JP2017531041A5 - - Google Patents

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Publication number
JP2017531041A5
JP2017531041A5 JP2017538930A JP2017538930A JP2017531041A5 JP 2017531041 A5 JP2017531041 A5 JP 2017531041A5 JP 2017538930 A JP2017538930 A JP 2017538930A JP 2017538930 A JP2017538930 A JP 2017538930A JP 2017531041 A5 JP2017531041 A5 JP 2017531041A5
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JP
Japan
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compound
alkyl
macrocyclic compound
alkenyl
aralkyl
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JP2017538930A
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English (en)
Japanese (ja)
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JP6678679B2 (ja
JP2017531041A (ja
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Priority claimed from PCT/US2015/055317 external-priority patent/WO2016061097A1/en
Publication of JP2017531041A publication Critical patent/JP2017531041A/ja
Publication of JP2017531041A5 publication Critical patent/JP2017531041A5/ja
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Publication of JP6678679B2 publication Critical patent/JP6678679B2/ja
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JP2017538930A 2014-10-13 2015-10-13 毛細血管拡張性運動失調症およびRad3関連(ATR)プロテインキナーゼ阻害剤 Active JP6678679B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201462063176P 2014-10-13 2014-10-13
US62/063,176 2014-10-13
US201562104274P 2015-01-16 2015-01-16
US62/104,274 2015-01-16
PCT/US2015/055317 WO2016061097A1 (en) 2014-10-13 2015-10-13 Ataxia telengiectasia and rad3-related (atr) protein kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2017531041A JP2017531041A (ja) 2017-10-19
JP2017531041A5 true JP2017531041A5 (US07794700-20100914-C00125.png) 2018-11-15
JP6678679B2 JP6678679B2 (ja) 2020-04-08

Family

ID=55654998

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2017538930A Active JP6678679B2 (ja) 2014-10-13 2015-10-13 毛細血管拡張性運動失調症およびRad3関連(ATR)プロテインキナーゼ阻害剤

Country Status (12)

Country Link
US (3) US9663535B2 (US07794700-20100914-C00125.png)
EP (1) EP3207031B1 (US07794700-20100914-C00125.png)
JP (1) JP6678679B2 (US07794700-20100914-C00125.png)
KR (1) KR102569226B1 (US07794700-20100914-C00125.png)
CN (1) CN107108527B (US07794700-20100914-C00125.png)
AU (1) AU2015333738B2 (US07794700-20100914-C00125.png)
BR (1) BR112017007708B8 (US07794700-20100914-C00125.png)
CA (1) CA2963973C (US07794700-20100914-C00125.png)
ES (1) ES2879441T3 (US07794700-20100914-C00125.png)
IL (1) IL251595B (US07794700-20100914-C00125.png)
MX (1) MX2017004515A (US07794700-20100914-C00125.png)
WO (1) WO2016061097A1 (US07794700-20100914-C00125.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3207031B1 (en) 2014-10-13 2021-04-14 Atrin Pharmaceuticals LLC Ataxia telengiectasia and rad3-related (atr) protein kinase inhibitors
WO2017180723A1 (en) * 2016-04-12 2017-10-19 Atrin Pharmaceuticals LLC Ataxia telengiectasia and rad3-related (atr) inhibitors and methods of their use
US10421765B2 (en) 2017-05-26 2019-09-24 Board Of Regents, The University Of Texas System Tetrahydropyrido[4,3-d]pyrimidine inhibitors of ATR kinase
CN111867590B (zh) 2017-07-13 2023-11-17 德州大学系统董事会 Atr激酶的杂环抑制剂
US10800774B2 (en) 2017-08-17 2020-10-13 Board Of Regents, The University Of Texas System Heterocyclic inhibitors of ATR kinase
US11267809B2 (en) 2017-09-14 2022-03-08 The Board Of Trustees Of The Leland Stanford Junior University BAF complex modulating compounds and methods of using the same
EP3765008B1 (en) 2018-03-16 2023-06-07 Board of Regents, The University of Texas System Heterocyclic inhibitors of atr kinase
CN110357905B (zh) * 2018-03-26 2021-10-01 武汉誉祥医药科技有限公司 作为蛋白激酶抑制剂的大环类衍生物及其制备方法和用途
WO2020014524A1 (en) 2018-07-12 2020-01-16 The Board Of Trustees Of The Leland Stanford Junior University Methods for reversing hiv latency using baf complex modulating compounds
CN110950890B (zh) * 2018-09-27 2022-07-01 北京赛林泰医药技术有限公司 取代的咪唑并[4,5-c]喹啉大环化合物作为多靶点激酶抑制剂
JP2023545196A (ja) 2020-10-16 2023-10-26 シャンハイ ドーァ ノボ ファーマテック カンパニー,リミティド 三複素環誘導体、その医薬組成物及び使用
WO2023201320A1 (en) 2022-04-14 2023-10-19 Atrin Pharmaceuticals LLC Atr inhibitors
WO2023242302A1 (en) 2022-06-15 2023-12-21 Astrazeneca Ab Combination therapy for treating cancer

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2517256C (en) 2003-02-26 2013-04-30 Sugen, Inc. Aminoheteroaryl compounds as protein kinase inhibitors
US7163939B2 (en) * 2003-11-05 2007-01-16 Abbott Laboratories Macrocyclic kinase inhibitors
MX2011006503A (es) * 2008-12-19 2011-09-06 Vertex Pharma Derivados de pirazina utiles como inhibidores de la cinasa de atr.
WO2011143425A2 (en) * 2010-05-12 2011-11-17 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
WO2012125603A1 (en) * 2011-03-16 2012-09-20 Cephalon, Inc. Macrocyclic compounds as alk, fak and jak2 inhibitors
SI2822953T1 (sl) * 2012-03-06 2017-04-26 Pfizer Inc. Makrociklični derivati za zdravljenje proliferativnih bolezni
NZ630901A (en) * 2012-03-17 2015-09-25 Polyphor Ag Conformationally constrained, fully synthetic macrocyclic compounds
CN104513253A (zh) * 2013-10-01 2015-04-15 南京波尔泰药业科技有限公司 用于治疗增殖性疾病的大环化合物
EP3207031B1 (en) 2014-10-13 2021-04-14 Atrin Pharmaceuticals LLC Ataxia telengiectasia and rad3-related (atr) protein kinase inhibitors

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