JP2013505290A5 - - Google Patents
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- Publication number
- JP2013505290A5 JP2013505290A5 JP2012530363A JP2012530363A JP2013505290A5 JP 2013505290 A5 JP2013505290 A5 JP 2013505290A5 JP 2012530363 A JP2012530363 A JP 2012530363A JP 2012530363 A JP2012530363 A JP 2012530363A JP 2013505290 A5 JP2013505290 A5 JP 2013505290A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- dihydropyrrolo
- pyrazol
- oxy
- piperidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24506909P | 2009-09-23 | 2009-09-23 | |
| US61/245,069 | 2009-09-23 | ||
| PCT/IB2010/053347 WO2011036576A1 (en) | 2009-09-23 | 2010-07-22 | Gpr 119 modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013505290A JP2013505290A (ja) | 2013-02-14 |
| JP2013505290A5 true JP2013505290A5 (https=) | 2013-07-25 |
Family
ID=42799871
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012530363A Withdrawn JP2013505290A (ja) | 2009-09-23 | 2010-07-22 | Ｇｐｒ１１９調節因子 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20130072427A1 (https=) |
| EP (1) | EP2480551A1 (https=) |
| JP (1) | JP2013505290A (https=) |
| CA (1) | CA2772188A1 (https=) |
| WO (1) | WO2011036576A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101913619B1 (ko) | 2011-06-09 | 2018-12-28 | 리젠 파마슈티컬스 소시에떼 아노님 | Gpr-119의 조절제로서의 신규한 화합물 |
| EP2780026B1 (en) | 2011-11-15 | 2019-10-23 | Merck Sharp & Dohme Corp. | Hcv ns3 protease inhibitors |
| CA2878625A1 (en) | 2012-07-11 | 2014-01-16 | Elcelyx Therapeutics, Inc. | Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk |
| RU2015118647A (ru) | 2012-11-20 | 2017-01-10 | Дженентек, Инк. | Аминопиримидиновые соединения в качестве ингибиторов содержащих т790м мутантных egfr |
| LT3728207T (lt) | 2017-12-21 | 2023-05-25 | Ribon Therapeutics Inc. | Chinazolinonai kaip parp14 inhibitoriai |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3839694A1 (de) | 1988-11-24 | 1990-05-31 | Ats Leichtmetallraeder Gmbh | Faltschachtel zur verpackung eines stossempfindlichen produkts, insbesondere einer leichtmetallfelge |
| ES1011809Y (es) | 1989-10-23 | 1991-08-01 | Minano Iglesias Jesus | Muneco-envase. |
| IL157253A0 (en) | 2001-02-28 | 2004-02-19 | Merck & Co Inc | Acylated piperidine derivatives as melanocortin-4 receptor agonists |
| US7135575B2 (en) * | 2003-03-03 | 2006-11-14 | Array Biopharma, Inc. | P38 inhibitors and methods of use thereof |
| UA84208C2 (en) | 2004-05-25 | 2008-09-25 | Пфайзер Продактс Инк. | Tetraazabenzo(e)azulene derivatives and analogs thereof |
| PA8660701A1 (es) | 2005-02-04 | 2006-09-22 | Pfizer Prod Inc | Agonistas de pyy y sus usos |
| CA2636757A1 (en) * | 2006-01-25 | 2007-08-02 | Tesfaye Biftu | Aminocyclohexanes as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes |
| TW200806669A (en) * | 2006-03-28 | 2008-02-01 | Merck & Co Inc | Aminotetrahydropyrans as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes |
| WO2008137436A1 (en) * | 2007-05-04 | 2008-11-13 | Bristol-Myers Squibb Company | [6,5]-bicyclic gpr119 g protein-coupled receptor agonists |
| AU2008279447A1 (en) | 2007-07-19 | 2009-01-29 | Metabolex, Inc. | N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders |
| JP5009736B2 (ja) | 2007-10-15 | 2012-08-22 | 日本曹達株式会社 | 環状アミノエーテルを用いたマンニッヒ反応 |
| EP2504342A1 (en) * | 2009-11-23 | 2012-10-03 | Pfizer Inc. | Imidazo-pyrazoles as gpr119 inhibitors |
-
2010
- 2010-07-22 US US13/392,935 patent/US20130072427A1/en not_active Abandoned
- 2010-07-22 JP JP2012530363A patent/JP2013505290A/ja not_active Withdrawn
- 2010-07-22 CA CA2772188A patent/CA2772188A1/en not_active Abandoned
- 2010-07-22 WO PCT/IB2010/053347 patent/WO2011036576A1/en not_active Ceased
- 2010-07-22 EP EP10747074A patent/EP2480551A1/en not_active Withdrawn
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