JP2018503647A5 - - Google Patents

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Publication number
JP2018503647A5
JP2018503647A5 JP2017539234A JP2017539234A JP2018503647A5 JP 2018503647 A5 JP2018503647 A5 JP 2018503647A5 JP 2017539234 A JP2017539234 A JP 2017539234A JP 2017539234 A JP2017539234 A JP 2017539234A JP 2018503647 A5 JP2018503647 A5 JP 2018503647A5
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JP
Japan
Prior art keywords
alkyl
compound
group
substituted
independently selected
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JP2017539234A
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English (en)
Japanese (ja)
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JP2018503647A (ja
JP6615896B2 (ja
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Priority claimed from PCT/US2016/015251 external-priority patent/WO2016123275A1/en
Publication of JP2018503647A publication Critical patent/JP2018503647A/ja
Publication of JP2018503647A5 publication Critical patent/JP2018503647A5/ja
Application granted granted Critical
Publication of JP6615896B2 publication Critical patent/JP6615896B2/ja
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JP2017539234A 2015-01-30 2016-01-28 アルドステロン合成酵素阻害剤 Active JP6615896B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562109890P 2015-01-30 2015-01-30
US62/109,890 2015-01-30
PCT/US2016/015251 WO2016123275A1 (en) 2015-01-30 2016-01-28 Aldosterone synthase inhibitors

Publications (3)

Publication Number Publication Date
JP2018503647A JP2018503647A (ja) 2018-02-08
JP2018503647A5 true JP2018503647A5 (https=) 2019-03-07
JP6615896B2 JP6615896B2 (ja) 2019-12-04

Family

ID=55361967

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017539234A Active JP6615896B2 (ja) 2015-01-30 2016-01-28 アルドステロン合成酵素阻害剤

Country Status (4)

Country Link
US (1) US10131642B1 (https=)
EP (1) EP3250569B1 (https=)
JP (1) JP6615896B2 (https=)
WO (1) WO2016123275A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019215709A1 (en) * 2018-02-02 2020-07-16 Boehringer Ingelheim International Gmbh Heterocyclyl-substituted oxadiazolopyridine derivatives for use as ghrelin O-acyl transferase (GOAT) inhibitors
EP3746449B1 (en) * 2018-02-02 2022-03-30 Boehringer Ingelheim International GmbH Pyrazole- and indazole-substituted oxadiazolopyridine derivatives for use as ghrelin o-acyl transferase (goat) inhibitors
WO2019149657A1 (en) 2018-02-02 2019-08-08 Boehringer Ingelheim International Gmbh Benzyl-, (pyridin-3-yl)methyl- or (pyridin-4-yl)methyl-substituted oxadiazolopyridine derivatives as ghrelin o-acyl transferase (goat) inhibitors
MX2020007994A (es) 2018-02-02 2020-09-09 Boehringer Ingelheim Int Derivados de triazolopirimidina para usar como inhibidores de ghrelin o-aciltransferasa (goat).
DK4153599T3 (da) 2020-05-22 2024-06-17 Boehringer Ingelheim Int Fremgangsmåde til at fremstille alkyl 7-amino-5-methyl-[1,2,5]oxadiazolo[3,4-b]pyridin-carboxylat
ES2991340T3 (es) 2020-05-22 2024-12-03 Boehringer Ingelheim Int Procedimiento continuo de fabricación de 7-amino-5-metil-[1,2,5]oxadiazolo[3,4-b]piridín-carboxilato de alquilo

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1484325B1 (en) * 2002-03-08 2014-06-18 Japan Science and Technology Agency Isoxazole derivatives and process for producing the same
DE102004035322A1 (de) * 2004-07-21 2006-02-16 Universität des Saarlandes Selektive Hemmstoffe humaner Corticoidsynthasen
WO2007117982A2 (en) * 2006-03-29 2007-10-18 Novartis Ag Organic compounds
MX2008015008A (es) * 2006-05-26 2008-12-05 Novartis Ag INHIBIDORES DE SINTASA DE ALDOSTERONA Y/O DE 11ß-HIDROXILASA.
ITMI20062102A1 (it) * 2006-11-02 2008-05-03 Abiogen Pharma Spa Nuovui sali di 3-benzil-2-metil-2,3,3a,4,5,6,7,7a-ottaidrobenzo-d-isossazol-4-one
CA2709784A1 (en) * 2007-12-21 2009-07-09 University Of Rochester Method for altering the lifespan of eukaryotic organisms

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