EA201690686A1 - Способ профилактики или лечения системной красной волчанки и/или волчаночного нефрита - Google Patents
Способ профилактики или лечения системной красной волчанки и/или волчаночного нефритаInfo
- Publication number
- EA201690686A1 EA201690686A1 EA201690686A EA201690686A EA201690686A1 EA 201690686 A1 EA201690686 A1 EA 201690686A1 EA 201690686 A EA201690686 A EA 201690686A EA 201690686 A EA201690686 A EA 201690686A EA 201690686 A1 EA201690686 A1 EA 201690686A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- lupine
- jade
- prevention
- treatment
- systemic red
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
В настоящем изобретении представлен способ профилактики или лечения системной красной волчанки и/или волчаночного нефрита у пациента, нуждающегося в этом, включающий введение пациенту эффективного количества [(1R)-1-({[(2,5-дихлорбензоил)амино]ацетил}амино)-3-метилбутил]бороновой кислоты или ее цитратного сложного эфира, или ее фармацевтически приемлемой соли.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361886403P | 2013-10-03 | 2013-10-03 | |
PCT/US2014/058738 WO2015051067A1 (en) | 2013-10-03 | 2014-10-02 | Method for the prophylaxis or treatment of systemic lupus erythematosus and/or lupus nephritis |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201690686A1 true EA201690686A1 (ru) | 2016-08-31 |
Family
ID=51842818
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201690686A EA201690686A1 (ru) | 2013-10-03 | 2014-10-02 | Способ профилактики или лечения системной красной волчанки и/или волчаночного нефрита |
Country Status (10)
Country | Link |
---|---|
US (2) | US20160250238A1 (ru) |
EP (1) | EP3052105A1 (ru) |
JP (1) | JP2016531886A (ru) |
KR (1) | KR20160058886A (ru) |
CN (1) | CN105705149A (ru) |
BR (1) | BR112016007237A2 (ru) |
CA (1) | CA2925935A1 (ru) |
EA (1) | EA201690686A1 (ru) |
MX (1) | MX2016003979A (ru) |
WO (1) | WO2015051067A1 (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP7304944B2 (ja) * | 2018-06-27 | 2023-07-07 | アルジャーノン・ファーマスーティカルズ・インコーポレイテッド | 腎線維症又は腎疾患の予防又は治療におけるアクタリットの使用 |
KR102344593B1 (ko) * | 2020-05-07 | 2021-12-29 | 주식회사 뉴로라이브 | 우울증 치료를 위한 사이클로세린 및 펜톡시필린 병용 요법 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6083903A (en) | 1994-10-28 | 2000-07-04 | Leukosite, Inc. | Boronic ester and acid compounds, synthesis and uses |
PT1355910E (pt) | 2001-01-25 | 2011-03-24 | Us Of America Represented By The Secretary Dept Of Health And Human Services | Formulação de compostos do ácido borónico |
KR20160040735A (ko) | 2007-08-06 | 2016-04-14 | 밀레니엄 파머슈티컬스 인코퍼레이티드 | 프로테아좀 억제제 |
US7442830B1 (en) | 2007-08-06 | 2008-10-28 | Millenium Pharmaceuticals, Inc. | Proteasome inhibitors |
EA027346B1 (ru) * | 2008-06-17 | 2017-07-31 | Милленниум Фармасьютикалз, Инк. | Соединения боронатного эфира и его фармацевтические составы |
AR075090A1 (es) | 2008-09-29 | 2011-03-09 | Millennium Pharm Inc | Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden. |
AR077033A1 (es) | 2009-06-11 | 2011-07-27 | Hoffmann La Roche | Compuestos inhibidores de las quinasas de janus y su uso en el tratamiento de enfermedades inmunologicas |
CN107266485A (zh) | 2010-03-31 | 2017-10-20 | 米伦纽姆医药公司 | 1‑氨基‑2‑环丙基乙硼酸衍生物 |
TW201309303A (zh) | 2011-03-03 | 2013-03-01 | Cephalon Inc | 用於治療狼瘡的蛋白酶體抑制劑 |
EP2723751A1 (en) * | 2011-06-22 | 2014-04-30 | Cephalon, Inc. | Proteasome inhibitors and processes for their preparation, purification and use |
-
2014
- 2014-10-02 US US15/026,417 patent/US20160250238A1/en not_active Abandoned
- 2014-10-02 CN CN201480060987.4A patent/CN105705149A/zh active Pending
- 2014-10-02 EP EP14790872.7A patent/EP3052105A1/en not_active Withdrawn
- 2014-10-02 KR KR1020167010114A patent/KR20160058886A/ko not_active Application Discontinuation
- 2014-10-02 EA EA201690686A patent/EA201690686A1/ru unknown
- 2014-10-02 BR BR112016007237A patent/BR112016007237A2/pt not_active IP Right Cessation
- 2014-10-02 JP JP2016519782A patent/JP2016531886A/ja active Pending
- 2014-10-02 MX MX2016003979A patent/MX2016003979A/es unknown
- 2014-10-02 WO PCT/US2014/058738 patent/WO2015051067A1/en active Application Filing
- 2014-10-02 CA CA2925935A patent/CA2925935A1/en not_active Abandoned
-
2017
- 2017-12-12 US US15/838,595 patent/US20180099000A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN105705149A (zh) | 2016-06-22 |
US20180099000A1 (en) | 2018-04-12 |
MX2016003979A (es) | 2016-06-15 |
BR112016007237A2 (pt) | 2017-09-12 |
KR20160058886A (ko) | 2016-05-25 |
JP2016531886A (ja) | 2016-10-13 |
EP3052105A1 (en) | 2016-08-10 |
WO2015051067A1 (en) | 2015-04-09 |
CA2925935A1 (en) | 2015-04-09 |
US20160250238A1 (en) | 2016-09-01 |
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