JP2013528649A - 肺高血圧症の処置のために使用するためのラノラジン - Google Patents
肺高血圧症の処置のために使用するためのラノラジン Download PDFInfo
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- JP2013528649A JP2013528649A JP2013515456A JP2013515456A JP2013528649A JP 2013528649 A JP2013528649 A JP 2013528649A JP 2013515456 A JP2013515456 A JP 2013515456A JP 2013515456 A JP2013515456 A JP 2013515456A JP 2013528649 A JP2013528649 A JP 2013528649A
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- ranolazine
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- pulmonary hypertension
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35546210P | 2010-06-16 | 2010-06-16 | |
| US61/355,462 | 2010-06-16 | ||
| US40786410P | 2010-10-28 | 2010-10-28 | |
| US61/407,864 | 2010-10-28 | ||
| PCT/US2011/040363 WO2011159706A1 (en) | 2010-06-16 | 2011-06-14 | Ranolazine for use for the treatment of pulmonary hypertension |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013528649A true JP2013528649A (ja) | 2013-07-11 |
| JP2013528649A5 JP2013528649A5 (enExample) | 2014-07-31 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2013515456A Withdrawn JP2013528649A (ja) | 2010-06-16 | 2011-06-14 | 肺高血圧症の処置のために使用するためのラノラジン |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20120004188A1 (enExample) |
| EP (1) | EP2582372A1 (enExample) |
| JP (1) | JP2013528649A (enExample) |
| AR (1) | AR081925A1 (enExample) |
| AU (1) | AU2011267871A1 (enExample) |
| CA (1) | CA2801707A1 (enExample) |
| TW (1) | TW201215392A (enExample) |
| UY (1) | UY33453A (enExample) |
| WO (1) | WO2011159706A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023542298A (ja) * | 2020-09-11 | 2023-10-06 | プルモシム セラピューティクス リミテッド ライアビリティ カンパニー | 肺高血圧症を治療又は予防する組成物及び方法 |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040063717A1 (en) | 2002-05-21 | 2004-04-01 | Andrew Wolff | Method of treating diabetes |
| US20130245469A1 (en) * | 2012-03-19 | 2013-09-19 | Cardiomems, Inc. | Pulmonary Arterial Hemodynamic Monitoring for Chronic Obstructive Pulmonary Disease Assessment and Treatment |
| WO2014066870A1 (en) | 2012-10-26 | 2014-05-01 | The Medicines Company | Methods for controlling blood pressure and reducing dyspnea in heart failure |
| WO2014081958A1 (en) | 2012-11-21 | 2014-05-30 | Cardiomems, Inc. | Devices, systems, and methods for pulmonary arterial hypertension (pah) assessment and treatment |
| US9198908B2 (en) | 2013-03-15 | 2015-12-01 | St. Jude Medical Luxembourg Holdings Ii S.A.R.L. (“Sjm Lux Ii”) | Methods for the treatment of cardiovascular conditions |
| KR20190005708A (ko) * | 2017-07-05 | 2019-01-16 | 이화여자대학교 산학협력단 | 에피디티오디옥소피페라진 화합물 또는 이의 유도체, 또는 이들의 약학적으로 허용가능한 염을 포함하는 폐동맥고혈압 예방 또는 치료용 약학적 조성물 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3845770A (en) | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
| US4326525A (en) | 1980-10-14 | 1982-04-27 | Alza Corporation | Osmotic device that improves delivery properties of agent in situ |
| US4567264A (en) | 1983-05-18 | 1986-01-28 | Syntex (U.S.A.) Inc. | Cardioselective aryloxy- and arylthio- hydroxypropylene-piperazinyl acetanilides which affect calcium entry |
| US5364620A (en) | 1983-12-22 | 1994-11-15 | Elan Corporation, Plc | Controlled absorption diltiazem formulation for once daily administration |
| US4902514A (en) | 1988-07-21 | 1990-02-20 | Alza Corporation | Dosage form for administering nilvadipine for treating cardiovascular symptoms |
| US5455045A (en) | 1993-05-13 | 1995-10-03 | Syntex (U.S.A.) Inc. | High dose formulations |
| US6303607B1 (en) | 1998-09-10 | 2001-10-16 | Cv Therapeutics, Inc. | Method for administering a sustained release ranolanolazine formulation |
| KR20070093988A (ko) | 2005-01-06 | 2007-09-19 | 씨브이 쎄러퓨틱스, 인코포레이티드 | 라놀라진 함유 서방성 약제학적 제형물 |
| US20100010024A1 (en) * | 2006-07-01 | 2010-01-14 | Bayer Healthcare Ag | Use of1,4-diaryl-dihydropyrimidine-2-on derivatives for treating pulmonary arterial hypertension |
| WO2010068461A1 (en) | 2008-11-25 | 2010-06-17 | Gilead Palo Alto, Inc. | Co-administration of ranolazine and cardiac glycosides |
-
2011
- 2011-06-10 TW TW100120385A patent/TW201215392A/zh unknown
- 2011-06-14 CA CA2801707A patent/CA2801707A1/en not_active Abandoned
- 2011-06-14 EP EP11726037.2A patent/EP2582372A1/en not_active Withdrawn
- 2011-06-14 UY UY0001033453A patent/UY33453A/es not_active Application Discontinuation
- 2011-06-14 AU AU2011267871A patent/AU2011267871A1/en not_active Abandoned
- 2011-06-14 AR ARP110102063A patent/AR081925A1/es unknown
- 2011-06-14 US US13/160,393 patent/US20120004188A1/en not_active Abandoned
- 2011-06-14 WO PCT/US2011/040363 patent/WO2011159706A1/en not_active Ceased
- 2011-06-14 JP JP2013515456A patent/JP2013528649A/ja not_active Withdrawn
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023542298A (ja) * | 2020-09-11 | 2023-10-06 | プルモシム セラピューティクス リミテッド ライアビリティ カンパニー | 肺高血圧症を治療又は予防する組成物及び方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2801707A1 (en) | 2011-12-22 |
| US20120004188A1 (en) | 2012-01-05 |
| TW201215392A (en) | 2012-04-16 |
| AR081925A1 (es) | 2012-10-31 |
| WO2011159706A1 (en) | 2011-12-22 |
| UY33453A (es) | 2012-01-31 |
| AU2011267871A1 (en) | 2013-01-10 |
| EP2582372A1 (en) | 2013-04-24 |
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