JP2012515776A5 - - Google Patents

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Publication number
JP2012515776A5
JP2012515776A5 JP2011547997A JP2011547997A JP2012515776A5 JP 2012515776 A5 JP2012515776 A5 JP 2012515776A5 JP 2011547997 A JP2011547997 A JP 2011547997A JP 2011547997 A JP2011547997 A JP 2011547997A JP 2012515776 A5 JP2012515776 A5 JP 2012515776A5
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JP
Japan
Prior art keywords
group
compound
salt according
heteroaryl
alkynyl
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Application number
JP2011547997A
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English (en)
Japanese (ja)
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JP2012515776A (ja
JP5576402B2 (ja
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Priority claimed from PCT/US2010/020373 external-priority patent/WO2010085377A2/en
Publication of JP2012515776A publication Critical patent/JP2012515776A/ja
Publication of JP2012515776A5 publication Critical patent/JP2012515776A5/ja
Application granted granted Critical
Publication of JP5576402B2 publication Critical patent/JP5576402B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011547997A 2009-01-23 2010-01-07 ヒドロキサム酸誘導体 Active JP5576402B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US14700209P 2009-01-23 2009-01-23
US61/147,002 2009-01-23
US15649609P 2009-02-28 2009-02-28
US61/156,496 2009-02-28
US25215609P 2009-10-15 2009-10-15
US61/252,156 2009-10-15
US25265209P 2009-10-17 2009-10-17
US61/252,652 2009-10-17
PCT/US2010/020373 WO2010085377A2 (en) 2009-01-23 2010-01-07 Hydroxamic acid derivatives

Publications (3)

Publication Number Publication Date
JP2012515776A JP2012515776A (ja) 2012-07-12
JP2012515776A5 true JP2012515776A5 (US07585860-20090908-C00112.png) 2013-02-21
JP5576402B2 JP5576402B2 (ja) 2014-08-20

Family

ID=42356377

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011547997A Active JP5576402B2 (ja) 2009-01-23 2010-01-07 ヒドロキサム酸誘導体

Country Status (17)

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US (3) US8609864B2 (US07585860-20090908-C00112.png)
EP (1) EP2389375B1 (US07585860-20090908-C00112.png)
JP (1) JP5576402B2 (US07585860-20090908-C00112.png)
CN (1) CN102186842B (US07585860-20090908-C00112.png)
CA (1) CA2750413C (US07585860-20090908-C00112.png)
CY (1) CY1116602T1 (US07585860-20090908-C00112.png)
DK (1) DK2389375T3 (US07585860-20090908-C00112.png)
ES (1) ES2544803T3 (US07585860-20090908-C00112.png)
HR (1) HRP20150778T1 (US07585860-20090908-C00112.png)
HU (1) HUE025349T2 (US07585860-20090908-C00112.png)
ME (1) ME02254B (US07585860-20090908-C00112.png)
PL (1) PL2389375T3 (US07585860-20090908-C00112.png)
PT (1) PT2389375E (US07585860-20090908-C00112.png)
RS (1) RS54192B1 (US07585860-20090908-C00112.png)
SI (1) SI2389375T1 (US07585860-20090908-C00112.png)
SM (1) SMT201500196B (US07585860-20090908-C00112.png)
WO (1) WO2010085377A2 (US07585860-20090908-C00112.png)

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UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
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WO2012096832A2 (en) * 2011-01-12 2012-07-19 Crystal Biopharmaceutical Llc Hdac inhibiting derivatives of camptothecin
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CN102432654A (zh) * 2011-09-26 2012-05-02 宋云龙 吉西他滨酰胺衍生物及其制备方法和用途
AR092790A1 (es) * 2012-02-01 2015-05-06 Euro Celtique Sa Derivados bencimidazolicos del acido hidroxamico
CN102584737A (zh) * 2012-02-07 2012-07-18 盛世泰科生物医药技术(苏州)有限公司 抑制组蛋白去乙酰酶的物质的组成和使用
EP2725029A1 (en) * 2012-10-29 2014-04-30 Laboratoire Biodim New antibacterial compounds and biological applications thereof
EP2945634A4 (en) 2012-12-28 2016-05-25 Dow Agrosciences Llc N- (SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDIN-1 (2H) -CARBOXAMIDE DERIVATIVES
RU2656101C2 (ru) 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
AU2013370493B2 (en) 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN103340845B (zh) * 2013-06-26 2015-03-18 浙江省食品药品检验研究院 药物组合物
US9944670B2 (en) * 2013-12-04 2018-04-17 Hangzhou Yuanchang Medical Sci-Tech Co., Ltd Gemcitabine derivatives, compositions comprising same and pharmaceutical applications thereof
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
UA122200C2 (uk) 2013-12-31 2020-10-12 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
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CN106883217B (zh) * 2017-04-01 2020-05-22 清华大学深圳研究生院 一种核苷碱基异羟肟酸衍生化合物及其制备方法与应用
GB201709403D0 (en) 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating sarcoma
GB201709406D0 (en) 2017-06-13 2017-07-26 Euro-Cletique S A Compounds for treating TNBC
GB201709402D0 (en) 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating t-pll
GB201709405D0 (en) * 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating ovarian cancer
EP3659307A4 (en) * 2017-07-28 2021-09-22 Yale University ANTI-CANCER MEDICINAL PRODUCTS AND THEIR MANUFACTURING AND USE PROCEDURES
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CN108299313B (zh) * 2018-01-16 2020-10-02 长沙霍滋生物科技有限公司 一种化合物及其在药学上的应用
CN109516957A (zh) * 2018-08-03 2019-03-26 杭州梯诺医药科技有限公司 Nl-101多晶型及其制备方法
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