JP2017531039A5 - - Google Patents

Download PDF

Info

Publication number
JP2017531039A5
JP2017531039A5 JP2017538467A JP2017538467A JP2017531039A5 JP 2017531039 A5 JP2017531039 A5 JP 2017531039A5 JP 2017538467 A JP2017538467 A JP 2017538467A JP 2017538467 A JP2017538467 A JP 2017538467A JP 2017531039 A5 JP2017531039 A5 JP 2017531039A5
Authority
JP
Japan
Prior art keywords
dihydro
thieno
azaspiro
oxa
carboxamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2017538467A
Other languages
English (en)
Japanese (ja)
Other versions
JP2017531039A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/GB2015/052945 external-priority patent/WO2016055792A1/en
Publication of JP2017531039A publication Critical patent/JP2017531039A/ja
Publication of JP2017531039A5 publication Critical patent/JP2017531039A5/ja
Withdrawn legal-status Critical Current

Links

JP2017538467A 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体 Withdrawn JP2017531039A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14188494.0 2014-10-10
EP14188494 2014-10-10
PCT/GB2015/052945 WO2016055792A1 (en) 2014-10-10 2015-10-08 Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivatives

Publications (2)

Publication Number Publication Date
JP2017531039A JP2017531039A (ja) 2017-10-19
JP2017531039A5 true JP2017531039A5 (enExample) 2018-11-22

Family

ID=51842340

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2017538466A Active JP6675407B2 (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体
JP2017538467A Withdrawn JP2017531039A (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2017538466A Active JP6675407B2 (ja) 2014-10-10 2015-10-08 新規5,6−ジヒドロ−4H−ベンゾ[b]チエノ−[2,3−d]アゼピン誘導体

Country Status (13)

Country Link
US (6) US9732098B2 (enExample)
EP (2) EP3204388B1 (enExample)
JP (2) JP6675407B2 (enExample)
KR (1) KR20170058921A (enExample)
CN (1) CN106852144B (enExample)
AU (1) AU2015329789B2 (enExample)
BR (1) BR112017005104B1 (enExample)
CA (1) CA2957868C (enExample)
EA (1) EA201790796A8 (enExample)
IL (1) IL250823A0 (enExample)
MX (1) MX2017004652A (enExample)
SG (1) SG11201701184WA (enExample)
WO (2) WO2016055792A1 (enExample)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3204388B1 (en) 2014-10-10 2018-12-12 Pulmocide Limited Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivatives
WO2016097761A1 (en) 2014-12-18 2016-06-23 Pulmocide Limited 4,5-dihydro-6h-thieno[3,2-d]benzazepine derivatives and their use to treat respiratory syncytial virus (rsv) infections
RU2738232C2 (ru) 2015-07-22 2020-12-09 Энанта Фармасьютикалс, Инк. Производные бензодиазепина как ингибиторы rsv
EP3402799B1 (en) 2016-01-15 2022-05-04 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
KR20180108598A (ko) * 2016-02-03 2018-10-04 얀센 사이언시즈 아일랜드 유씨 Rsv의 치료를 위한 조합 생성물
WO2017175000A1 (en) * 2016-04-08 2017-10-12 Pulmocide Limited Compounds
WO2018129287A1 (en) 2017-01-06 2018-07-12 Enanta Pharmaceuticals, Inc. Heteroaryldiazepine derivatives as rsv inhibitors
MX379326B (es) 2017-02-16 2025-03-11 Enanta Pharm Inc Procesos para la preparación de derivados de benzodiazepina
WO2018226801A1 (en) 2017-06-07 2018-12-13 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as rsv inhibitors
WO2019006291A1 (en) * 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
WO2019006295A1 (en) * 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
AU2018339068B2 (en) 2017-09-29 2022-12-15 Enanta Pharmaceuticals, Inc. Combination pharmaceutical agents as RSV inhibitors
CN111343990B (zh) 2017-11-13 2023-08-04 英安塔制药有限公司 苯并二氮杂䓬-2-酮和苯并氮杂䓬-2-酮衍生物的拆分方法
US10647711B2 (en) 2017-11-13 2020-05-12 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as RSV inhibitors
WO2019199908A1 (en) * 2018-04-11 2019-10-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
PH12021552201A1 (en) 2019-03-18 2022-05-30 Enanta Pharm Inc Benzodiazepine derivatives as rsv inhibitors
US11179400B2 (en) 2019-04-09 2021-11-23 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
TWI864048B (zh) 2019-10-04 2024-12-01 美商安塔製藥公司 抗病毒雜環化合物、其醫藥組成物及其用途
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
US11534439B2 (en) 2020-07-07 2022-12-27 Enanta Pharmaceuticals, Inc. Dihydroquinoxaline and dihydropyridopyrazine derivatives as RSV inhibitors
WO2022086840A1 (en) 2020-10-19 2022-04-28 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents
JP2024507561A (ja) 2021-02-26 2024-02-20 エナンタ ファーマシューティカルズ インコーポレイテッド 抗ウイルス複素環式化合物
AR129003A1 (es) 2022-04-07 2024-07-03 Enanta Pharm Inc Compuestos heterocíclicos antivirales
WO2023211997A1 (en) 2022-04-27 2023-11-02 Enanta Pharmaceuticals, Inc. Antiviral compounds

