JP2015504432A5 - - Google Patents

Download PDF

Info

Publication number
JP2015504432A5
JP2015504432A5 JP2014542646A JP2014542646A JP2015504432A5 JP 2015504432 A5 JP2015504432 A5 JP 2015504432A5 JP 2014542646 A JP2014542646 A JP 2014542646A JP 2014542646 A JP2014542646 A JP 2014542646A JP 2015504432 A5 JP2015504432 A5 JP 2015504432A5
Authority
JP
Japan
Prior art keywords
relates
trimethoxyphenyl
hydrazide
hydrazones
present
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2014542646A
Other languages
English (en)
Japanese (ja)
Other versions
JP2015504432A (ja
Filing date
Publication date
Priority claimed from BRPI1107312-8A external-priority patent/BRPI1107312B1/pt
Application filed filed Critical
Publication of JP2015504432A publication Critical patent/JP2015504432A/ja
Publication of JP2015504432A5 publication Critical patent/JP2015504432A5/ja
Pending legal-status Critical Current

Links

JP2014542646A 2011-11-25 2012-11-26 アシル−ヒドラゾンおよびオキサジアゾール化合物、これらを含有する医薬組成物およびその使用 Pending JP2015504432A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
BRPI1107312-8A BRPI1107312B1 (pt) 2011-11-25 2011-11-25 Composto de acil-hidrazona
BRPI1107312-8 2011-11-25
PCT/BR2012/000480 WO2013075199A1 (pt) 2011-11-25 2012-11-26 "compostos acil-hidrazonas e oxadiazóis, composições farmacêuticas compreendendo os mesmos e seus usos

Publications (2)

Publication Number Publication Date
JP2015504432A JP2015504432A (ja) 2015-02-12
JP2015504432A5 true JP2015504432A5 (enExample) 2016-01-21

Family

ID=48468927

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014542646A Pending JP2015504432A (ja) 2011-11-25 2012-11-26 アシル−ヒドラゾンおよびオキサジアゾール化合物、これらを含有する医薬組成物およびその使用

Country Status (9)

Country Link
US (1) US20150191445A1 (enExample)
EP (1) EP2784061B1 (enExample)
JP (1) JP2015504432A (enExample)
KR (1) KR102189562B1 (enExample)
CN (1) CN104159887A (enExample)
BR (2) BRPI1107312B1 (enExample)
CA (1) CA2869807C (enExample)
RU (1) RU2664327C2 (enExample)
WO (1) WO2013075199A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101719541B1 (ko) 2015-08-13 2017-03-24 연세대학교 산학협력단 항암용 약학 조성물 및 ano1 활성억제제
KR20170141542A (ko) * 2016-06-15 2017-12-26 국립암센터 위암을 예방 및 치료하는 rhoa 억제제의 약학적 조성물
CN110498809B (zh) * 2018-05-17 2022-04-05 香港科技大学深圳研究院 基于酰腙配体类的有机硼化合物及其制备方法和应用
KR102131331B1 (ko) 2018-09-19 2020-07-07 연세대학교 산학협력단 항암용 신규 약학 조성물 및 ano1 활성억제제
CN113336729B (zh) * 2021-05-31 2022-05-27 四川大学华西医院 硝呋齐特类衍生物及其制备方法和用途

