JP2018535996A5 - - Google Patents

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Publication number
JP2018535996A5
JP2018535996A5 JP2018528591A JP2018528591A JP2018535996A5 JP 2018535996 A5 JP2018535996 A5 JP 2018535996A5 JP 2018528591 A JP2018528591 A JP 2018528591A JP 2018528591 A JP2018528591 A JP 2018528591A JP 2018535996 A5 JP2018535996 A5 JP 2018535996A5
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JP
Japan
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pharmaceutically acceptable
composition
acceptable salt
effective amount
administered
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JP2018528591A
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English (en)
Japanese (ja)
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JP6944936B2 (ja
JP2018535996A (ja
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Priority claimed from PCT/US2016/064824 external-priority patent/WO2017096303A2/en
Publication of JP2018535996A publication Critical patent/JP2018535996A/ja
Publication of JP2018535996A5 publication Critical patent/JP2018535996A5/ja
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Publication of JP6944936B2 publication Critical patent/JP6944936B2/ja
Expired - Fee Related legal-status Critical Current
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JP2018528591A 2015-12-04 2016-12-02 血液癌を処置するためのセルデュラチニブ Expired - Fee Related JP6944936B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201562263582P 2015-12-04 2015-12-04
US62/263,582 2015-12-04
US201662342755P 2016-05-27 2016-05-27
US201662342727P 2016-05-27 2016-05-27
US62/342,727 2016-05-27
US62/342,755 2016-05-27
US201662371145P 2016-08-04 2016-08-04
US62/371,145 2016-08-04
PCT/US2016/064824 WO2017096303A2 (en) 2015-12-04 2016-12-02 Cerdulatinib for treating hematological cancers

Publications (3)

Publication Number Publication Date
JP2018535996A JP2018535996A (ja) 2018-12-06
JP2018535996A5 true JP2018535996A5 (enExample) 2020-01-09
JP6944936B2 JP6944936B2 (ja) 2021-10-06

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ID=57614468

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018528591A Expired - Fee Related JP6944936B2 (ja) 2015-12-04 2016-12-02 血液癌を処置するためのセルデュラチニブ

Country Status (8)

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US (2) US10736895B2 (enExample)
EP (1) EP3383396B1 (enExample)
JP (1) JP6944936B2 (enExample)
CN (1) CN108367006B (enExample)
AU (1) AU2016363005A1 (enExample)
CA (1) CA2950640A1 (enExample)
ES (1) ES2959692T3 (enExample)
WO (1) WO2017096303A2 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107683139A (zh) * 2015-05-29 2018-02-09 博尔托拉制药公司 用于治疗b细胞恶性肿瘤的赛度替尼
ES2913119T3 (es) 2015-08-12 2022-05-31 Portola Pharm Inc Cerdulatinib para tratar mieloma
WO2019138291A2 (en) * 2018-01-09 2019-07-18 Dermavant Sciences GmbH Cerdulatinib-containing topical skin pharmaceutical compositions and uses thereof
WO2019213545A1 (en) 2018-05-04 2019-11-07 Portola Pharmaceuticals, Inc. Synthesis of cerdulatinib
KR20210003789A (ko) * 2018-05-04 2021-01-12 포톨라 파마슈티컬스, 인코포레이티드 림프종을 치료하는 방법
US10865198B2 (en) 2018-05-04 2020-12-15 Alexion Pharmaceuticals, Inc. Solid forms of cerdulatinib
AU2020222359A1 (en) * 2019-02-15 2021-09-02 Janssen Biotech, Inc. Combination therapy for treatment of B-cell malignancies
US20230181581A1 (en) * 2020-05-26 2023-06-15 Alexion Pharmaceuticals, Inc. Circulating b cell subpopulations in indolent b cell lymphoma

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Publication number Priority date Publication date Assignee Title
JP4135318B2 (ja) 1997-12-15 2008-08-20 アステラス製薬株式会社 新規なピリミジン−5−カルボキサミド誘導体
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
AU2003244098A1 (en) 2002-06-28 2004-01-19 Yamanouchi Pharmaceutical Co., Ltd. Diaminopyrimidinecarboxa mide derivative
EP2046759A1 (en) 2006-07-21 2009-04-15 Novartis AG 2, 4 -di (arylaminio) -pyrimidine-5-carboxamide compounds as jak kinases inhibitors
EP2526934B1 (en) 2006-09-22 2015-12-09 Pharmacyclics LLC Inhibitors of bruton's tyrosine kinase
MY155639A (en) 2008-04-16 2015-11-13 Portola Pharm Inc 2, 6-diamino-pyrimidin-5-yl-carboxamides as syk or jak kinases inhibitors
US8138339B2 (en) 2008-04-16 2012-03-20 Portola Pharmaceuticals, Inc. Inhibitors of protein kinases
AR076550A1 (es) 2009-05-06 2011-06-22 Portola Pharm Inc Inhibidores de la janus tirosina kinasa (jak)
UY32668A (es) 2009-05-26 2010-12-31 Abbott Lab Agentes inductores de la apoptosis para el tratamiento del cáncer y de enfermedades inmunes y autoinmunes
CA2780759A1 (en) 2009-12-01 2011-06-09 Rigel Pharmaceuticals, Inc. Protein kinase c inhibitors and uses thereof
US9357229B2 (en) 2010-07-28 2016-05-31 Qualcomm Incorporated Coding motion vectors in video coding
EP2621489A1 (en) 2010-09-30 2013-08-07 Portola Pharmaceuticals, Inc. Combinations of 4-(cyclopropylamino)-2-(4-(4-(ethylsulfonyl)piperazin-1-yl)phenylamino)pyrimidine-5-carboxamide and fludarabine
JP6141188B2 (ja) 2010-11-23 2017-06-07 アッヴィ・インコーポレイテッド アポトーシス誘導剤の塩および結晶の形態
WO2013023119A1 (en) 2011-08-10 2013-02-14 Novartis Pharma Ag JAK P13K/mTOR COMBINATION THERAPY
KR20150032340A (ko) 2012-07-24 2015-03-25 파마시클릭스, 인코포레이티드 브루톤 티로신 키나제(btk)의 억제제에 대한 내성과 관련된 돌연변이
EP2903970A4 (en) 2012-10-08 2016-11-30 Portola Pharm Inc SUBSTITUTED PYRIMIDINYL KINASE INHIBITORS
EA201590822A1 (ru) 2012-11-02 2016-01-29 Фармасайкликс, Инк. Адъювантная терапия ингибитором киназы семейства tec
WO2016040858A1 (en) 2014-09-12 2016-03-17 G1 Therapeutics, Inc. Combinations and dosing regimes to treat rb-positive tumors
CN107683139A (zh) 2015-05-29 2018-02-09 博尔托拉制药公司 用于治疗b细胞恶性肿瘤的赛度替尼
ES2913119T3 (es) 2015-08-12 2022-05-31 Portola Pharm Inc Cerdulatinib para tratar mieloma
US10865198B2 (en) 2018-05-04 2020-12-15 Alexion Pharmaceuticals, Inc. Solid forms of cerdulatinib

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