 2018541607 A JP2018541607 A JP 2018541607A JP 2019507745 A5 JP2019507745 A5 JP 2019507745A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cyano
- alkoxy
- group
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 44
- 229910052739 hydrogen Inorganic materials 0.000 claims description 43
- 239000001257 hydrogen Substances 0.000 claims description 43
- 229910052736 halogen Inorganic materials 0.000 claims description 41
- 150000002367 halogens Chemical class 0.000 claims description 41
- 125000001072 heteroaryl group Chemical group 0.000 claims description 21
- 125000000547 substituted alkyl group Chemical group 0.000 claims description 20
- 125000003118 aryl group Chemical group 0.000 claims description 18
- 125000003342 alkenyl group Chemical group 0.000 claims description 16
- 125000000304 alkynyl group Chemical group 0.000 claims description 16
- 125000005346 substituted cycloalkyl group Chemical group 0.000 claims description 14
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 claims description 12
- 125000003710 aryl alkyl group Chemical group 0.000 claims description 11
- 229910052760 oxygen Inorganic materials 0.000 claims description 10
- 125000005842 heteroatom Chemical group 0.000 claims description 9
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 8
- 125000003545 alkoxy group Chemical group 0.000 claims description 8
- 229910052717 sulfur Chemical group 0.000 claims description 8
- 125000001931 aliphatic group Chemical group 0.000 claims description 7
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims description 7
- 239000001301 oxygen Substances 0.000 claims description 7
- 150000003839 salts Chemical class 0.000 claims description 7
- 125000000217 alkyl group Chemical group 0.000 claims description 6
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 6
- 229920006395 saturated elastomer Polymers 0.000 claims description 6
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims description 5
- 229910052757 nitrogen Inorganic materials 0.000 claims description 5
- 239000011593 sulfur Chemical group 0.000 claims description 5
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 4
- 125000004438 haloalkoxy group Chemical group 0.000 claims description 4
- 125000001188 haloalkyl group Chemical group 0.000 claims description 4
- 125000004433 nitrogen atom Chemical group N* 0.000 claims description 3
- 125000003107 substituted aryl group Chemical group 0.000 claims description 3
- 125000004429 atom Chemical group 0.000 claims description 2
- 125000004430 oxygen atom Chemical group O* 0.000 claims description 2
- 150000003254 radicals Chemical class 0.000 claims description 2
- 125000006413 ring segment Chemical group 0.000 claims description 2
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 30
- 150000002431 hydrogen Chemical class 0.000 claims 27
- -1 C 1 -C 4 -alkoxy Chemical group 0.000 claims 22
- 229910052731 fluorine Inorganic materials 0.000 claims 15
- 239000011737 fluorine Substances 0.000 claims 15
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 15
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims 14
- 229910052801 chlorine Inorganic materials 0.000 claims 14
- 239000000460 chlorine Substances 0.000 claims 14
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 13
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 12
- 125000001424 substituent group Chemical group 0.000 claims 12
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 claims 11
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 claims 11
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 claims 11
- 229910052794 bromium Inorganic materials 0.000 claims 11
- 150000001875 compounds Chemical class 0.000 claims 11
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 11
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 8
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 8
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 7
