JP2013503134A5 - - Google Patents
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- Publication number
- JP2013503134A5 JP2013503134A5 JP2012526048A JP2012526048A JP2013503134A5 JP 2013503134 A5 JP2013503134 A5 JP 2013503134A5 JP 2012526048 A JP2012526048 A JP 2012526048A JP 2012526048 A JP2012526048 A JP 2012526048A JP 2013503134 A5 JP2013503134 A5 JP 2013503134A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- anhydrous crystalline
- crystalline form
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23743509P | 2009-08-27 | 2009-08-27 | |
| US61/237,435 | 2009-08-27 | ||
| PCT/EP2010/062420 WO2011023733A1 (en) | 2009-08-27 | 2010-08-25 | Anhydrate forms of a pyridine derivative |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015139845A Division JP6404186B2 (ja) | 2009-08-27 | 2015-07-13 | 無水形態のピリジン誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013503134A JP2013503134A (ja) | 2013-01-31 |
| JP2013503134A5 true JP2013503134A5 (https=) | 2013-09-19 |
Family
ID=42790943
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012526048A Pending JP2013503134A (ja) | 2009-08-27 | 2010-08-25 | 無水形態のピリジン誘導体 |
| JP2015139845A Active JP6404186B2 (ja) | 2009-08-27 | 2015-07-13 | 無水形態のピリジン誘導体 |
| JP2017114602A Pending JP2017193564A (ja) | 2009-08-27 | 2017-06-09 | 無水形態のピリジン誘導体 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015139845A Active JP6404186B2 (ja) | 2009-08-27 | 2015-07-13 | 無水形態のピリジン誘導体 |
| JP2017114602A Pending JP2017193564A (ja) | 2009-08-27 | 2017-06-09 | 無水形態のピリジン誘導体 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US8796269B2 (https=) |
| EP (1) | EP2470545B1 (https=) |
| JP (3) | JP2013503134A (https=) |
| KR (1) | KR20120056258A (https=) |
| CN (1) | CN102639536B (https=) |
| AU (1) | AU2010288502B2 (https=) |
| CA (1) | CA2772168C (https=) |
| DK (1) | DK2470545T3 (https=) |
| EA (1) | EA021411B1 (https=) |
| ES (1) | ES2440938T3 (https=) |
| IL (1) | IL217922A (https=) |
| IN (1) | IN2012DN01292A (https=) |
| MX (1) | MX2012002369A (https=) |
| PL (1) | PL2470545T3 (https=) |
| SG (1) | SG178231A1 (https=) |
| WO (1) | WO2011023733A1 (https=) |
| ZA (1) | ZA201200812B (https=) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102639536B (zh) * | 2009-08-27 | 2015-03-18 | 尼尔医疗有限公司 | 吡啶衍生物的无水晶型 |
| WO2015200594A2 (en) | 2014-06-25 | 2015-12-30 | Emory University | Methods of managing conditioned fear with neurokinin receptor antagonists |
| EP3574907B1 (en) * | 2015-05-18 | 2023-08-23 | KaNDy Therapeutics Limited | A dual nk-1/nk-3 receptor antagonist for the treatment of sex-hormone-dependent diseases |
| CA3044773A1 (en) * | 2016-12-15 | 2018-06-21 | Glaxosmithkline Intellectual Property Development Limited | Nrf2 activators |
| JP7433252B2 (ja) * | 2018-03-14 | 2024-02-19 | キャンディ・セラピューティクス・リミテッド | Ｎｋ－１／ｎｋ－３受容体二重アンタゴニストを含む新規な医薬製剤 |
| WO2021030335A1 (en) * | 2019-08-12 | 2021-02-18 | Millendo Therapeutics, Inc. | A stereoisomerically pure nk-3 receptor antagonist and crystalline forms thereof |
| KR102950227B1 (ko) | 2019-11-15 | 2026-04-08 | 칸디 테라퓨틱스 리미티드 | Nt-814의 핵심 중간체인 6-클로로-4-(4-플루오로-2-메틸페닐)피리딘-3-아민의 새로운 화학적 제조 방법 |
| EP4431512A1 (en) | 2023-03-16 | 2024-09-18 | Bayer Consumer Care AG | Novel dual nk-1/nk-3 receptor antagonists |