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60105621A (ja) * 1983-11-14 1985-06-11 Agency Of Ind Science & Technol 細胞の分化誘導作用を有する生理活性物質およびその製法
IL94389A0 (en) * 1989-06-01 1991-03-10 Health Research Inc Monoclonal antibody reactive to a unique antigen widely present on various human leukemia and lymphoma cells and method of using same for diagnosis and treatment
US5372808A (en) * 1990-10-17 1994-12-13 Amgen Inc. Methods and compositions for the treatment of diseases with consensus interferon while reducing side effect
US6197806B1 (en) * 1995-12-20 2001-03-06 Nippon Zoki Pharmaceutical Co., Ltd. Eliminating agent for activated oxygen and free radicals
CA2400996A1 (en) 2002-09-03 2004-03-03 Lisa Mckerracher 1,4-substituted cyclohexane derivatives
KR101155883B1 (ko) 2003-12-23 2012-06-20 아제닉스 유에스에이 인코포레이티드 사이클린 의존적 키나제 저해제, 그 조성물 및 그의 용도
DE102004010207A1 (de) 2004-03-02 2005-09-15 Aventis Pharma S.A. Neue 4-Benzimidazol-2-yl-pyridazin-3-on-Derivate
WO2005097763A2 (en) * 2004-04-01 2005-10-20 Aventis Pharmaceuticals Inc. 1,3,4-oxadiazol-2-ones as ppar delta
AR052559A1 (es) 2005-01-21 2007-03-21 Astex Therapeutics Ltd Derivados de pirazol para inhibir cdk's y gsk's
WO2006101937A1 (en) 2005-03-18 2006-09-28 Janssen Pharmaceutica N.V. Acylhydrazones as kinase modulators
CN1824657A (zh) * 2006-04-05 2006-08-30 贵州大学 3-取代-2-芳基取代-5-(3,4,5-三烷氧基苯基)-1,3,4-噁二唑衍生物及制备方法和用途
US20110189306A1 (en) * 2010-01-13 2011-08-04 Norbert Kartner COMPOUNDS, COMPOSITIONS AND TREATMENTS FOR V-ATPase RELATED DISEASES

Similar Documents

Publication Publication Date Title
LT4303583T (lt) Csf1r inhibitoriai, skirti panaudoti gydant tenosinovinius gigantinių ląstelių navikus
HK1217215A1 (zh) 用於改变细胞表型的信号传感器多核苷酸
CN110198943A (zh) 作为Wee1抑制剂的1,2-二氢-3H-吡唑[3,4-d]嘧啶-3-酮衍生物
WO2014191359A9 (en) Aptamers and use of the aptamers in the diagnosis and treatment of cancer
DE112012006327A5 (de) Kombinationsbehandlung (z.B. mit ABT-072 oder ABT-333 von DAAs zur Verwendung in der Behandlung von HCV)
CA2900335C (en) Synthetic analogs of epipolythiodioxopiperazines and uses thereof
JP2014530840A5 (enExample)
WO2015067715A3 (en) Gip-glp-1 dual agonist compounds and methods
DK3124043T3 (da) Hidtil ukendt immunterapi mod flere forskellige tumorer, herunder nerve- og hjernetumorer
MX2014011134A (es) Compuestos de carbamato y preparacion y uso de los mismos.
CO6791606A2 (es) Composiciones y métodos para el tratamiento en aplicaciones clínicas de amplio espectro, no diferenciadas o combinadas
DK3195873T3 (da) Hidtil ukendt immunterapi mod flere forskellige tumortyper, herunder mave-tarm-cancer og mavecancer
CN109843873A (zh) 炔代杂环化合物、其制备方法及其在医药学上的应用
CL2014000849A1 (es) Compuestos derivados de benzilindazoles sustituido, inhibidores de la quinasa bub1; procedimiento de fabricacion; composicion farmaceutica; combinacion farmaceutica; y su uso en el tratamiento de enfermedades hiperproliferativas.
HK1217650A1 (zh) 用於治疗剧痛的组合物及方法
BRPI0909818A2 (pt) métodos, formas de dosagem e conjunto para administrar ziprasidona sem alimentos
JP2015502958A5 (enExample)
JP2015504432A5 (enExample)
JP2014519480A5 (enExample)
WO2011159693A3 (en) Oral treatment of digital ischemic lesions
CL2011002965A1 (es) Compuestos derivados de piperidinas sustituidas; procedimiento de preparacion; composicion farmaceutica; y uso de dichos compuestos para el tratamiento y/o profilaxis de trastornos cardiovasculares, tromboembolicos y/o tumores.
JP2013231052A5 (enExample)
JP2016503275A5 (enExample)
JP2014510253A5 (enExample)
JP2013100268A5 (enExample)