JP2016534124A - 代謝並びに体重関連疾患の処置のための組成物および方法 - Google Patents

代謝並びに体重関連疾患の処置のための組成物および方法 Download PDF

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JP2016534124A
JP2016534124A JP2016537878A JP2016537878A JP2016534124A JP 2016534124 A JP2016534124 A JP 2016534124A JP 2016537878 A JP2016537878 A JP 2016537878A JP 2016537878 A JP2016537878 A JP 2016537878A JP 2016534124 A JP2016534124 A JP 2016534124A
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compound
fatostatin
cancer
srebp
alkyl
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JP2016534124A5 (enrdf_load_stackoverflow
Inventor
志成 上杉
志成 上杉
ワキル，サリフ，ジェイ．
アブ−エルヘイガ，ルトフィ
瑞貴 渡邉
瑞貴 渡邉
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Baylor College of Medicine
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Baylor College of Medicine
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Priority claimed from US14/013,918 external-priority patent/US9085566B2/en
Priority claimed from US14/052,074 external-priority patent/US9187485B2/en
Priority claimed from US14/270,130 external-priority patent/US9233941B2/en
Application filed by Baylor College of Medicine filed Critical Baylor College of Medicine
Publication of JP2016534124A publication Critical patent/JP2016534124A/ja
Publication of JP2016534124A5 publication Critical patent/JP2016534124A5/ja
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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JP2016537878A 2013-08-29 2014-08-29 代謝並びに体重関連疾患の処置のための組成物および方法 Pending JP2016534124A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US14/013,918 US9085566B2 (en) 2007-02-02 2013-08-29 Compositions and methods for the treatment of metabolic and related disorders
US14/013,918 2013-08-29
US14/052,074 2013-10-11
US14/052,074 US9187485B2 (en) 2007-02-02 2013-10-11 Methods and compositions for the treatment of cancer and related hyperproliferative disorders
US14/270,130 2014-05-05
US14/270,130 US9233941B2 (en) 2007-02-02 2014-05-05 Methods and compositions for the treatment of body weight related disorders
PCT/US2014/053334 WO2015031710A1 (en) 2013-08-29 2014-08-29 Compositions and methods for the treatment of metabolic and body weight related disorders

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JP2016534124A true JP2016534124A (ja) 2016-11-04
JP2016534124A5 JP2016534124A5 (enrdf_load_stackoverflow) 2017-10-12

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AU (1) AU2014312227A1 (enrdf_load_stackoverflow)
CA (1) CA2922703A1 (enrdf_load_stackoverflow)
WO (1) WO2015031710A1 (enrdf_load_stackoverflow)

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WO2018049080A1 (en) * 2016-09-07 2018-03-15 Fgh Biotech, Inc. Di-substituted pyrazole compounds for the treatment of diseases
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CN112424159B (zh) 2018-07-24 2023-10-31 普罗泰克株式会社 新颖的p62配体化合物及包含其的用于预防、改善或治疗蛋白质构象病的组合物
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