JP2017504590A5 - - Google Patents
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- Publication number
- JP2017504590A5 JP2017504590A5 JP2016538745A JP2016538745A JP2017504590A5 JP 2017504590 A5 JP2017504590 A5 JP 2017504590A5 JP 2016538745 A JP2016538745 A JP 2016538745A JP 2016538745 A JP2016538745 A JP 2016538745A JP 2017504590 A5 JP2017504590 A5 JP 2017504590A5
- Authority
- JP
- Japan
- Prior art keywords
- composition
- eudragit
- item
- linaclotide
- use according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021078445A JP7483656B2 (ja) | 2013-12-11 | 2021-05-06 | リナクロチドの遅延放出組成物 |
| JP2023115832A JP2023126475A (ja) | 2013-12-11 | 2023-07-14 | リナクロチドの遅延放出組成物 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361914951P | 2013-12-11 | 2013-12-11 | |
| US201361914952P | 2013-12-11 | 2013-12-11 | |
| US61/914,951 | 2013-12-11 | ||
| US61/914,952 | 2013-12-11 | ||
| PCT/US2014/069838 WO2015089326A1 (en) | 2013-12-11 | 2014-12-11 | Delayed release compositions of linaclotide |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019029432A Division JP2019073559A (ja) | 2013-12-11 | 2019-02-21 | リナクロチドの遅延放出組成物 |
| JP2021078445A Division JP7483656B2 (ja) | 2013-12-11 | 2021-05-06 | リナクロチドの遅延放出組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017504590A JP2017504590A (ja) | 2017-02-09 |
| JP2017504590A5 true JP2017504590A5 (enExample) | 2018-01-25 |
| JP6964380B2 JP6964380B2 (ja) | 2021-11-10 |
Family
ID=52293217
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016538745A Expired - Fee Related JP6964380B2 (ja) | 2013-12-11 | 2014-12-11 | リナクロチドの遅延放出組成物 |
| JP2019029432A Pending JP2019073559A (ja) | 2013-12-11 | 2019-02-21 | リナクロチドの遅延放出組成物 |
| JP2021078445A Active JP7483656B2 (ja) | 2013-12-11 | 2021-05-06 | リナクロチドの遅延放出組成物 |
| JP2023115832A Pending JP2023126475A (ja) | 2013-12-11 | 2023-07-14 | リナクロチドの遅延放出組成物 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019029432A Pending JP2019073559A (ja) | 2013-12-11 | 2019-02-21 | リナクロチドの遅延放出組成物 |
| JP2021078445A Active JP7483656B2 (ja) | 2013-12-11 | 2021-05-06 | リナクロチドの遅延放出組成物 |
| JP2023115832A Pending JP2023126475A (ja) | 2013-12-11 | 2023-07-14 | リナクロチドの遅延放出組成物 |
Country Status (29)
| Country | Link |
|---|---|
| US (7) | US20160310560A1 (enExample) |
| EP (2) | EP3079669B1 (enExample) |
| JP (4) | JP6964380B2 (enExample) |
| KR (3) | KR102509291B1 (enExample) |
| CN (3) | CN112569199A (enExample) |
| AU (3) | AU2014362220B2 (enExample) |
| CA (1) | CA2933587C (enExample) |
| CL (1) | CL2016001424A1 (enExample) |
| CY (1) | CY1123953T1 (enExample) |
| DK (1) | DK3079669T3 (enExample) |
| EA (1) | EA201691216A1 (enExample) |
| EC (2) | ECSP16059106A (enExample) |
| ES (1) | ES2838007T3 (enExample) |
| HR (1) | HRP20201753T1 (enExample) |
| HU (1) | HUE052981T2 (enExample) |
| IL (2) | IL246155A0 (enExample) |
| LT (1) | LT3079669T (enExample) |
| MX (2) | MX386584B (enExample) |