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 7
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 6
- 125000000623 heterocyclic group Chemical group 0.000 claims 6
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims 5
- 241000607479 Yersinia pestis Species 0.000 claims 4
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims 4
- 125000001153 fluoro group Chemical group F* 0.000 claims 4
- 239000000203 mixture Substances 0.000 claims 4
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 claims 3
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 claims 3
- 239000004067 bulking agent Substances 0.000 claims 3
- 125000001028 difluoromethyl group Chemical group [H]C(F)(F)* 0.000 claims 3
- 125000001301 ethoxy group Chemical group [H]C([H])([H])C([H])([H])O* 0.000 claims 3
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 3
- 239000003090 pesticide formulation Substances 0.000 claims 3
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 2
- 238000000034 method Methods 0.000 claims 2
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims 2
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 claims 2
- 239000004094 surface-active agent Substances 0.000 claims 2
- 125000004205 trifluoroethyl group Chemical group [H]C([H])(*)C(F)(F)F 0.000 claims 2
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 claims 1
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 claims 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- UQZPGHOJMQTOHB-UHFFFAOYSA-N 2-chloro-n-(2-chloroethyl)-n-ethylethanamine Chemical compound ClCCN(CC)CCCl UQZPGHOJMQTOHB-UHFFFAOYSA-N 0.000 claims 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 1
- 239000003905 agrochemical Substances 0.000 claims 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 claims 1
- 125000004414 alkyl thio group Chemical group 0.000 claims 1
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 claims 1
- 125000006001 difluoroethyl group Chemical group 0.000 claims 1
- 125000003754 ethoxycarbonyl group Chemical group C(=O)(OCC)* 0.000 claims 1
- 125000005448 ethoxyethyl group Chemical group [H]C([H])([H])C([H])([H])OC([H])([H])C([H])([H])* 0.000 claims 1
- 125000005745 ethoxymethyl group Chemical group [H]C([H])([H])C([H])([H])OC([H])([H])* 0.000 claims 1
- 125000004785 fluoromethoxy group Chemical group [H]C([H])(F)O* 0.000 claims 1
- 238000009472 formulation Methods 0.000 claims 1
- 125000003253 isopropoxy group Chemical group [H]C([H])([H])C([H])(O*)C([H])([H])[H] 0.000 claims 1
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 claims 1
- 125000004184 methoxymethyl group Chemical group [H]C([H])([H])OC([H])([H])* 0.000 claims 1
- 125000004458 methylaminocarbonyl group Chemical group [H]N(C(*)=O)C([H])([H])[H] 0.000 claims 1
- 125000002816 methylsulfanyl group Chemical group [H]C([H])([H])S[*] 0.000 claims 1
- 210000000056 organ Anatomy 0.000 claims 1
- 238000006467 substitution reaction Methods 0.000 claims 1
- 230000001225 therapeutic effect Effects 0.000 claims 1
- 238000011282 treatment Methods 0.000 claims 1
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 claims 1
- 125000004435 hydrogen atom Chemical class [H]* 0.000 description 10
- 0 CC(C)*(C)=C[C@@](CN)N* Chemical compound CC(C)*(C)=C[C@@](CN)N* 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP16155136 | 2016-02-11 | ||
| EP16155136.1 | 2016-02-11 | ||
| PCT/EP2017/052497 WO2017137337A1 (de) | 2016-02-11 | 2017-02-06 | Substituierte imidazolyl-carboxamide als schädlingsbekämpfungsmittel |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019507745A JP2019507745A (ja) | 2019-03-22 |
| JP2019507745A5 true JP2019507745A5 (enExample) | 2020-03-12 |
| JP6892452B2 JP6892452B2 (ja) | 2021-06-23 |
Family
ID=55411188
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018541607A Expired - Fee Related JP6892452B2 (ja) | 2016-02-11 | 2017-02-06 | 有害生物防除剤としての置換イミダゾリル−カルボキサミド類 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US10501441B2 (enExample) |
