JP2017516772A5 - - Google Patents

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Publication number
JP2017516772A5
JP2017516772A5 JP2016568812A JP2016568812A JP2017516772A5 JP 2017516772 A5 JP2017516772 A5 JP 2017516772A5 JP 2016568812 A JP2016568812 A JP 2016568812A JP 2016568812 A JP2016568812 A JP 2016568812A JP 2017516772 A5 JP2017516772 A5 JP 2017516772A5
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JP
Japan
Prior art keywords
dodeca
oxo
triazatricyclo
trifluoromethyl
tetraen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2016568812A
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English (en)
Japanese (ja)
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JP6580074B2 (ja
JP2017516772A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2015/061468 external-priority patent/WO2015177367A1/en
Publication of JP2017516772A publication Critical patent/JP2017516772A/ja
Publication of JP2017516772A5 publication Critical patent/JP2017516772A5/ja
Application granted granted Critical
Publication of JP6580074B2 publication Critical patent/JP6580074B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2016568812A 2014-05-23 2015-05-22 S100阻害薬として有用な新規化合物 Expired - Fee Related JP6580074B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14169757.3 2014-05-23
EP14169757 2014-05-23
PCT/EP2015/061468 WO2015177367A1 (en) 2014-05-23 2015-05-22 Novel compounds useful as s100-inhibitors

Publications (3)

Publication Number Publication Date
JP2017516772A JP2017516772A (ja) 2017-06-22
JP2017516772A5 true JP2017516772A5 (OSRAM) 2018-05-10
JP6580074B2 JP6580074B2 (ja) 2019-09-25

Family

ID=50774707

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016568812A Expired - Fee Related JP6580074B2 (ja) 2014-05-23 2015-05-22 S100阻害薬として有用な新規化合物

Country Status (12)

Country Link
US (1) US9771372B2 (OSRAM)
EP (1) EP2991990B1 (OSRAM)
JP (1) JP6580074B2 (OSRAM)
KR (1) KR20170005868A (OSRAM)
CN (1) CN106414448B (OSRAM)
AU (1) AU2015261775B2 (OSRAM)
BR (1) BR112016024749A2 (OSRAM)
CA (1) CA2948436A1 (OSRAM)
EA (1) EA030604B1 (OSRAM)
ES (1) ES2620751T3 (OSRAM)
MX (1) MX2016014483A (OSRAM)
WO (1) WO2015177367A1 (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019208290A1 (ja) 2018-04-27 2019-10-31 国立大学法人 岡山大学 抗s100a8/a9抗体とその用途
US11197908B2 (en) 2018-07-17 2021-12-14 The Board Of Trustees Of The University Of Arkansas Peptoids and methods for attenuating inflammatory response
CN114555119A (zh) 2019-10-30 2022-05-27 国立大学法人冈山大学 炎症性肺疾病的预防和/或治疗剂
WO2023209141A1 (en) 2022-04-29 2023-11-02 Westfälische Wilhelms-Universität Münster Benzo[d]imidazo[1,2-a]imidazoles and their use in diagnosis
WO2025132458A1 (en) 2023-12-18 2025-06-26 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6248755B1 (en) 1999-04-06 2001-06-19 Merck & Co., Inc. Pyrrolidine modulators of chemokine receptor activity
AR029489A1 (es) 2000-03-10 2003-07-02 Euro Celtique Sa Piridinas, pirimidinas, pirazinas, triazinas sustituidas por arilo, composiciones farmaceuticas y el uso de las mismas para la manufactura de un medicamento
US7361678B2 (en) * 2002-03-05 2008-04-22 Transtech Pharma, Inc. Azole derivatives and fused bicyclic azole derivatives as therapeutic agents
DE60125373T2 (de) 2000-07-26 2007-10-18 Smithkline Beecham P.L.C., Brentford Aminopiperidin chinoline und ihre azaisosteren analoga mit antibakterieller wirkung
AU2002245590B2 (en) * 2001-03-05 2006-06-29 Transtech Pharma, Inc. Benzimidazole derivatives as therapeutic agents
GB0117506D0 (en) 2001-07-18 2001-09-12 Bayer Ag Imidazopyridinones
SE0104331D0 (sv) 2001-12-19 2001-12-19 Astrazeneca Ab Novel compounds
US20060111416A1 (en) 2004-11-24 2006-05-25 Lane Charlotte A L Octahydropyrrolo[3,4-C]pyrrole derivatives
US8088767B2 (en) 2006-09-28 2012-01-03 Exelixis, Inc. JAK-2 modulators and methods of use
US7919498B2 (en) 2007-03-23 2011-04-05 Amgen Inc. Substituted pyrazolo[3,4-d]pyrimidines as PI3K inhibitors
EP1986009A1 (en) * 2007-04-26 2008-10-29 Active Biotech AB Screening method
CA2689980A1 (en) 2007-06-13 2008-12-24 Glaxosmithkline Llc Farnesoid x receptor agonists
WO2009093747A1 (en) * 2008-01-22 2009-07-30 Takeda Pharmaceutical Company Limited Tricyclic compounds having corticotropin-releasing factor antagonistic activity and pharmaceutical compositions containing them
TW201004941A (en) 2008-07-16 2010-02-01 Wyeth Corp Alpha7 nicotinic acetylcholine receptor inhibitors
WO2010101949A1 (en) 2009-03-02 2010-09-10 Sirtris Pharmaceuticals, Inc. 8-substituted quinolines and related analogs as sirtuin modulators
ES2552514T3 (es) 2011-11-03 2015-11-30 Hoffmann-La Roche Ag Compuestos bicíclicos de piperazina
GB201321728D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents

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