JP2013510155A5 - - Google Patents

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Publication number
JP2013510155A5
JP2013510155A5 JP2012537925A JP2012537925A JP2013510155A5 JP 2013510155 A5 JP2013510155 A5 JP 2013510155A5 JP 2012537925 A JP2012537925 A JP 2012537925A JP 2012537925 A JP2012537925 A JP 2012537925A JP 2013510155 A5 JP2013510155 A5 JP 2013510155A5
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JP
Japan
Prior art keywords
amino
alkyl
quinazolinyl
methyloxy
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2012537925A
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English (en)
Japanese (ja)
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JP2013510155A (ja
JP5836963B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2010/054927 external-priority patent/WO2011056740A1/en
Publication of JP2013510155A publication Critical patent/JP2013510155A/ja
Publication of JP2013510155A5 publication Critical patent/JP2013510155A5/ja
Application granted granted Critical
Publication of JP5836963B2 publication Critical patent/JP5836963B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2012537925A 2009-11-03 2010-11-01 キナゾリン化合物 Expired - Fee Related JP5836963B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25764609P 2009-11-03 2009-11-03
US61/257,646 2009-11-03
PCT/US2010/054927 WO2011056740A1 (en) 2009-11-03 2010-11-01 Quinazoline compounds

Publications (3)

Publication Number Publication Date
JP2013510155A JP2013510155A (ja) 2013-03-21
JP2013510155A5 true JP2013510155A5 (https=) 2013-12-19
JP5836963B2 JP5836963B2 (ja) 2015-12-24

Family

ID=43970282

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012537925A Expired - Fee Related JP5836963B2 (ja) 2009-11-03 2010-11-01 キナゾリン化合物

Country Status (13)

Country Link
US (1) US8859571B2 (https=)
EP (1) EP2501233B1 (https=)
JP (1) JP5836963B2 (https=)
KR (1) KR101736521B1 (https=)
CN (1) CN102711474B (https=)
AU (1) AU2010315361B2 (https=)
BR (1) BR112012010524A2 (https=)
CA (1) CA2779989A1 (https=)
EA (1) EA021439B1 (https=)
ES (1) ES2523465T3 (https=)
IL (1) IL219504A (https=)
MX (1) MX2012005155A (https=)
WO (1) WO2011056740A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5603883B2 (ja) * 2009-02-17 2014-10-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング B−Rafキナーゼを阻害するためのピリミドピリミジン誘導体
CN103159685A (zh) * 2013-04-11 2013-06-19 苏州立新制药有限公司 4-氯-6,7-二(2-甲氧基乙氧基)喹唑啉的制备方法
JP6527513B2 (ja) * 2013-11-20 2019-06-05 シグナルケム・ライフサイエンシーズ・コーポレイションSignalchem Lifesciences Corporation Tamファミリーキナーゼ阻害剤としてのキナゾリン誘導体
CN105849044B (zh) 2013-12-26 2018-10-26 埃克森美孚研究工程公司 Zsm-48晶体的合成
CN111868039A (zh) * 2017-09-26 2020-10-30 加利福尼亚大学董事会 用于治疗癌症的组合物和方法
JP7785663B2 (ja) 2019-09-16 2025-12-15 ノバルティス アーゲー 二機能性分解誘導薬及びそれらの使用方法
WO2023049312A1 (en) 2021-09-23 2023-03-30 Erasca, Inc. Egfr inhibitor polymorph forms

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9508565D0 (en) * 1995-04-27 1995-06-14 Zeneca Ltd Quiazoline derivative
PT2213661E (pt) 2003-09-26 2011-12-15 Exelixis Inc Moduladores de c-met e métodos de uso
CN103626742B (zh) * 2005-11-01 2017-04-26 塔格根公司 激酶的联-芳基间-嘧啶抑制剂

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