JP2019501140A5 - - Google Patents

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JP2019501140A5
JP2019501140A5 JP2018527799A JP2018527799A JP2019501140A5 JP 2019501140 A5 JP2019501140 A5 JP 2019501140A5 JP 2018527799 A JP2018527799 A JP 2018527799A JP 2018527799 A JP2018527799 A JP 2018527799A JP 2019501140 A5 JP2019501140 A5 JP 2019501140A5
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cancer
pharmaceutically acceptable
acceptable salt
compound
leukemia
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JP2018527799A
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Japanese (ja)
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JP6882289B2 (ja
JP2019501140A (ja
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Priority claimed from PCT/US2016/063485 external-priority patent/WO2017091661A1/en
Publication of JP2019501140A publication Critical patent/JP2019501140A/ja
Publication of JP2019501140A5 publication Critical patent/JP2019501140A5/ja
Priority to JP2021078741A priority Critical patent/JP7112567B2/ja
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JP2018527799A 2015-11-25 2016-11-23 二環式ｂｅｔブロモドメイン阻害剤及びその使用 Active JP6882289B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2021078741A JP7112567B2 (ja) 2015-11-25 2021-05-06 二環式ｂｅｔブロモドメイン阻害剤及びその使用

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562259894P 2015-11-25 2015-11-25
US62/259,894 2015-11-25
PCT/US2016/063485 WO2017091661A1 (en) 2015-11-25 2016-11-23 Bicyclic bet bromodomain inhibitors and uses thereof

Related Child Applications (1)

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JP2021078741A Division JP7112567B2 (ja) 2015-11-25 2021-05-06 二環式ｂｅｔブロモドメイン阻害剤及びその使用

Publications (3)

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JP2019501140A JP2019501140A (ja) 2019-01-17
JP2019501140A5 true JP2019501140A5 (OSRAM) 2020-01-09
JP6882289B2 JP6882289B2 (ja) 2021-06-02

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JP2018527799A Active JP6882289B2 (ja) 2015-11-25 2016-11-23 二環式ｂｅｔブロモドメイン阻害剤及びその使用
JP2021078741A Active JP7112567B2 (ja) 2015-11-25 2021-05-06 二環式ｂｅｔブロモドメイン阻害剤及びその使用

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Country Status (8)

Country Link
US (2) US10508106B2 (OSRAM)
EP (2) EP3380469B1 (OSRAM)
JP (2) JP6882289B2 (OSRAM)
CN (2) CN109641886B (OSRAM)
AU (3) AU2016361441B2 (OSRAM)
CA (1) CA3006300C (OSRAM)
ES (2) ES2918589T3 (OSRAM)
WO (1) WO2017091661A1 (OSRAM)

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CN109111426B (zh) * 2017-06-23 2021-12-14 中国科学院上海药物研究所 一类稠合双环杂芳基或芳基化合物，及其用途
WO2019201296A1 (zh) * 2018-04-18 2019-10-24 南京明德新药研发有限公司 作为rho激酶抑制剂的吡唑类化合物
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WO2022083657A1 (zh) * 2020-10-20 2022-04-28 苏州泽璟生物制药股份有限公司 取代苯并或吡啶并嘧啶胺类抑制剂及其制备方法和应用
CN117279914A (zh) * 2021-01-29 2023-12-22 南京再明医药有限公司 Sos1抑制剂及其制备方法和应用
WO2022171018A1 (zh) * 2021-02-09 2022-08-18 苏州泽璟生物制药股份有限公司 取代苯并或吡啶并嘧啶胺类抑制剂及其制备方法和应用
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WO2022199670A1 (zh) * 2021-03-26 2022-09-29 南京明德新药研发有限公司 6-氨基甲酸酯取代的杂芳环衍生物
WO2024043319A1 (ja) * 2022-08-26 2024-02-29 エーザイ・アール・アンド・ディー・マネジメント株式会社 抗体薬物複合体
WO2024235225A1 (zh) * 2023-05-15 2024-11-21 苏州泽璟生物制药股份有限公司 取代嘧啶并环类抑制剂及其制备方法和应用
WO2025209570A1 (zh) * 2024-04-03 2025-10-09 北京大学 Bet抑制剂及其应用

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