| NZ (2) | NZ759512A (enExample) |
| PE (2) | PE20211976A1 (enExample) |
| PH (1) | PH12016501122B1 (enExample) |
| PL (1) | PL3079669T3 (enExample) |
| PT (1) | PT3079669T (enExample) |
| RS (1) | RS61133B1 (enExample) |
| SG (2) | SG11201604729QA (enExample) |
| SI (1) | SI3079669T1 (enExample) |
| SM (1) | SMT202000686T1 (enExample) |
| UA (1) | UA119335C2 (enExample) |
| WO (2) | WO2015089326A1 (enExample) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA119335C2 (uk) * | 2013-12-11 | 2019-06-10 | Айронвуд Фармасьютикалз, Інк. | Композиції лінаклотиду з затриманим вивільненням |
| WO2016020901A1 (en) | 2014-08-07 | 2016-02-11 | Acerta Pharma B.V. | Methods of treating cancers, immune and autoimmune diseases, and inflammatory diseases based on btk occupancy and btk resynthesis rate |
| CA3018328A1 (en) | 2014-10-31 | 2016-04-30 | Purdue Pharma | Methods and compositions particularly for treatment of attention deficit disorder |
| WO2016125064A1 (en) * | 2015-02-02 | 2016-08-11 | Aurobindo Pharma Ltd | Stable compositions comprising linaclotide |
| JP2018516937A (ja) * | 2015-06-05 | 2018-06-28 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | リナクロチドの改変または標的放出製剤 |
| US10588864B2 (en) | 2016-03-11 | 2020-03-17 | Gateway Pharmaceuticals LLC | Pharmaceutical compositions for colon-specific delivery |
| WO2017156214A1 (en) * | 2016-03-11 | 2017-09-14 | Gateway Pharmaceutical LLC | Pharmaceutical compositions for colon-specific delivery |
| US11534404B2 (en) * | 2016-10-06 | 2022-12-27 | Sucampo Ag | Multilayer beads for pharmaceutical use |
| CN110475564A (zh) * | 2016-12-21 | 2019-11-19 | 硬木药品公司 | 用利那洛肽的修饰的或延迟释放制剂治疗肠易激综合征的方法 |
| KR102227486B1 (ko) * | 2017-06-30 | 2021-03-12 | 롯데정밀화학 주식회사 | 프로톤 펌프 저해제를 포함하는 경구용 고형제제 조성물, 이를 포함하는 경구용 고형제제 및 그 제조방법 |
| EA202092275A1 (ru) * | 2018-03-23 | 2021-02-09 | Палатин Текнолоджиз, Инк. | Составы пептидов, специфичных к рецептору меланокортина, и способы доставки в желудочно-кишечный тракт |
| US10722473B2 (en) | 2018-11-19 | 2020-07-28 | Purdue Pharma L.P. | Methods and compositions particularly for treatment of attention deficit disorder |
| CN114206324A (zh) * | 2019-06-10 | 2022-03-18 | 硬木药品公司 | 治疗与腹泻占主导的肠易激综合征相关的腹部疼痛 |
| KR102104507B1 (ko) * | 2019-08-23 | 2020-04-24 | 브릿지바이오테라퓨틱스(주) | 팔미토일-l-프롤릴-l-프롤릴-글리실-l-타이로신 나트륨을 포함하는 약제학적 제제 및 이의 제조방법 |
| CN110935007B (zh) * | 2019-12-12 | 2023-06-23 | 烟台大学 | 利那洛肽复方组合物、制剂及其用途和制备方法 |
| GB202017863D0 (en) * | 2020-11-12 | 2020-12-30 | Intract Pharma Ltd | Novel compositions |
| CN115105582A (zh) * | 2021-03-17 | 2022-09-27 | 江苏豪森药业集团有限公司 | 一种含利那洛肽或其盐的药物组合物及其制备方法 |
| WO2022245650A1 (en) * | 2021-05-19 | 2022-11-24 | Alberto Paz | Orally administered compositions for cancer treatment |
| IL319961A (en) * | 2022-10-03 | 2025-05-01 | Brim Biotechnology Inc | Preparations including PEDF-derived short peptides (PDSP) and their uses |
