JP2012509321A5 - - Google Patents

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Publication number
JP2012509321A5
JP2012509321A5 JP2011537428A JP2011537428A JP2012509321A5 JP 2012509321 A5 JP2012509321 A5 JP 2012509321A5 JP 2011537428 A JP2011537428 A JP 2011537428A JP 2011537428 A JP2011537428 A JP 2011537428A JP 2012509321 A5 JP2012509321 A5 JP 2012509321A5
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JP
Japan
Prior art keywords
pharmaceutical composition
compound
ray powder
disintegrant
powder diffraction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011537428A
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English (en)
Japanese (ja)
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JP2012509321A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/006235 external-priority patent/WO2010059239A2/en
Publication of JP2012509321A publication Critical patent/JP2012509321A/ja
Publication of JP2012509321A5 publication Critical patent/JP2012509321A5/ja
Pending legal-status Critical Current

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JP2011537428A 2008-11-21 2009-11-20 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物 Pending JP2012509321A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US19988808P 2008-11-21 2008-11-21
US61/199,888 2008-11-21
US21039809P 2009-03-17 2009-03-17
US61/210,398 2009-03-17
PCT/US2009/006235 WO2010059239A2 (en) 2008-11-21 2009-11-20 Lactate salt of 4-(6-methoxy-7-(3-piperidin-1-yl-propoxy)quinazolin-4-yl]piperazine-1-carboxylic acid(4-isopropoxyphenyl)-amide and pharmaceutical compositions thereof for the treatment of cancer and other diseases or disorders

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014193355A Division JP2015017116A (ja) 2008-11-21 2014-09-24 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物

Publications (2)

Publication Number Publication Date
JP2012509321A JP2012509321A (ja) 2012-04-19
JP2012509321A5 true JP2012509321A5 (enExample) 2012-12-27

Family

ID=41508688

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2011537428A Pending JP2012509321A (ja) 2008-11-21 2009-11-20 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物
JP2014193355A Pending JP2015017116A (ja) 2008-11-21 2014-09-24 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2014193355A Pending JP2015017116A (ja) 2008-11-21 2014-09-24 癌および他の疾患または障害の処置のための、４−［６−メトキシ−７−（３−ピペリジン−１−イル−プロポキシ）キナゾリン−４−イル］ピペラジン−１−カルボン酸（４−イソプロポキシフェニル）−アミドの乳酸塩およびその薬学的組成物

Country Status (4)

Country Link
US (1) US20100273808A1 (enExample)
EP (1) EP2370417A2 (enExample)
JP (2) JP2012509321A (enExample)
WO (1) WO2010059239A2 (enExample)

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EP3064595B1 (en) 2009-10-21 2019-02-27 Agios Pharmaceuticals, Inc. Methods for cell-proliferation-related disorders
CN103764147B (zh) 2011-05-03 2018-05-22 安吉奥斯医药品有限公司 用于治疗的丙酮酸激酶活化剂
CN102827170A (zh) 2011-06-17 2012-12-19 安吉奥斯医药品有限公司 治疗活性组合物和它们的使用方法
CN102827073A (zh) 2011-06-17 2012-12-19 安吉奥斯医药品有限公司 治疗活性组合物和它们的使用方法
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AU2014287121B2 (en) 2013-07-11 2018-11-15 Agios Pharmaceuticals, Inc. 2,4- or 4,6-diaminopyrimidine compounds as IDH2 mutants inhibitors for the treatment of cancer
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JP6564796B2 (ja) * 2014-03-14 2019-08-21 アジオス ファーマシューティカルズ， インコーポレイテッド 治療活性化合物の医薬組成物
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