JP2014532621A5 - - Google Patents

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Publication number
JP2014532621A5
JP2014532621A5 JP2014537107A JP2014537107A JP2014532621A5 JP 2014532621 A5 JP2014532621 A5 JP 2014532621A5 JP 2014537107 A JP2014537107 A JP 2014537107A JP 2014537107 A JP2014537107 A JP 2014537107A JP 2014532621 A5 JP2014532621 A5 JP 2014532621A5
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JP
Japan
Prior art keywords
group
hydroxy
hydrogen
alkyl
compound
Prior art date
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Application number
JP2014537107A
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English (en)
Japanese (ja)
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JP2014532621A (ja
JP6072811B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2012/059315 external-priority patent/WO2013059021A1/en
Publication of JP2014532621A publication Critical patent/JP2014532621A/ja
Publication of JP2014532621A5 publication Critical patent/JP2014532621A5/ja
Application granted granted Critical
Publication of JP6072811B2 publication Critical patent/JP6072811B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2014537107A 2011-10-21 2012-10-09 ２−メチレン−ビタミンｄ類似体およびそれらの使用 Expired - Fee Related JP6072811B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161550147P 2011-10-21 2011-10-21
US61/550,147 2011-10-21
PCT/US2012/059315 WO2013059021A1 (en) 2011-10-21 2012-10-09 2-methylene-vitamin d analogs and their uses

Publications (3)

Publication Number Publication Date
JP2014532621A JP2014532621A (ja) 2014-12-08
JP2014532621A5 true JP2014532621A5 (enExample) 2015-11-26
JP6072811B2 JP6072811B2 (ja) 2017-02-01

Family

ID=47080842

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014537107A Expired - Fee Related JP6072811B2 (ja) 2011-10-21 2012-10-09 ２−メチレン−ビタミンｄ類似体およびそれらの使用

Country Status (6)

Country Link
US (1) US8455467B2 (enExample)
EP (1) EP2768803B1 (enExample)
JP (1) JP6072811B2 (enExample)
AU (1) AU2012326538B2 (enExample)
CA (1) CA2851275C (enExample)
WO (1) WO2013059021A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010300539B9 (en) * 2009-10-02 2018-07-19 Wisconsin Alumni Research Foundation 1-desoxy-2-methylene-19-nor-vitamin D analogs and their uses
US9688596B2 (en) * 2015-08-05 2017-06-27 Wisconsin Alumni Research Foundation Synthesis and biological activity of 2-methylene analogs of calcitriol and related compounds

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4666634A (en) * 1984-12-05 1987-05-19 Chugai Seiyaku Kabushiki Kaisha vitamin D3 derivatives having a substituent at 2-position
US5086191A (en) 1991-05-28 1992-02-04 Wisconsin Alumni Research Foundation Intermediates for the synthesis of 19-nor vitamin D compounds
JP2898882B2 (ja) 1993-04-05 1999-06-02 ウイスコンシン アラムナイ リサーチ フオンデーシヨン ２−位に置換基を有する１９−ノル−ビタミンｄ３ 化合物
US5843928A (en) 1997-03-17 1998-12-01 Wisconsin Alumni Research Foundation 2-alkylidene-19-nor-vitamin D compounds
US5945410A (en) 1997-03-17 1999-08-31 Wisconsin Alumni Research Foundation 2-alkyl-19-nor-vitamin D compounds
US6392071B1 (en) 1997-03-17 2002-05-21 Wisconsin Alumni: Research Foundation 26,27-homologated-20-EPI-2-alkylidene-19-nor-vitamin D compounds
US6382071B1 (en) 2000-08-07 2002-05-07 Gilbert A. Bertani Bola capturing apparatus
AU7544501A (en) 2000-09-08 2002-03-22 Wisconsin Alumni Res Found 1alpha-hydroxy-2-methylene-19-nor-homopregnacalciferol and its therapeutic applications
WO2003051828A2 (en) * 2001-12-13 2003-06-26 Wisconsin Alumni Research Foundation (20s)-1alpha-hydroxy-2-methylene-19-nor-bishomopregnacalciferol and its uses
US6627622B2 (en) 2002-02-18 2003-09-30 Wisconsin Alumni Research Foundation (20S)-1α-hydroxy-2-methylene-19-nor-bishomopregnacalciferol and its uses
US6566352B1 (en) * 2002-02-18 2003-05-20 Wisconsin Alumni Research Foudation 1 α-hydroxy-2-methylene-19-nor-pregnacalciferol and its uses
US20080249068A1 (en) * 2002-09-05 2008-10-09 Deluca Hector F Method of Extending the Dose Range of Vitamin D Compounds
AU2010300539B9 (en) * 2009-10-02 2018-07-19 Wisconsin Alumni Research Foundation 1-desoxy-2-methylene-19-nor-vitamin D analogs and their uses

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