| TW202440065A (zh) * | 2022-12-28 | 2024-10-16 | 日商中外製藥股份有限公司 | 包含分散對象物質的固體分散體、包含其之醫藥組合物及其製造方法 |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7304036B2 (en) | 2003-01-28 | 2007-12-04 | Microbia, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| US7371727B2 (en) | 2003-01-28 | 2008-05-13 | Microbia, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| CN201252259Y (zh) * | 2008-07-24 | 2009-06-03 | 富士康(昆山)电脑接插件有限公司 | 电连接器 |
| RS60101B1 (sr) * | 2008-08-15 | 2020-05-29 | Ironwood Pharmaceuticals Inc | Formulacije koje sadrže linaklotid za oralnu primenu |
| JP5964589B2 (ja) * | 2008-12-03 | 2016-08-03 | シナジー ファーマシューティカルズ インコーポレイテッド | グアニル酸シクラーゼcアゴニストの製剤およびその使用方法 |
| US20130012454A1 (en) * | 2009-07-06 | 2013-01-10 | Ironwood Pharmaceuticals, Inc. | Orally Disintegrating Compositions of Linaclotide |
| WO2011019819A1 (en) * | 2009-08-12 | 2011-02-17 | Forest Laboratories Holdings Limited | Orally disintegrating compositions of linaclotide |
| US8748573B2 (en) * | 2009-08-06 | 2014-06-10 | Ironwood Pharmaceuticals, Inc. | Formulations comprising linaclotide |
| RU2012109415A (ru) * | 2009-08-13 | 2013-09-20 | Айронвуд Фармасьютикалз, Инк. | Способ модуляции фармакодинамического эффекта перорально вводимых агонистов рецептора гуанилатциклазы |
| CA2790213A1 (en) * | 2010-02-17 | 2011-08-25 | Ironwood Pharmaceuticals, Inc. | Treatments for gastrointestinal disorders |
| ES2763404T3 (es) * | 2010-08-11 | 2020-05-28 | Ironwood Pharmaceuticals Inc | Formulaciones estables de linaclotida |
| US20140162963A1 (en) * | 2010-09-11 | 2014-06-12 | Forest Laboratories Holdings Limited | Treatment of Constipation-Predominant Irritable Bowel Syndrome |
| JP2012155108A (ja) * | 2011-01-26 | 2012-08-16 | Kyocera Document Solutions Inc | 現像ローラ、現像装置および画像形成装置 |
| CN104053449B (zh) * | 2011-08-17 | 2016-12-07 | 硬木药品公司 | 胃肠疾患的治疗 |
| WO2013047795A1 (ja) * | 2011-09-30 | 2013-04-04 | アステラス製薬株式会社 | 粒子状医薬組成物 |
| JP2016521249A (ja) * | 2012-07-12 | 2016-07-21 | フォレスト ラボラトリーズ ホールディングス リミテッド | リナクロチド組成物 |
| EP2958577A2 (en) * | 2013-02-25 | 2015-12-30 | Synergy Pharmaceuticals Inc. | Guanylate cyclase receptor agonists for use in colonic cleansing |
| UA119335C2 (uk) * | 2013-12-11 | 2019-06-10 | Айронвуд Фармасьютикалз, Інк. | Композиції лінаклотиду з затриманим вивільненням |
-
2014
- 2014-11-12 UA UAA201607434A patent/UA119335C2/uk unknown
- 2014-12-11 PE PE2021000748A patent/PE20211976A1/es unknown
- 2014-12-11 NZ NZ759512A patent/NZ759512A/en unknown
- 2014-12-11 EP EP14824655.6A patent/EP3079669B1/en active Active
- 2014-12-11 WO PCT/US2014/069838 patent/WO2015089326A1/en not_active Ceased
- 2014-12-11 SM SM20200686T patent/SMT202000686T1/it unknown
- 2014-12-11 PH PH1/2016/501122A patent/PH12016501122B1/en unknown
- 2014-12-11 KR KR1020217039962A patent/KR102509291B1/ko active Active
- 2014-12-11 PT PT148246556T patent/PT3079669T/pt unknown
- 2014-12-11 KR KR1020237008167A patent/KR20230039764A/ko not_active Ceased
