JP2013543881A - 秩序化したメソポーラスシリカの圧縮製剤 - Google Patents
秩序化したメソポーラスシリカの圧縮製剤 Download PDFInfo
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- JP2013543881A JP2013543881A JP2013540410A JP2013540410A JP2013543881A JP 2013543881 A JP2013543881 A JP 2013543881A JP 2013540410 A JP2013540410 A JP 2013540410A JP 2013540410 A JP2013540410 A JP 2013540410A JP 2013543881 A JP2013543881 A JP 2013543881A
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- Prior art keywords
- formulation
- mesoporous silica
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- drug
- croscarmellose sodium
- Prior art date
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
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- A61K9/143—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
Landscapes
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- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10192938 | 2010-11-29 | ||
| EP10192938.8 | 2010-11-29 | ||
| PCT/EP2011/071186 WO2012072580A1 (en) | 2010-11-29 | 2011-11-28 | Compressed formulations of ordered mesoporous silicas |
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| JP2013543881A true JP2013543881A (ja) | 2013-12-09 |
| JP2013543881A5 JP2013543881A5 (enExample) | 2014-03-06 |
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| JP2013540410A Pending JP2013543881A (ja) | 2010-11-29 | 2011-11-28 | 秩序化したメソポーラスシリカの圧縮製剤 |
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| Country | Link |
|---|---|
| US (1) | US20130243833A1 (enExample) |
| EP (1) | EP2646005B1 (enExample) |
| JP (1) | JP2013543881A (enExample) |
| ES (1) | ES2744926T3 (enExample) |
| PL (1) | PL2646005T3 (enExample) |
| WO (1) | WO2012072580A1 (enExample) |
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|---|---|---|---|---|
| GB201212866D0 (en) * | 2012-07-20 | 2012-09-05 | Formac Pharmaceuticals Nv | Dry granulates of mesoporous silica powders |
| US20170246111A1 (en) | 2014-09-15 | 2017-08-31 | Pharmasol Gmbh | Active-loaded particulate materials for topical administration |
| KR20210089210A (ko) | 2018-11-07 | 2021-07-15 | 디스럽티브 매터리얼즈 파마 아베 | 실질적 비정질인 메조포러스 탄산마그네슘을 포함하는 신규한 비정질 활성 제약 성분 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003531083A (ja) * | 1997-12-09 | 2003-10-21 | ザ・リージェンツ・オブ・ザ・ユニバーシティー・オブ・カリフォルニア | メソ構造の無機酸化物材料のブロックポリマー処理方法 |
| JP2006528194A (ja) * | 2003-07-22 | 2006-12-14 | アイオワ ステート ユニバーシティー リサーチ ファウンデーション，インク． | キャップドメソポーラス珪酸塩 |
| WO2009133100A2 (en) * | 2008-04-28 | 2009-11-05 | Formac Pharmaceuticals N.V. | Ordered mesoporous silica material |
| WO2010091197A2 (en) * | 2009-02-06 | 2010-08-12 | Gilead Sciences, Inc. | Tablets for combination therapy |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060018966A1 (en) | 2003-07-22 | 2006-01-26 | Lin Victor S | Antimicrobial mesoporous silica nanoparticles |
-
2011
- 2011-11-28 EP EP11822806.3A patent/EP2646005B1/en active Active
- 2011-11-28 PL PL11822806T patent/PL2646005T3/pl unknown
- 2011-11-28 JP JP2013540410A patent/JP2013543881A/ja active Pending
- 2011-11-28 WO PCT/EP2011/071186 patent/WO2012072580A1/en not_active Ceased
- 2011-11-28 US US13/988,687 patent/US20130243833A1/en not_active Abandoned
- 2011-11-28 ES ES11822806T patent/ES2744926T3/es active Active
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003531083A (ja) * | 1997-12-09 | 2003-10-21 | ザ・リージェンツ・オブ・ザ・ユニバーシティー・オブ・カリフォルニア | メソ構造の無機酸化物材料のブロックポリマー処理方法 |
| JP2006528194A (ja) * | 2003-07-22 | 2006-12-14 | アイオワ ステート ユニバーシティー リサーチ ファウンデーション，インク． | キャップドメソポーラス珪酸塩 |
| WO2009133100A2 (en) * | 2008-04-28 | 2009-11-05 | Formac Pharmaceuticals N.V. | Ordered mesoporous silica material |
| WO2010091197A2 (en) * | 2009-02-06 | 2010-08-12 | Gilead Sciences, Inc. | Tablets for combination therapy |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2646005A1 (en) | 2013-10-09 |
| PL2646005T3 (pl) | 2019-12-31 |
| WO2012072580A1 (en) | 2012-06-07 |
| US20130243833A1 (en) | 2013-09-19 |
| EP2646005B1 (en) | 2019-06-26 |
| ES2744926T3 (es) | 2020-02-26 |
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