JP2012526772A - ホスホイノシチド３−キナーゼ阻害剤および抗糖尿病性化合物の組合せ剤 - Google Patents
ホスホイノシチド３−キナーゼ阻害剤および抗糖尿病性化合物の組合せ剤 Download PDFInfo
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Landscapes
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021525802A (ja) * | 2018-06-01 | 2021-09-27 | コーネル・ユニバーシティーＣｏｒｎｅｌｌ Ｕｎｉｖｅｒｓｉｔｙ | Ｐｉ３ｋに関連する疾患または障害に対する併用療法 |
| JP2021532139A (ja) * | 2018-07-23 | 2021-11-25 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | Ｐｉ３ｋ阻害剤であるｇｄｃ−００７７による癌の治療方法 |
| JP2022504388A (ja) * | 2018-10-08 | 2022-01-13 | エフ・ホフマン－ラ・ロシュ・アクチェンゲゼルシャフト | Ｐｉ３ｋアルファ阻害剤およびメトホルミンを用いたがんの処置方法 |
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| AR081060A1 (es) | 2010-04-15 | 2012-06-06 | Bayer Schering Pharma Ag | Procedimiento para preparar 4-{4-[({[4-cloro-3-(trifluorometil)fenil]amino}carbonil)amino]-3-fluorofenoxi}-n-metilpiridin-2-carboxamida |
| CN104945373A (zh) * | 2010-10-01 | 2015-09-30 | 诺华有限公司 | 制造嘧啶衍生物的方法 |
| SG11201509707QA (en) | 2013-04-12 | 2015-12-30 | Rebecca Lambert Bent | Cancer therapy |
| MX2019001467A (es) * | 2016-08-03 | 2019-10-02 | Remd Biotherapeutics Inc | Combinación de antagonistas del receptor de glucagon e inhibidores de la trayectoria p13k para el tratamiento del cáncer. |
| AU2020407573A1 (en) * | 2019-12-20 | 2022-07-14 | Recurium Ip Holdings, Llc | Combinations |
| CN120361228B (zh) * | 2025-04-08 | 2025-11-21 | 复旦大学附属妇产科医院 | 一种葡萄糖激酶激活剂与pi3k抑制剂的组合物 |
Citations (4)
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| JP2006516620A (ja) * | 2003-01-24 | 2006-07-06 | ブリストル−マイヤーズ スクイブ カンパニー | 甲状腺受容体におけるシクロアルキル含有アニリドリガンド |
| WO2007084786A1 (en) * | 2006-01-20 | 2007-07-26 | Novartis Ag | Pyrimidine derivatives used as pi-3 kinase inhibitors |
| JP2008540599A (ja) * | 2005-05-20 | 2008-11-20 | ノバルティス アクチエンゲゼルシャフト | 脂質キナーゼ阻害剤としてのイミダゾキノリン |
| JP2009500408A (ja) * | 2004-07-09 | 2009-01-08 | プロルックス ファーマシューティカルズ コープ． | ワートマニン類似体及び化学療法薬と組み合わせた同一物を使用する方法 |
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| WO2006069186A2 (en) * | 2004-12-22 | 2006-06-29 | The Ohio State Research Foundation | Small molecule bcl-xl/bcl-2 binding inhibitors |
| US20080044390A1 (en) * | 2006-08-11 | 2008-02-21 | Xiaowei Jin | Methods and compositions for the treatment of neurodegenerative disorders |
| EP2120909A2 (en) * | 2006-12-15 | 2009-11-25 | Ordway Research Institute | Treatments of therapy-resistant diseases comprising drug combinations |
| AU2008335469A1 (en) * | 2007-12-13 | 2009-06-18 | Novartis Ag | Combinations of therapeutic agents for treating cancer |
| WO2009155659A1 (en) * | 2008-06-27 | 2009-12-30 | The University Of Queensland | Combination therapy |
| KR20110028651A (ko) * | 2008-07-11 | 2011-03-21 | 노파르티스 아게 | (ａ) 포스포이노시타이드 3-키나제 억제제 및 (ｂ) ｒａｓ/ｒａｆ/ｍｅｋ 경로의 조절제의 조합물 |
