JP2015512447A5 - - Google Patents
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- Publication number
- JP2015512447A5 JP2015512447A5 JP2015504647A JP2015504647A JP2015512447A5 JP 2015512447 A5 JP2015512447 A5 JP 2015512447A5 JP 2015504647 A JP2015504647 A JP 2015504647A JP 2015504647 A JP2015504647 A JP 2015504647A JP 2015512447 A5 JP2015512447 A5 JP 2015512447A5
- Authority
- JP
- Japan
- Prior art keywords
- tyrosine kinase
- inhibitor
- fgfr
- pharmaceutically acceptable
- met
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261619502P | 2012-04-03 | 2012-04-03 | |
| US61/619,502 | 2012-04-03 | ||
| PCT/US2013/034759 WO2013151913A1 (en) | 2012-04-03 | 2013-04-01 | Tyrosine kinase inhibitor combinations and their use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2015512447A JP2015512447A (ja) | 2015-04-27 |
| JP2015512447A5 true JP2015512447A5 (enExample) | 2016-05-19 |
Family
ID=48184451
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015504647A Pending JP2015512447A (ja) | 2012-04-03 | 2013-04-01 | チロシンキナーゼ阻害薬の組合せおよびその使用 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20150051210A1 (enExample) |
| EP (1) | EP2833917A1 (enExample) |
| JP (1) | JP2015512447A (enExample) |
| KR (1) | KR20140146086A (enExample) |
| CN (1) | CN104244982A (enExample) |
| AU (1) | AU2013243737B2 (enExample) |
| CA (1) | CA2866321A1 (enExample) |
| IN (1) | IN2014DN07410A (enExample) |
| MX (1) | MX2014011987A (enExample) |
| RU (1) | RU2014143213A (enExample) |
| WO (1) | WO2013151913A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102479693B1 (ko) | 2014-03-26 | 2022-12-22 | 아스텍스 테라퓨틱스 리미티드 | 조합물 |
| JP6526789B2 (ja) * | 2014-07-31 | 2019-06-05 | ノバルティス アーゲー | 組み合わせ療法 |
| JP6503450B2 (ja) | 2015-03-25 | 2019-04-17 | 国立研究開発法人国立がん研究センター | 胆管癌治療剤 |
| CN108367000A (zh) | 2015-12-17 | 2018-08-03 | 卫材R&D管理有限公司 | 用于乳腺癌的治疗剂 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0512324D0 (en) | 2005-06-16 | 2005-07-27 | Novartis Ag | Organic compounds |
| DE102005038537A1 (de) | 2005-08-16 | 2007-02-22 | Merck Patent Gmbh | 1-Acyldihydropyrazolderivate |
| JP5292102B2 (ja) | 2005-12-21 | 2013-09-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | チロシンキナーゼ調節剤としてのトリアゾロピリダジン類 |
| NL2000613C2 (nl) | 2006-05-11 | 2007-11-20 | Pfizer Prod Inc | Triazoolpyrazinederivaten. |
| PE20121506A1 (es) | 2006-07-14 | 2012-11-26 | Amgen Inc | Compuestos triazolopiridinas como inhibidores de c-met |
| EA200970403A1 (ru) | 2006-10-23 | 2009-10-30 | ЭсДжиЭкс ФАРМАСЬЮТИКАЛЗ, ИНК. | Бициклические триазолы в качестве модуляторов протеинкиназы |
| SI2497470T1 (sl) | 2006-11-22 | 2016-02-29 | Incyte Holdings Corporation | Imidazotriazini in imidazopirimidini kot inhibitorji kinaz |
| JP4994044B2 (ja) * | 2007-01-05 | 2012-08-08 | シェブロンジャパン株式会社 | 潤滑油組成物 |
| EP2851091B1 (en) * | 2007-04-13 | 2017-12-27 | Dana-Farber Cancer Institute, Inc. | Methods for treating cancer resistant to ERBB therapeutics |
| MX2010011959A (es) * | 2008-04-29 | 2010-11-30 | Novartis Ag | Metodos para monitorear la modulacion de la actividad de cinasa del receptor del factor de crecimiento de fibroblastos y uso de dichos metodos. |
| CA2723617A1 (en) * | 2008-05-14 | 2009-11-19 | Amgen Inc. | Combinations vegf(r) inhibitors and hepatocyte growth factor (c-met) inhibitors for the treatment of cancer |
| KR20120089643A (ko) | 2009-08-12 | 2012-08-13 | 노파르티스 아게 | 헤테로시클릭 히드라존 화합물, 및 암 및 염증을 치료하기 위한 그의 용도 |
| JP2013537918A (ja) * | 2010-09-27 | 2013-10-07 | エクセリクシス, インク. | 去勢抵抗性前立腺癌および骨芽細胞骨転移の治療のためのmetおよびvegfの二元阻害薬 |
-
2013
- 2013-04-01 IN IN7410DEN2014 patent/IN2014DN07410A/en unknown
- 2013-04-01 CA CA2866321A patent/CA2866321A1/en not_active Abandoned
- 2013-04-01 WO PCT/US2013/034759 patent/WO2013151913A1/en not_active Ceased
- 2013-04-01 CN CN201380018928.6A patent/CN104244982A/zh active Pending
- 2013-04-01 MX MX2014011987A patent/MX2014011987A/es unknown
- 2013-04-01 US US14/388,251 patent/US20150051210A1/en not_active Abandoned
- 2013-04-01 EP EP13718671.4A patent/EP2833917A1/en not_active Withdrawn
- 2013-04-01 JP JP2015504647A patent/JP2015512447A/ja active Pending
- 2013-04-01 KR KR1020147027542A patent/KR20140146086A/ko not_active Withdrawn
- 2013-04-01 AU AU2013243737A patent/AU2013243737B2/en not_active Ceased
- 2013-04-01 RU RU2014143213A patent/RU2014143213A/ru not_active Application Discontinuation
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