JP2015042663A5 - - Google Patents

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Publication number
JP2015042663A5
JP2015042663A5 JP2014219074A JP2014219074A JP2015042663A5 JP 2015042663 A5 JP2015042663 A5 JP 2015042663A5 JP 2014219074 A JP2014219074 A JP 2014219074A JP 2014219074 A JP2014219074 A JP 2014219074A JP 2015042663 A5 JP2015042663 A5 JP 2015042663A5
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JP
Japan
Prior art keywords
group
hydrogen atom
substituent
optionally
formula
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Application number
JP2014219074A
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English (en)
Japanese (ja)
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JP2015042663A (ja
JP5891576B2 (ja
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Priority to JP2014219074A priority Critical patent/JP5891576B2/ja
Priority claimed from JP2014219074A external-priority patent/JP5891576B2/ja
Publication of JP2015042663A publication Critical patent/JP2015042663A/ja
Publication of JP2015042663A5 publication Critical patent/JP2015042663A5/ja
Application granted granted Critical
Publication of JP5891576B2 publication Critical patent/JP5891576B2/ja
Active legal-status Critical Current
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JP2014219074A 2011-03-31 2014-10-28 新規フラノン誘導体 Active JP5891576B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2014219074A JP5891576B2 (ja) 2011-03-31 2014-10-28 新規フラノン誘導体

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2011080185 2011-03-31
JP2011080185 2011-03-31
JP2014219074A JP5891576B2 (ja) 2011-03-31 2014-10-28 新規フラノン誘導体

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2013507805A Division JP5659356B2 (ja) 2011-03-31 2012-03-30 新規フラノン誘導体

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016020407A Division JP6256927B2 (ja) 2011-03-31 2016-02-05 新規フラノン誘導体

Publications (3)

Publication Number Publication Date
JP2015042663A JP2015042663A (ja) 2015-03-05
JP2015042663A5 true JP2015042663A5 (enExample) 2015-04-30
JP5891576B2 JP5891576B2 (ja) 2016-03-23

Family

ID=46931496

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2013507805A Active JP5659356B2 (ja) 2011-03-31 2012-03-30 新規フラノン誘導体
JP2014219074A Active JP5891576B2 (ja) 2011-03-31 2014-10-28 新規フラノン誘導体
JP2016020407A Active JP6256927B2 (ja) 2011-03-31 2016-02-05 新規フラノン誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2013507805A Active JP5659356B2 (ja) 2011-03-31 2012-03-30 新規フラノン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2016020407A Active JP6256927B2 (ja) 2011-03-31 2016-02-05 新規フラノン誘導体

Country Status (12)

Country Link
US (3) US8742113B2 (enExample)
EP (1) EP2692728B1 (enExample)
JP (3) JP5659356B2 (enExample)
KR (1) KR101964479B1 (enExample)
CN (1) CN103459388B (enExample)
AU (3) AU2012233246B2 (enExample)
BR (1) BR112013024957A2 (enExample)
CA (1) CA2830148C (enExample)
DK (1) DK2692728T3 (enExample)
ES (1) ES2687450T3 (enExample)
MX (1) MX344474B (enExample)
WO (1) WO2012133802A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8742113B2 (en) 2011-03-31 2014-06-03 Sbi Biotech Co., Ltd. Furanone derivative
JP6569908B2 (ja) * 2014-01-31 2019-09-04 カルナバイオサイエンス株式会社 抗がん剤組成物
CN104744353B (zh) * 2015-03-31 2017-11-24 山东友帮生化科技有限公司 2‑氨基‑3‑碘‑5‑氯吡啶的合成方法
AU2017354372A1 (en) * 2016-11-04 2019-06-20 Carna Biosciences, Inc. Furanone derivates and methods of use thereof
GB201807147D0 (en) 2018-05-01 2018-06-13 Oncologica Uk Ltd Therapeutic combination
US12533353B2 (en) * 2018-09-24 2026-01-27 Carna Biosciences, Inc. Methods of treatment of cancer comprising CDC7 inhibitors

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6987113B2 (en) 1997-06-11 2006-01-17 Sugen, Inc. Tyrosine kinase inhibitors
US6335342B1 (en) 2000-06-19 2002-01-01 Pharmacia & Upjohn S.P.A. Azaindole derivatives, process for their preparation, and their use as antitumor agents
JP2006501191A (ja) 2002-07-17 2006-01-12 ファルマシア・イタリア・エス・ピー・エー キナーゼ阻害剤としてのヘテロ二環式ピラゾール誘導体
US20050137220A1 (en) 2003-07-23 2005-06-23 Pharmacia Corporation Beta-carboline compounds and analogues thereof as mitogen-activated protein kinase-activated protein kinase-2 inhibitors
DE602004014163D1 (de) 2003-08-08 2008-07-10 Pfizer Italia Srl Pyrimidylpyrrolderivate, die als kinaseinhibitoren wirken
US20050043346A1 (en) 2003-08-08 2005-02-24 Pharmacia Italia S.P.A. Pyridylpyrrole derivatives active as kinase inhibitors
FR2876103B1 (fr) 2004-10-01 2008-02-22 Aventis Pharma Sa Nouveaux derives bis-azaindoles, leur preparation et leur utilisation pharmaceutique comme inhibiteurs de kinases
AU2005293831B2 (en) * 2004-10-14 2011-01-06 F. Hoffmann-La Roche Ag Novel Azaindole thiazolinones as anti-cancer agents
US20060122232A1 (en) * 2004-12-06 2006-06-08 Development Center For Biotechnology 4-Hydroxyfuroic acid derivatives
US7371862B2 (en) * 2005-11-11 2008-05-13 Pfizer Italia S.R.L. Azaindolylidene derivatives as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
KR20090008286A (ko) 2006-03-27 2009-01-21 네르비아노 메디칼 사이언시스 에스.알.엘. 키나제 억제제로서의 피리딜- 및 피리미디닐-치환된 피롤-,티오펜- 및 푸란- 유도체
FR2907120B1 (fr) 2006-10-12 2013-01-11 Sanofi Aventis Nouveaux derives imidazolones,leur preparation a titre de medicaments,compositions pharmaceutiques,utilisation comme inhibiteurs de proteines kinases notamment cdc7
WO2008109443A2 (en) 2007-03-02 2008-09-12 Mdrna, Inc. Nucleic acid compounds for inhibiting cdk2 gene expression and uses thereof
WO2009155052A1 (en) 2008-05-28 2009-12-23 Wyeth 3-substituted-1h-pyrrolo[2,3-b]pyridine and 3-substituted-1h-pyrrolo[3,2-b]pyridine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses
WO2010030727A1 (en) * 2008-09-10 2010-03-18 Wyeth Llc 3-substituted-1h-indole, 3-substituted-1h-pyrrolo[2,3-b]pyridine and 3-substituted-1h-pyrrolo[3,2-b]pyridine compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses
CA2767089A1 (en) 2009-07-15 2011-01-20 Abbott Laboratories Pyrrolopyridine inhibitors of kinases
TW201127384A (en) 2009-11-18 2011-08-16 Nerviano Medical Sciences Srl Therapeutic combination comprising a Cdc7 inhibitor and an antineoplastic agent
US20120135989A1 (en) 2010-06-29 2012-05-31 Crystalgenomics, Inc. Azaindole derivative
US8742113B2 (en) 2011-03-31 2014-06-03 Sbi Biotech Co., Ltd. Furanone derivative
JP6569908B2 (ja) 2014-01-31 2019-09-04 カルナバイオサイエンス株式会社 抗がん剤組成物

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