- 2014-12-11 CN CN202011156517.1A patent/CN112569199A/zh active Pending
- 2014-12-11 DK DK14824655.6T patent/DK3079669T3/da active
- 2014-12-11 RS RS20201435A patent/RS61133B1/sr unknown
- 2014-12-11 HR HRP20201753TT patent/HRP20201753T1/hr unknown
- 2014-12-11 NZ NZ721952A patent/NZ721952A/en unknown
- 2014-12-11 CN CN202210517834.4A patent/CN115089556A/zh active Pending
- 2014-12-11 CN CN201480075352.1A patent/CN106659687A/zh active Pending
- 2014-12-11 US US15/103,634 patent/US20160310560A1/en not_active Abandoned
- 2014-12-11 SG SG11201604729QA patent/SG11201604729QA/en unknown
- 2014-12-11 KR KR1020167018606A patent/KR102337809B1/ko active Active
- 2014-12-11 SI SI201431715T patent/SI3079669T1/sl unknown
- 2014-12-11 EA EA201691216A patent/EA201691216A1/ru unknown
- 2014-12-11 CA CA2933587A patent/CA2933587C/en active Active
- 2014-12-11 AU AU2014362220A patent/AU2014362220B2/en not_active Ceased
- 2014-12-11 ES ES14824655T patent/ES2838007T3/es active Active
- 2014-12-11 WO PCT/US2014/069851 patent/WO2015089335A1/en not_active Ceased
- 2014-12-11 US US15/103,616 patent/US20160310559A1/en not_active Abandoned
- 2014-12-11 EP EP20198666.8A patent/EP3821881A1/en active Pending
- 2014-12-11 PE PE2016000804A patent/PE20161373A1/es unknown
- 2014-12-11 PL PL14824655T patent/PL3079669T3/pl unknown
- 2014-12-11 HU HUE14824655A patent/HUE052981T2/hu unknown
- 2014-12-11 JP JP2016538745A patent/JP6964380B2/ja not_active Expired - Fee Related
- 2014-12-11 LT LTEP14824655.6T patent/LT3079669T/lt unknown
- 2014-12-11 SG SG10201804817TA patent/SG10201804817TA/en unknown
- 2014-12-11 MX MX2016007625A patent/MX386584B/es unknown
-
2016
- 2016-06-09 IL IL246155A patent/IL246155A0/en unknown
- 2016-06-10 MX MX2021011906A patent/MX2021011906A/es unknown
- 2016-06-10 CL CL2016001424A patent/CL2016001424A1/es unknown
- 2016-07-08 EC ECIEPI201659106A patent/ECSP16059106A/es unknown
-
2017
- 2017-02-17 US US15/435,701 patent/US20170157200A1/en not_active Abandoned
- 2017-09-28 US US15/718,075 patent/US20180015139A1/en not_active Abandoned
-
2019
- 2019-02-21 JP JP2019029432A patent/JP2019073559A/ja active Pending
- 2019-09-11 US US16/567,082 patent/US20200038476A1/en not_active Abandoned
-
2020
- 2020-04-01 AU AU2020202319A patent/AU2020202319B2/en not_active Ceased
- 2020-11-26 CY CY20201101128T patent/CY1123953T1/el unknown
-
2021
- 2021-05-06 JP JP2021078445A patent/JP7483656B2/ja active Active
- 2021-05-06 IL IL283012A patent/IL283012A/en unknown
- 2021-09-28 EC ECSENADI202172161A patent/ECSP21072161A/es unknown
- 2021-10-18 US US17/503,601 patent/US20220031802A1/en not_active Abandoned
-
2022
- 2022-03-18 AU AU2022201891A patent/AU2022201891A1/en not_active Abandoned
-
2023
- 2023-07-14 JP JP2023115832A patent/JP2023126475A/ja active Pending
- 2023-11-09 US US18/505,414 patent/US20240075094A1/en not_active Abandoned
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