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2010
- 2010-05-12 CA CA2760179A patent/CA2760179A1/en not_active Abandoned
- 2010-05-12 MX MX2011012201A patent/MX2011012201A/es not_active Application Discontinuation
- 2010-05-12 US US13/319,536 patent/US20120059005A1/en not_active Abandoned
- 2010-05-12 EP EP10718226A patent/EP2429516A2/en not_active Withdrawn
- 2010-05-12 JP JP2012510289A patent/JP2012526772A/ja active Pending
- 2010-05-12 RU RU2011150619/02A patent/RU2011150619A/ru not_active Application Discontinuation
- 2010-05-12 KR KR1020117027030A patent/KR20120096869A/ko not_active Withdrawn
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- 2010-05-12 BR BRPI1010979A patent/BRPI1010979A2/pt not_active IP Right Cessation
- 2010-05-12 CN CN2010800199053A patent/CN102958518A/zh active Pending
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006516620A (ja) * | 2003-01-24 | 2006-07-06 | ブリストル−マイヤーズ スクイブ カンパニー | 甲状腺受容体におけるシクロアルキル含有アニリドリガンド |
| JP2009500408A (ja) * | 2004-07-09 | 2009-01-08 | プロルックス ファーマシューティカルズ コープ． | ワートマニン類似体及び化学療法薬と組み合わせた同一物を使用する方法 |
| JP2008540599A (ja) * | 2005-05-20 | 2008-11-20 | ノバルティス アクチエンゲゼルシャフト | 脂質キナーゼ阻害剤としてのイミダゾキノリン |
| WO2007084786A1 (en) * | 2006-01-20 | 2007-07-26 | Novartis Ag | Pyrimidine derivatives used as pi-3 kinase inhibitors |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021525802A (ja) * | 2018-06-01 | 2021-09-27 | コーネル・ユニバーシティーＣｏｒｎｅｌｌ Ｕｎｉｖｅｒｓｉｔｙ | Ｐｉ３ｋに関連する疾患または障害に対する併用療法 |
| US12324807B2 (en) | 2018-06-01 | 2025-06-10 | Cornell University | Combination therapy for PI3K-associated disease or disorder |
| JP2025160313A (ja) * | 2018-06-01 | 2025-10-22 | コーネル・ユニバーシティー | Ｐｉ３ｋに関連する疾患または障害に対する併用療法 |
| JP7768505B2 (ja) | 2018-06-01 | 2025-11-12 | コーネル・ユニバーシティー | Ｐｉ３ｋに関連する疾患または障害に対する併用療法 |
| JP2021532139A (ja) * | 2018-07-23 | 2021-11-25 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | Ｐｉ３ｋ阻害剤であるｇｄｃ−００７７による癌の治療方法 |
| JP2024001009A (ja) * | 2018-07-23 | 2024-01-09 | エフ・ホフマン－ラ・ロシュ・アクチェンゲゼルシャフト | Ｐｉ３ｋ阻害剤であるｇｄｃ－００７７による癌の治療方法 |
| JP2022504388A (ja) * | 2018-10-08 | 2022-01-13 | エフ・ホフマン－ラ・ロシュ・アクチェンゲゼルシャフト | Ｐｉ３ｋアルファ阻害剤およびメトホルミンを用いたがんの処置方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| CN102958518A (zh) | 2013-03-06 |
| WO2010130779A2 (en) | 2010-11-18 |
| US20120059005A1 (en) | 2012-03-08 |
| BRPI1010979A2 (pt) | 2018-03-06 |
| CA2760179A1 (en) | 2010-11-18 |
| RU2011150619A (ru) | 2013-06-20 |
| KR20120096869A (ko) | 2012-08-31 |
| EP2429516A2 (en) | 2012-03-21 |
| AU2010247397B2 (en) | 2012-07-12 |
| WO2010130779A3 (en) | 2013-03-28 |
| AU2010247397A1 (en) | 2011-11-03 |
| MX2011012201A (es) | 2011-12-08 |
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