JP2013544277A - Ｋａｔｉｉ阻害剤 - Google Patents
Ｋａｔｉｉ阻害剤 Download PDFInfo
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- JP2013544277A JP2013544277A JP2013541446A JP2013541446A JP2013544277A JP 2013544277 A JP2013544277 A JP 2013544277A JP 2013541446 A JP2013541446 A JP 2013541446A JP 2013541446 A JP2013541446 A JP 2013541446A JP 2013544277 A JP2013544277 A JP 2013544277A
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- Prior art keywords
- alkyl
- aryl
- cycloalkyl
- heteroaryl
- mmol
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- YEHNWRNMGIYLAL-NSHDSACASA-N (5s)-5-amino-2-benzyl-7-hydroxy-4,5-dihydropyrazolo[3,4-b]pyridin-6-one Chemical compound C([C@@H](C(N(O)C1=N2)=O)N)C1=CN2CC1=CC=CC=C1 YEHNWRNMGIYLAL-NSHDSACASA-N 0.000 claims description 2
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Landscapes
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| US41880210P | 2010-12-01 | 2010-12-01 | |
| US61/418,802 | 2010-12-01 | ||
| PCT/IB2011/055158 WO2012073143A1 (en) | 2010-12-01 | 2011-11-17 | Kat ii inhibitors |
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| JP2013544277A true JP2013544277A (ja) | 2013-12-12 |
| JP2013544277A5 JP2013544277A5 (enExample) | 2014-09-25 |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015163339A1 (ja) * | 2014-04-23 | 2015-10-29 | 田辺三菱製薬株式会社 | 新規二環性または三環性複素環化合物 |
| WO2017069275A1 (ja) * | 2015-10-22 | 2017-04-27 | 田辺三菱製薬株式会社 | 新規二環性複素環化合物 |
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| WO2012073146A1 (en) | 2010-12-01 | 2012-06-07 | Pfizer Inc. | Kat ii inhibitors |
| US10154988B2 (en) | 2012-11-14 | 2018-12-18 | The Johns Hopkins University | Methods and compositions for treating schizophrenia |
| WO2016164703A1 (en) | 2015-04-09 | 2016-10-13 | Eisai R & D Management Co., Ltd. | Fgfr4 inhibitors |
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| JPWO2017069275A1 (ja) * | 2015-10-22 | 2018-08-09 | 田辺三菱製薬株式会社 | 新規二環性複素環化合物 |
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| US20140057938A1 (en) | 2014-02-27 |
| KR20130108618A (ko) | 2013-10-04 |
| WO2012073143A1 (en) | 2012-06-07 |
| CA2819102A1 (en) | 2012-06-07 |
| US8933095B2 (en) | 2015-01-13 |
| MX2013005773A (es) | 2013-06-18 |
| DK2646443T3 (en) | 2014-11-17 |
| EP2646443A1 (en) | 2013-10-09 |
| CN103228660A (zh) | 2013-07-31 |
| AU2011336214B2 (en) | 2015-08-20 |
| ES2524423T3 (es) | 2014-12-09 |
| ZA201303360B (en) | 2014-07-30 |
| US20120302599A1 (en) | 2012-11-29 |
| US8598200B2 (en) | 2013-12-03 |
| SG190207A1 (en) | 2013-06-28 |
| KR101544290B1 (ko) | 2015-08-12 |
| AU2011336214A1 (en) | 2013-05-30 |
| EP2646443B1 (en) | 2014-09-24 |
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