CN112569199A - 利那洛肽的延迟释放组合物 - Google Patents

利那洛肽的延迟释放组合物 Download PDF

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Publication number
CN112569199A
CN112569199A CN202011156517.1A CN202011156517A CN112569199A CN 112569199 A CN112569199 A CN 112569199A CN 202011156517 A CN202011156517 A CN 202011156517A CN 112569199 A CN112569199 A CN 112569199A
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CN
China
Prior art keywords
composition
linaclotide
composition comprises
eudragit
weight
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN202011156517.1A
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English (en)
Chinese (zh)
Inventor
A.弗雷岑
M.G.卡里
A.哈沙什
M.德迪亚
Y.莫
A.齐赫特里
M.米勒
R.桑维
M.M.巴里
A.格里尔
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Elastagen Pty Ltd
Ironwood Pharmaceuticals Inc
Original Assignee
Forest Laboratories Holdings ULC
Ironwood Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52293217&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN112569199(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Forest Laboratories Holdings ULC, Ironwood Pharmaceuticals Inc filed Critical Forest Laboratories Holdings ULC
Publication of CN112569199A publication Critical patent/CN112569199A/zh
Pending legal-status Critical Current

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    • A61K38/10—Peptides having 12 to 20 amino acids
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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nutrition Science (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
CN202011156517.1A 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物 Pending CN112569199A (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361914951P 2013-12-11 2013-12-11
US201361914952P 2013-12-11 2013-12-11
US61/914952 2013-12-11
US61/914951 2013-12-11
CN201480075352.1A CN106659687A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CN201480075352.1A Division CN106659687A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物

Publications (1)

Publication Number Publication Date
CN112569199A true CN112569199A (zh) 2021-03-30

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ID=52293217

Family Applications (3)

Application Number Title Priority Date Filing Date
CN202011156517.1A Pending CN112569199A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物
CN202210517834.4A Pending CN115089556A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物
CN201480075352.1A Pending CN106659687A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物

Family Applications After (2)

Application Number Title Priority Date Filing Date
CN202210517834.4A Pending CN115089556A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物
CN201480075352.1A Pending CN106659687A (zh) 2013-12-11 2014-12-11 利那洛肽的延迟释放组合物

Country Status (29)

Country Link
US (7) US20160310559A1 (enExample)
EP (2) EP3079669B1 (enExample)
JP (4) JP6964380B2 (enExample)
KR (3) KR102337809B1 (enExample)
CN (3) CN112569199A (enExample)
AU (3) AU2014362220B2 (enExample)
CA (1) CA2933587C (enExample)
CL (1) CL2016001424A1 (enExample)
CY (1) CY1123953T1 (enExample)
DK (1) DK3079669T3 (enExample)
EA (1) EA201691216A1 (enExample)
EC (2) ECSP16059106A (enExample)
ES (1) ES2838007T3 (enExample)
HR (1) HRP20201753T1 (enExample)
HU (1) HUE052981T2 (enExample)
IL (2) IL246155A0 (enExample)
LT (1) LT3079669T (enExample)
MX (2) MX386584B (enExample)
NZ (2) NZ721952A (enExample)
PE (2) PE20211976A1 (enExample)
PH (1) PH12016501122B1 (enExample)
PL (1) PL3079669T3 (enExample)
PT (1) PT3079669T (enExample)
RS (1) RS61133B1 (enExample)
SG (2) SG10201804817TA (enExample)
SI (1) SI3079669T1 (enExample)
SM (1) SMT202000686T1 (enExample)
UA (1) UA119335C2 (enExample)
WO (2) WO2015089335A1 (enExample)

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CA2902911C (en) 2014-10-31 2017-06-27 Purdue Pharma Methods and compositions particularly for treatment of attention deficit disorder
US20180008547A1 (en) * 2015-02-02 2018-01-11 Aurobindo Pharma Ltd Stable Compositions comprising Linaclotide
EP3302440B1 (en) * 2015-06-05 2021-01-06 Ironwood Pharmaceuticals, Inc. Modified or targeted release formulations of linaclotide
US10588864B2 (en) 2016-03-11 2020-03-17 Gateway Pharmaceuticals LLC Pharmaceutical compositions for colon-specific delivery
WO2017156214A1 (en) * 2016-03-11 2017-09-14 Gateway Pharmaceutical LLC Pharmaceutical compositions for colon-specific delivery
WO2018065826A1 (en) * 2016-10-06 2018-04-12 Sucampo Ag Multilayer beads for pharmaceutical use
MA47112A (fr) * 2016-12-21 2019-10-30 Ironwood Pharmaceuticals Inc Procédés de traitement du syndrome du côlon irritable avec des formulations à libération modifiée ou retardée de linaclotide
KR102227486B1 (ko) * 2017-06-30 2021-03-12 롯데정밀화학 주식회사 프로톤 펌프 저해제를 포함하는 경구용 고형제제 조성물, 이를 포함하는 경구용 고형제제 및 그 제조방법
WO2019183472A1 (en) * 2018-03-23 2019-09-26 Palatin Technologies, Inc. Melanocortin receptor-specific peptide formulations and methods for gastrointestinal tract-specific delivery
US10722473B2 (en) 2018-11-19 2020-07-28 Purdue Pharma L.P. Methods and compositions particularly for treatment of attention deficit disorder
US20220241367A1 (en) * 2019-06-10 2022-08-04 Ironwood Pharmaceutical, Inc. Treatment of Abdominal Pain Associated with Diarrhea-Predominant Irritable Bowel Syndrome
KR102104507B1 (ko) * 2019-08-23 2020-04-24 브릿지바이오테라퓨틱스(주) 팔미토일-l-프롤릴-l-프롤릴-글리실-l-타이로신 나트륨을 포함하는 약제학적 제제 및 이의 제조방법
CN110935007B (zh) * 2019-12-12 2023-06-23 烟台大学 利那洛肽复方组合物、制剂及其用途和制备方法
GB202017863D0 (en) * 2020-11-12 2020-12-30 Intract Pharma Ltd Novel compositions
EP4340838A4 (en) * 2021-05-19 2025-04-16 Alberto Paz ORALLY ADMINISTERED COMPOSITIONS FOR CANCER TREATMENT
AU2023356242A1 (en) * 2022-10-03 2025-04-24 Brim Biotechnology, Inc. Compositions comprising pedf-derived short peptides (pdsp) and uses thereof
CN120418354A (zh) * 2022-12-28 2025-08-01 中外制药株式会社 含有待分散的物质的固体分散体、含有其的药物组合物及其生产方法

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