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5693635A (en) 1993-07-29 1997-12-02 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
KR100693771B1 (ko) 1999-04-28 2007-03-12 사노피-아벤티스 도이칠란트 게엠베하 Ppar 수용체 리간드로서의 트리아릴 산 유도체 및 이를 포함하는 약제학적 조성물
CA2711644A1 (en) * 2008-01-07 2009-07-16 Synta Pharmaceuticals Corp. Compounds for inflammation and immune-related uses
US8999969B2 (en) 2009-07-09 2015-04-07 Gilead Sciences, Inc. Anti-RSV compounds
CN102656141B (zh) 2009-10-13 2016-04-06 利亘制药公司 模拟造血生长因子的小分子化合物及其用途
CA2806341C (en) 2010-07-29 2020-03-24 Rigel Pharmaceuticals, Inc. Ampk-activating heterocyclic compounds and methods for using the same
US9464065B2 (en) 2011-03-24 2016-10-11 The Scripps Research Institute Compounds and methods for inducing chondrogenesis
AU2015301334A1 (en) 2014-08-05 2017-02-23 Alios Biopharma, Inc. Combination therapy for treating a paramyxovirus
EP3204388B1 (en) * 2014-10-10 2018-12-12 Pulmocide Limited Novel 5,6-dihydro-4h-benzo[b]thieno-[2,3-d]azepine derivatives
EP3402799B1 (en) 2016-01-15 2022-05-04 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
KR20180108598A (ko) 2016-02-03 2018-10-04 얀센 사이언시즈 아일랜드 유씨 Rsv의 치료를 위한 조합 생성물
WO2019006295A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
WO2019006291A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS

Similar Documents

Publication Publication Date Title
JP2017531039A5 (enExample)
JP5911638B2 (ja) ベンゾチアゾール−6−イル酢酸誘導体およびhiv感染を処置するためのそれらの使用
AU2018254577B2 (en) Combination therapies with EHMT2 inhibitors
AU2011367809B2 (en) Piperidine derivatives and compositions for the inhibition of nicotinamide phosphoribosyltransferase (NAMPT)
ES2620612T3 (es) Derivados de sulfóxidos y sulfonas de piridinilo y pirimidinilo
JP2009529047A5 (enExample)
AU2013345107B2 (en) Heteroaromatic compounds as PI3 kinase modulators and methods of use
CA2954488C (en) Pyridone derivative having tetrahydropyranylmethyl group
JP2020514267A5 (enExample)
HRP20191268T1 (hr) Derivati tieno[2,3-c]pirol-4-ona kao inhibitori erk
KR20140062120A (ko) 키나아제 저해제로서의 벤조니트릴 유도체
CA3198809A1 (en) Heterocyclic spiro compounds and methods of use
RU2018134981A (ru) Конъюгаты, содержащие ингибиторы RIPK2
AU2009266090A1 (en) Pyrrolopyridinylpyrimidin-2-ylamine derivatives
US9364482B2 (en) Substituted benzofuran compounds and methods of use thereof for the treatment of viral diseases
AU2021370660A1 (en) Heterocyclic spiro compounds and methods of use
AU2012342891A1 (en) 3-Cyanoaryl-1H-pyrrolo[2.3-b]pyridine derivatives
JP2016517877A5 (enExample)
KR20250081951A (ko) 금속 채널 활성화제를 포함하는 병용 요법
US20160108049A1 (en) Novel Phthalazinone-Pyrrolopyrimidinecarboxamide Derivatives
CN114341125A (zh) Trex1调节剂
RU2014127984A (ru) Хинолиновые производные как ингибиторы фермента pde10a
CA3005921C (en) Substituted-(pyrrolo[2,3-b]pyridin-3-yl)-pyrimidin derivatives and use thereof as inhibitors of influenza virus replication
WO2024022481A1 (zh) 苯基取代的二氢萘啶类化合物及其制备与用途
HK40023961A (en) Novel benzoimidazoles as selective inhibitors of indoleamine 2, 3-dioxygenases