JP2016538262A - 抗菌剤を含む医薬品組成物 - Google Patents
抗菌剤を含む医薬品組成物 Download PDFInfo
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- JP2016538262A JP2016538262A JP2016525559A JP2016525559A JP2016538262A JP 2016538262 A JP2016538262 A JP 2016538262A JP 2016525559 A JP2016525559 A JP 2016525559A JP 2016525559 A JP2016525559 A JP 2016525559A JP 2016538262 A JP2016538262 A JP 2016538262A
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- Prior art keywords
- pharmaceutically acceptable
- acceptable derivative
- compound
- formula
- imipenem
- Prior art date
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Hydrogenated Pyridines (AREA)
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|---|---|---|---|
| IN3308/MUM/2013 | 2013-10-22 | ||
| PCT/IB2014/065521 WO2015059642A1 (en) | 2013-10-22 | 2014-10-22 | Pharmaceutical compositions comprising antibacterial agents |
| IN3308MU2013 IN2013MU03308A (enrdf_load_stackoverflow) | 2013-10-22 | 2014-10-22 |
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| JP2016538262A true JP2016538262A (ja) | 2016-12-08 |
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| JP2016525559A Pending JP2016538262A (ja) | 2013-10-22 | 2014-10-22 | 抗菌剤を含む医薬品組成物 |
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Families Citing this family (3)
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| WO2018193368A1 (en) * | 2017-04-18 | 2018-10-25 | Wockhardt Limited | Antibacterial compositions |
| US11905286B2 (en) | 2018-08-09 | 2024-02-20 | Antabio Sas | Diazabicyclooctanones as inhibitors of serine beta-lactamases |
| IL280770B2 (en) | 2018-08-09 | 2024-05-01 | Antabio Sas | Diazabicyclooctanones as inhibitors of serine beta-lactamases |
Citations (1)
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| WO2013038330A1 (en) * | 2011-09-13 | 2013-03-21 | Wockhardt Limited | Nitrogen containing compounds and their use |
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| KR101590739B1 (ko) * | 2005-09-22 | 2016-02-01 | 메이지 세이카 파루마 가부시키가이샤 | 메탈로-β-락타마제 저해제 |
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2014
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- 2014-10-22 JP JP2016525559A patent/JP2016538262A/ja active Pending
- 2014-10-22 EP EP14806073.4A patent/EP3060208B1/en not_active Not-in-force
- 2014-10-22 CA CA2928358A patent/CA2928358A1/en not_active Abandoned
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- 2014-10-22 MX MX2016005160A patent/MX2016005160A/es unknown
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- 2014-10-22 RU RU2016115374A patent/RU2016115374A/ru not_active Application Discontinuation
- 2014-10-22 CN CN201480069849.2A patent/CN106132411A/zh active Pending
- 2014-10-22 US US15/030,310 patent/US9789097B2/en not_active Expired - Fee Related
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013038330A1 (en) * | 2011-09-13 | 2013-03-21 | Wockhardt Limited | Nitrogen containing compounds and their use |
Non-Patent Citations (4)
| Title |
|---|
| DIAGNOSTIC MICROBIOLOGY AND INFECTIOUS DISEASE, vol. 63, no. 4, JPN5016010997, 2009, pages 426 - 433 * |
| PHARMACOTHERAPY, vol. 30, no. 4, JPN5016010995, 2010, pages 354 - 360 * |
| 日薬理誌, vol. Vol.107, JPN6018024982, 1996, pages 53 - 66 * |
| 第十四改正日本薬局方解説書, JPN6018024981, 2001, pages C-273〜C-275 * |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2928358A1 (en) | 2015-04-30 |
| RU2016115374A (ru) | 2017-11-28 |
| MX2016005160A (es) | 2016-10-05 |
| CN106132411A (zh) | 2016-11-16 |
| EP3060208A1 (en) | 2016-08-31 |
| RU2016115374A3 (enrdf_load_stackoverflow) | 2018-08-15 |
| EP3060208B1 (en) | 2018-09-19 |
| IN2013MU03308A (enrdf_load_stackoverflow) | 2015-07-17 |
| AU2014338611A1 (en) | 2016-05-12 |
| US9789097B2 (en) | 2017-10-17 |
| US20160303094A1 (en) | 2016-10-20 |
| WO2015059642A1 (en) | 2015-04-30 |
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