| WO2025242584A1 (en) | 2024-05-24 | 2025-11-27 | Bayer Consumer Care Ag | A stable soft gelatin capsule formulation for elinzanetant |
| WO2025242585A1 (en) | 2024-05-24 | 2025-11-27 | Bayer Consumer Care Ag | Crystalline forms of salts of elinzanetant and compositions containing salts of elinzanetant |
| WO2025242583A1 (en) | 2024-05-24 | 2025-11-27 | Bayer Consumer Care Ag | Novel formulation comprising elinzanetant in a solid dispersion |
| WO2025261856A1 (en) * | 2024-06-18 | 2025-12-26 | Bayer Consumer Care Ag | Improved process for producing an elinzanetant precursor |
| US12533358B1 (en) | 2025-05-14 | 2026-01-27 | Bayer Consumer Care Ag | Methods of treatment with elinzanetant |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1394150B1 (en) * | 1999-02-24 | 2011-01-19 | F. Hoffmann-La Roche AG | 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists |
| GB0203022D0 (en) * | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
| ATE366576T1 (de) * | 2003-01-31 | 2007-08-15 | Hoffmann La Roche | Neue kristallmodifikation von 2-(3,5-bis- trifluormethyl-phenyl)-n-6-(1,1-dioxo-1lamda-6- |
| SI1643998T1 (sl) * | 2003-07-03 | 2007-12-31 | Hoffmann La Roche | Dvojni nk1/nk3 antagonisti za zdravljenje shizofrenije |
| EP1928886B1 (en) * | 2005-09-09 | 2011-04-13 | GlaxoSmithKline LLC | Pyridine derivatives and their use in the treatment of psychotic disorders |
| WO2009087667A2 (en) * | 2007-12-11 | 2009-07-16 | Cipla Ltd. | A new method for preparation of zopiclone and its polymorphs |
| GB0814340D0 (en) * | 2008-08-05 | 2008-09-10 | Smithkline Beecham Corp | Anhydrous crystol form fo a pyridine derivative |
| CN102639536B (zh) * | 2009-08-27 | 2015-03-18 | 尼尔医疗有限公司 | 吡啶衍生物的无水晶型 |
| JP6342662B2 (ja) * | 2014-01-29 | 2018-06-13 | 京セラ株式会社 | ドリルおよびそれを用いた切削加工物の製造方法 |
-
2010
- 2010-08-25 CN CN201080037918.3A patent/CN102639536B/zh active Active
- 2010-08-25 US US13/389,525 patent/US8796269B2/en active Active
- 2010-08-25 WO PCT/EP2010/062420 patent/WO2011023733A1/en not_active Ceased
- 2010-08-25 DK DK10747619.4T patent/DK2470545T3/da active
- 2010-08-25 SG SG2012007464A patent/SG178231A1/en unknown
- 2010-08-25 AU AU2010288502A patent/AU2010288502B2/en active Active
- 2010-08-25 PL PL10747619T patent/PL2470545T3/pl unknown
- 2010-08-25 KR KR1020127004865A patent/KR20120056258A/ko not_active Ceased
- 2010-08-25 EA EA201270302A patent/EA021411B1/ru not_active IP Right Cessation
- 2010-08-25 CA CA2772168A patent/CA2772168C/en active Active
- 2010-08-25 JP JP2012526048A patent/JP2013503134A/ja active Pending
- 2010-08-25 EP EP10747619.4A patent/EP2470545B1/en active Active
- 2010-08-25 IN IN1292DEN2012 patent/IN2012DN01292A/en unknown
- 2010-08-25 ES ES10747619.4T patent/ES2440938T3/es active Active
- 2010-08-25 MX MX2012002369A patent/MX2012002369A/es active IP Right Grant
-
2012
- 2012-02-02 ZA ZA2012/00812A patent/ZA201200812B/en unknown
- 2012-02-02 IL IL217922A patent/IL217922A/en active IP Right Grant
-
2015
- 2015-07-13 JP JP2015139845A patent/JP6404186B2/ja active Active
-
2017
- 2017-06-09 JP JP2017114602A patent/JP2017193564A/ja active Pending
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