JP2018515514A5 - - Google Patents

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Publication number
JP2018515514A5
JP2018515514A5 JP2017558660A JP2017558660A JP2018515514A5 JP 2018515514 A5 JP2018515514 A5 JP 2018515514A5 JP 2017558660 A JP2017558660 A JP 2017558660A JP 2017558660 A JP2017558660 A JP 2017558660A JP 2018515514 A5 JP2018515514 A5 JP 2018515514A5
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JP
Japan
Prior art keywords
amino
alkyl
substituted
compound according
cancer
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JP2017558660A
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English (en)
Japanese (ja)
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JP6863901B2 (ja
JP2018515514A (ja
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Priority claimed from PCT/US2016/031996 external-priority patent/WO2016183278A1/en
Publication of JP2018515514A publication Critical patent/JP2018515514A/ja
Publication of JP2018515514A5 publication Critical patent/JP2018515514A5/ja
Application granted granted Critical
Publication of JP6863901B2 publication Critical patent/JP6863901B2/ja
Expired - Fee Related legal-status Critical Current
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JP2017558660A 2015-05-13 2016-05-12 キナーゼ阻害のためのヘテロアリール化合物 Expired - Fee Related JP6863901B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562160989P 2015-05-13 2015-05-13
US62/160,989 2015-05-13
PCT/US2016/031996 WO2016183278A1 (en) 2015-05-13 2016-05-12 Heteroaryl compounds for kinase inhibition

Publications (3)

Publication Number Publication Date
JP2018515514A JP2018515514A (ja) 2018-06-14
JP2018515514A5 true JP2018515514A5 (cg-RX-API-DMAC7.html) 2019-06-13
JP6863901B2 JP6863901B2 (ja) 2021-04-28

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ID=57249337

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017558660A Expired - Fee Related JP6863901B2 (ja) 2015-05-13 2016-05-12 キナーゼ阻害のためのヘテロアリール化合物

Country Status (5)

Country Link
US (1) US20210323976A1 (cg-RX-API-DMAC7.html)
EP (1) EP3294712A4 (cg-RX-API-DMAC7.html)
JP (1) JP6863901B2 (cg-RX-API-DMAC7.html)
HK (1) HK1251567A1 (cg-RX-API-DMAC7.html)
WO (1) WO2016183278A1 (cg-RX-API-DMAC7.html)

Families Citing this family (13)

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Publication number Priority date Publication date Assignee Title
EA201391626A1 (ru) 2011-05-04 2014-03-31 Ариад Фармасьютикалз, Инк. Соединения для ингибирования клеточной пролиферации в egfr-стимулированных типах рака
AU2013204563B2 (en) 2012-05-05 2016-05-19 Takeda Pharmaceutical Company Limited Compounds for inhibiting cell proliferation in EGFR-driven cancers
WO2017120429A1 (en) 2016-01-07 2017-07-13 CS Pharmasciences, Inc. Selective inhibitors of clinically important mutants of the egfr tyrosine kinase
CN108299419B (zh) * 2017-01-11 2022-04-26 南京圣和药业股份有限公司 一种新型egfr激酶抑制剂的几种新晶型及其制备方法
CN109705118B (zh) * 2017-10-25 2021-12-28 南京圣和药业股份有限公司 三环类egfr激酶抑制剂的制备方法
CN109705117A (zh) * 2017-10-25 2019-05-03 南京圣和药业股份有限公司 三环类化合物、其制备方法及用途
CN108191861B (zh) * 2018-03-01 2020-10-02 天津大学 N-[5-(嘧啶-2-氨基)-2,4-二取代苯基]-反式-2,4-戊二烯酰胺
BR112021025764A2 (pt) * 2019-06-20 2022-02-01 Oncobix Co Ltd Derivado de pirimidina que inibe o crescimento de células cancerígenas e uso medicinal do mesmo
CN115052878B (zh) 2020-02-03 2024-07-09 勃林格殷格翰国际有限公司 作为HER2抑制剂的[1,3]二嗪并[5,4-d]嘧啶
WO2021156180A1 (en) 2020-02-03 2021-08-12 Boehringer Ingelheim International Gmbh [1,3]diazino[5,4-d]pyrimidines as her2 inhibitors
US11608343B2 (en) * 2020-04-24 2023-03-21 Boehringer Ingelheim International Gmbh Substituted pyrimido[5,4-d]pyrimidines as HER2 inhibitors
CN112409192A (zh) * 2020-11-26 2021-02-26 启东东岳药业有限公司 一种4-氟-2-甲氧基苯胺的纯化方法
CA3213079A1 (en) 2021-04-13 2022-10-20 Kristin Lynne ANDREWS Amino-substituted heterocycles for treating cancers with egfr mutations

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003000251A1 (en) * 2001-06-21 2003-01-03 Ariad Pharmaceuticals, Inc. Novel idolinones and uses thereof
US7982036B2 (en) * 2007-10-19 2011-07-19 Avila Therapeutics, Inc. 4,6-disubstitued pyrimidines useful as kinase inhibitors
PT2300013T (pt) * 2008-05-21 2017-10-31 Ariad Pharma Inc Derivados de fósforo como inibidores de cinases
US9273077B2 (en) * 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
CA3031835C (en) * 2008-06-27 2021-09-07 Celgene Car Llc Heteroaryl compounds and uses thereof
CN105198862B (zh) * 2011-07-27 2018-01-23 阿斯利康(瑞典)有限公司 取代的n‑(4‑氟‑2‑甲氧基‑5‑硝基苯基)嘧啶‑2‑胺化合物及其盐
EP3057954A2 (en) * 2013-10-18 2016-08-24 Syros Pharmaceuticals, Inc. Heteromaromatic compounds useful for the treatment of proliferative diseases
EP3143015B1 (en) * 2014-05-13 2019-02-20 ARIAD Pharmaceuticals, Inc. Heteroaryl compounds for kinase inhibition
SG11201610517PA (en) * 2014-06-19 2017-01-27 Ariad Pharma Inc Heteroaryl compounds for kinase inhibition
EP3312179B1 (en) * 2015-04-29 2019-07-10 Nanjing Sanhome Pharmaceutical Co., Ltd. Fused-ring or tricyclic aryl pyrimidine compound used as kinase inhibitor

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