| JP (1) | JP6892452B2 (enExample) |
| KR (1) | KR20180107141A (enExample) |
| CN (1) | CN109071507A (enExample) |
| AR (1) | AR107588A1 (enExample) |
| AU (1) | AU2017217580A1 (enExample) |
| BR (1) | BR112018016362A2 (enExample) |
| CA (1) | CA3013960A1 (enExample) |
| CL (1) | CL2018002295A1 (enExample) |
| CO (1) | CO2018008397A2 (enExample) |
| IL (1) | IL260829B (enExample) |
| MX (1) | MX2018009805A (enExample) |
| PH (1) | PH12018501705A1 (enExample) |
| RU (1) | RU2018132164A (enExample) |
| TW (1) | TW201741299A (enExample) |
| UY (1) | UY37119A (enExample) |
| WO (1) | WO2017137337A1 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN108713017A (zh) * | 2016-02-11 | 2018-10-26 | 拜耳作物科学股份公司 | 用作害虫防治剂的取代的氧基咪唑基羧酰胺 |
| MX2018009809A (es) * | 2016-02-11 | 2018-09-10 | Bayer Cropscience Ag | 2-oximidazolilcarboxamidas sustituidas como plaguicidas. |
| CA3013962A1 (en) * | 2016-02-11 | 2017-08-17 | Bayer Cropscience Aktiengesellschaft | Substituted 2-(het)aryl-imidazolyl-carboxyamides as pest control agents |
| KR20190037305A (ko) * | 2016-08-10 | 2019-04-05 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 해충 방제제로서의 치환된 2-헤테로시클릴 이미다졸릴-카르복스아미드 |
| WO2019137995A1 (en) | 2018-01-11 | 2019-07-18 | Basf Se | Novel pyridazine compounds for controlling invertebrate pests |
| CN111116483B (zh) * | 2019-11-25 | 2022-12-20 | 浙江师范大学 | 一种2-咪唑基咪唑类化合物及其制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL364660A1 (en) * | 2001-03-05 | 2004-12-13 | E.I.Du Pont De Nemours And Company | Heterocyclic diamide invertebrate pest control agents |
| FR2827286A1 (fr) * | 2001-07-11 | 2003-01-17 | Aventis Cropscience Sa | Nouveaux composes fongicides |
| EP1690863A1 (en) * | 2003-11-26 | 2006-08-16 | Dainippon Sumitomo Pharma Co., Ltd. | Novel condensed imidazole derivative |
| EP2236505A1 (de) * | 2009-04-03 | 2010-10-06 | Bayer CropScience AG | Acylierte Aminopyridine und - pyridazine als Insektizide |
| AU2010259002B2 (en) * | 2009-06-08 | 2014-03-20 | Nantbio, Inc. | Triazine derivatives and their therapeutical applications |
| US9125414B2 (en) | 2009-07-24 | 2015-09-08 | Basf Se | Pyridine derivatives compounds for controlling invertebrate pests |
| TWI702212B (zh) * | 2015-02-09 | 2020-08-21 | 德商拜耳作物科學股份有限公司 | 作為除害劑之經取代的２－硫基咪唑基羧醯胺類 |
| MX2018009809A (es) * | 2016-02-11 | 2018-09-10 | Bayer Cropscience Ag | 2-oximidazolilcarboxamidas sustituidas como plaguicidas. |
| CA3013962A1 (en) * | 2016-02-11 | 2017-08-17 | Bayer Cropscience Aktiengesellschaft | Substituted 2-(het)aryl-imidazolyl-carboxyamides as pest control agents |
-
2017
- 2017-02-06 AU AU2017217580A patent/AU2017217580A1/en not_active Abandoned
- 2017-02-06 CA CA3013960A patent/CA3013960A1/en not_active Abandoned
- 2017-02-06 CN CN201780022855.6A patent/CN109071507A/zh active Pending
- 2017-02-06 MX MX2018009805A patent/MX2018009805A/es unknown
- 2017-02-06 RU RU2018132164A patent/RU2018132164A/ru not_active Application Discontinuation
- 2017-02-06 US US16/076,797 patent/US10501441B2/en not_active Expired - Fee Related
- 2017-02-06 KR KR1020187022834A patent/KR20180107141A/ko not_active Withdrawn
- 2017-02-06 BR BR112018016362-7A patent/BR112018016362A2/pt not_active Application Discontinuation
- 2017-02-06 WO PCT/EP2017/052497 patent/WO2017137337A1/de not_active Ceased
- 2017-02-06 JP JP2018541607A patent/JP6892452B2/ja not_active Expired - Fee Related
- 2017-02-09 TW TW106104209A patent/TW201741299A/zh unknown
- 2017-02-10 AR ARP170100332A patent/AR107588A1/es unknown
- 2017-02-10 UY UY0001037119A patent/UY37119A/es not_active Application Discontinuation
-
2018
- 2018-07-29 IL IL260829A patent/IL260829B/en active IP Right Grant
- 2018-08-10 CL CL2018002295A patent/CL2018002295A1/es unknown
- 2018-08-10 PH PH12018501705A patent/PH12018501705A1/en unknown
- 2018-08-10 CO CONC2018/0008397A patent/CO2018008397A2/es unknown