JP2016531886A - 全身性エリテマトーデス及び／または狼瘡腎炎の予防または治療のための方法 - Google Patents

全身性エリテマトーデス及び／または狼瘡腎炎の予防または治療のための方法 Download PDF

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Publication number
JP2016531886A
JP2016531886A JP2016519782A JP2016519782A JP2016531886A JP 2016531886 A JP2016531886 A JP 2016531886A JP 2016519782 A JP2016519782 A JP 2016519782A JP 2016519782 A JP2016519782 A JP 2016519782A JP 2016531886 A JP2016531886 A JP 2016531886A
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JP
Japan
Prior art keywords
compound
treatment
amino
hydrochloride
prevention
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2016519782A
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English (en)
Japanese (ja)
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JP2016531886A5 (OSRAM
Inventor
河村　透
透 河村
靖志 藤谷
靖志 藤谷
瀧澤　正之
正之 瀧澤
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Millennium Pharmaceuticals Inc
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Millennium Pharmaceuticals Inc
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Publication date
Application filed by Millennium Pharmaceuticals Inc filed Critical Millennium Pharmaceuticals Inc
Publication of JP2016531886A publication Critical patent/JP2016531886A/ja
Publication of JP2016531886A5 publication Critical patent/JP2016531886A5/ja
Pending legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2016519782A 2013-10-03 2014-10-02 全身性エリテマトーデス及び／または狼瘡腎炎の予防または治療のための方法 Pending JP2016531886A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361886403P 2013-10-03 2013-10-03
US61/886,403 2013-10-03
PCT/US2014/058738 WO2015051067A1 (en) 2013-10-03 2014-10-02 Method for the prophylaxis or treatment of systemic lupus erythematosus and/or lupus nephritis

Publications (2)

Publication Number Publication Date
JP2016531886A true JP2016531886A (ja) 2016-10-13
JP2016531886A5 JP2016531886A5 (OSRAM) 2017-11-02

Family

ID=51842818

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016519782A Pending JP2016531886A (ja) 2013-10-03 2014-10-02 全身性エリテマトーデス及び／または狼瘡腎炎の予防または治療のための方法

Country Status (10)

Country Link
US (2) US20160250238A1 (OSRAM)
EP (1) EP3052105A1 (OSRAM)
JP (1) JP2016531886A (OSRAM)
KR (1) KR20160058886A (OSRAM)
CN (1) CN105705149A (OSRAM)
BR (1) BR112016007237A2 (OSRAM)
CA (1) CA2925935A1 (OSRAM)
EA (1) EA201690686A1 (OSRAM)
MX (1) MX2016003979A (OSRAM)
WO (1) WO2015051067A1 (OSRAM)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3813817A4 (en) * 2018-06-27 2022-08-10 Algernon Pharmaceuticals Inc. USE OF ACTARIT IN THE PROPHYLAXIS OR TREATMENT OF KIDNEY FIBROSIS OR KIDNEY DISEASE
CN115515578A (zh) * 2020-05-07 2022-12-23 诺罗瑞韦有限公司 用于治疗抑郁症的环丝氨酸和己酮可可碱联合疗法
CN121041156A (zh) * 2025-08-27 2025-12-02 复皙药业(上海)有限公司 含有替普瑞酮的具有祛红功效的膏霜及其制备方法

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010535759A (ja) * 2007-08-06 2010-11-25 ミレニアム・ファーマシューティカルズ・インコーポレイテッド プロテアソーム阻害剤
JP2011524903A (ja) * 2008-06-17 2011-09-08 ミレニアム・ファーマシューティカルズ・インコーポレイテッド ボロン酸エステル化合物およびその医薬組成物
WO2012119056A1 (en) * 2011-03-03 2012-09-07 Cephalon, Inc. Proteasome inhibitor delanzomib for use in the treatment of lupus

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6083903A (en) 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
PT3078667T (pt) 2001-01-25 2018-12-28 The United States Of America Represented By The Sec Dep Of Health And Human Services Formulação de compostos de ácido borónico
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
AR075090A1 (es) 2008-09-29 2011-03-09 Millennium Pharm Inc Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden.
TW201103904A (en) 2009-06-11 2011-02-01 Hoffmann La Roche Janus kinase inhibitor compounds and methods
JP5933523B2 (ja) 2010-03-31 2016-06-08 ミレニアム ファーマシューティカルズ， インコーポレイテッドＭｉｌｌｅｎｎｉｕｍ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ， Ｉｎｃ． １−アミノ−２−シクロプロピルエチルボロン酸の誘導体
MX2013015308A (es) * 2011-06-22 2014-05-20 Cephalon Inc Inhibidores de proteasoma y procesos para su preparacion, purificacion y uso.

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010535759A (ja) * 2007-08-06 2010-11-25 ミレニアム・ファーマシューティカルズ・インコーポレイテッド プロテアソーム阻害剤
JP2011524903A (ja) * 2008-06-17 2011-09-08 ミレニアム・ファーマシューティカルズ・インコーポレイテッド ボロン酸エステル化合物およびその医薬組成物
WO2012119056A1 (en) * 2011-03-03 2012-09-07 Cephalon, Inc. Proteasome inhibitor delanzomib for use in the treatment of lupus

Non-Patent Citations (5)

* Cited by examiner, † Cited by third party
Title
ARTHRITIS RHEUM., vol. 64, no. 2, JPN6018016772, 2012, pages 493 - 503, ISSN: 0003930210 *
CHEM. BIOL., vol. 19, JPN6018016766, 2012, pages 99 - 115, ISSN: 0003930207 *
DRUGS FUTURE, vol. 37, no. 8, JPN6018016773, 2012, pages 561 - 565, ISSN: 0003930211 *
NAT. MED., vol. 14, no. 7, JPN6018016768, 2008, pages 748 - 755, ISSN: 0003930208 *
NEPHRON EXP. NEPHROL., vol. 120, JPN6018016771, 2012, pages 47 - 58, ISSN: 0003930209 *

Also Published As

Publication number Publication date
EP3052105A1 (en) 2016-08-10
US20160250238A1 (en) 2016-09-01
CA2925935A1 (en) 2015-04-09
WO2015051067A1 (en) 2015-04-09
US20180099000A1 (en) 2018-04-12
EA201690686A1 (ru) 2016-08-31
MX2016003979A (es) 2016-06-15
KR20160058886A (ko) 2016-05-25
CN105705149A (zh) 2016-06-22
BR112016007237A2 (pt) 2017-09-12

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