JP2015512447A5 - - Google Patents

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Publication number
JP2015512447A5
JP2015512447A5 JP2015504647A JP2015504647A JP2015512447A5 JP 2015512447 A5 JP2015512447 A5 JP 2015512447A5 JP 2015504647 A JP2015504647 A JP 2015504647A JP 2015504647 A JP2015504647 A JP 2015504647A JP 2015512447 A5 JP2015512447 A5 JP 2015512447A5
Authority
JP
Japan
Prior art keywords
tyrosine kinase
inhibitor
fgfr
pharmaceutically acceptable
met
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2015504647A
Other languages
English (en)
Japanese (ja)
Other versions
JP2015512447A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2013/034759 external-priority patent/WO2013151913A1/en
Publication of JP2015512447A publication Critical patent/JP2015512447A/ja
Publication of JP2015512447A5 publication Critical patent/JP2015512447A5/ja
Pending legal-status Critical Current

Links

JP2015504647A 2012-04-03 2013-04-01 チロシンキナーゼ阻害薬の組合せおよびその使用 Pending JP2015512447A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261619502P 2012-04-03 2012-04-03
US61/619,502 2012-04-03
PCT/US2013/034759 WO2013151913A1 (en) 2012-04-03 2013-04-01 Tyrosine kinase inhibitor combinations and their use

Publications (2)

Publication Number Publication Date
JP2015512447A JP2015512447A (ja) 2015-04-27
JP2015512447A5 true JP2015512447A5 (enExample) 2016-05-19

Family

ID=48184451

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015504647A Pending JP2015512447A (ja) 2012-04-03 2013-04-01 チロシンキナーゼ阻害薬の組合せおよびその使用

Country Status (11)

Country Link
US (1) US20150051210A1 (enExample)
EP (1) EP2833917A1 (enExample)
JP (1) JP2015512447A (enExample)
KR (1) KR20140146086A (enExample)
CN (1) CN104244982A (enExample)
AU (1) AU2013243737B2 (enExample)
CA (1) CA2866321A1 (enExample)
IN (1) IN2014DN07410A (enExample)
MX (1) MX2014011987A (enExample)
RU (1) RU2014143213A (enExample)
WO (1) WO2013151913A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102479693B1 (ko) 2014-03-26 2022-12-22 아스텍스 테라퓨틱스 리미티드 조합물
JP6526789B2 (ja) * 2014-07-31 2019-06-05 ノバルティス アーゲー 組み合わせ療法
JP6503450B2 (ja) 2015-03-25 2019-04-17 国立研究開発法人国立がん研究センター 胆管癌治療剤
CN108367000A (zh) 2015-12-17 2018-08-03 卫材R&D管理有限公司 用于乳腺癌的治疗剂

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0512324D0 (en) 2005-06-16 2005-07-27 Novartis Ag Organic compounds
DE102005038537A1 (de) 2005-08-16 2007-02-22 Merck Patent Gmbh 1-Acyldihydropyrazolderivate
JP5292102B2 (ja) 2005-12-21 2013-09-18 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ チロシンキナーゼ調節剤としてのトリアゾロピリダジン類
NL2000613C2 (nl) 2006-05-11 2007-11-20 Pfizer Prod Inc Triazoolpyrazinederivaten.
PE20121506A1 (es) 2006-07-14 2012-11-26 Amgen Inc Compuestos triazolopiridinas como inhibidores de c-met
EA200970403A1 (ru) 2006-10-23 2009-10-30 ЭсДжиЭкс ФАРМАСЬЮТИКАЛЗ, ИНК. Бициклические триазолы в качестве модуляторов протеинкиназы
SI2497470T1 (sl) 2006-11-22 2016-02-29 Incyte Holdings Corporation Imidazotriazini in imidazopirimidini kot inhibitorji kinaz
JP4994044B2 (ja) * 2007-01-05 2012-08-08 シェブロンジャパン株式会社 潤滑油組成物
EP2851091B1 (en) * 2007-04-13 2017-12-27 Dana-Farber Cancer Institute, Inc. Methods for treating cancer resistant to ERBB therapeutics
MX2010011959A (es) * 2008-04-29 2010-11-30 Novartis Ag Metodos para monitorear la modulacion de la actividad de cinasa del receptor del factor de crecimiento de fibroblastos y uso de dichos metodos.
CA2723617A1 (en) * 2008-05-14 2009-11-19 Amgen Inc. Combinations vegf(r) inhibitors and hepatocyte growth factor (c-met) inhibitors for the treatment of cancer
KR20120089643A (ko) 2009-08-12 2012-08-13 노파르티스 아게 헤테로시클릭 히드라존 화합물, 및 암 및 염증을 치료하기 위한 그의 용도
JP2013537918A (ja) * 2010-09-27 2013-10-07 エクセリクシス, インク. 去勢抵抗性前立腺癌および骨芽細胞骨転移の治療のためのmetおよびvegfの二元阻害薬

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