JP2015537008A5 - - Google Patents

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Publication number
JP2015537008A5
JP2015537008A5 JP2015542121A JP2015542121A JP2015537008A5 JP 2015537008 A5 JP2015537008 A5 JP 2015537008A5 JP 2015542121 A JP2015542121 A JP 2015542121A JP 2015542121 A JP2015542121 A JP 2015542121A JP 2015537008 A5 JP2015537008 A5 JP 2015537008A5
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JP
Japan
Prior art keywords
optionally substituted
membered monocyclic
alkyl
phenyl
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2015542121A
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English (en)
Japanese (ja)
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JP2015537008A (ja
JP6377068B2 (ja
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Priority claimed from PCT/CA2013/000957 external-priority patent/WO2014075168A1/en
Publication of JP2015537008A publication Critical patent/JP2015537008A/ja
Publication of JP2015537008A5 publication Critical patent/JP2015537008A5/ja
Application granted granted Critical
Publication of JP6377068B2 publication Critical patent/JP6377068B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2015542121A 2012-11-16 2013-11-15 ピラゾロピリミジン化合物 Active JP6377068B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261727581P 2012-11-16 2012-11-16
US61/727,581 2012-11-16
US201361808152P 2013-04-03 2013-04-03
US61/808,152 2013-04-03
PCT/CA2013/000957 WO2014075168A1 (en) 2012-11-16 2013-11-15 Pyrazolopyrimidine compounds

Publications (3)

Publication Number Publication Date
JP2015537008A JP2015537008A (ja) 2015-12-24
JP2015537008A5 true JP2015537008A5 (OSRAM) 2017-02-09
JP6377068B2 JP6377068B2 (ja) 2018-08-22

Family

ID=50730425

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015542121A Active JP6377068B2 (ja) 2012-11-16 2013-11-15 ピラゾロピリミジン化合物

Country Status (24)

Country Link
US (9) US9573954B2 (OSRAM)
EP (2) EP2920181B1 (OSRAM)
JP (1) JP6377068B2 (OSRAM)
CN (1) CN105793261B (OSRAM)
AU (1) AU2013344716B2 (OSRAM)
BR (1) BR112016010080B1 (OSRAM)
CA (1) CA2889919C (OSRAM)
CY (1) CY1120480T1 (OSRAM)
DK (1) DK3068786T3 (OSRAM)
ES (1) ES2686097T3 (OSRAM)
HR (1) HRP20181041T1 (OSRAM)
HU (1) HUE039351T2 (OSRAM)
IL (1) IL245187B (OSRAM)
LT (1) LT3068786T (OSRAM)
ME (1) ME03093B (OSRAM)
MX (1) MX373713B (OSRAM)
NZ (1) NZ707432A (OSRAM)
PL (1) PL3068786T3 (OSRAM)
PT (1) PT3068786T (OSRAM)
RS (1) RS57481B1 (OSRAM)
SG (1) SG11201603102TA (OSRAM)
SI (1) SI3068786T1 (OSRAM)
TW (1) TWI679201B (OSRAM)
WO (2) WO2014075168A1 (OSRAM)

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CN111377925B (zh) * 2018-12-28 2024-03-12 四川科伦博泰生物医药股份有限公司 嘌呤类衍生物、其制备方法及其在医药上的应用
CN112142744A (zh) 2019-06-28 2020-12-29 上海瑛派药业有限公司 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用
TW202146416A (zh) * 2019-12-11 2021-12-16 德商拜耳廠股份有限公司 吡唑并三𠯤
CN113773324B (zh) * 2021-09-07 2022-07-26 武汉九州钰民医药科技有限公司 抗肿瘤药cfi-402257的合成制备工艺
CN116396298A (zh) * 2023-06-06 2023-07-07 四川维亚本苑生物科技有限公司 CDK Ligand-1的中间体XII及CDK Ligand-1的制备方法

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