JP2012508726A - ベンゾイミダゾール誘導体及びgabaaレセプター複合体を調節するためのそれらの使用 - Google Patents

ベンゾイミダゾール誘導体及びgabaaレセプター複合体を調節するためのそれらの使用 Download PDF

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JP2012508726A
JP2012508726A JP2011536026A JP2011536026A JP2012508726A JP 2012508726 A JP2012508726 A JP 2012508726A JP 2011536026 A JP2011536026 A JP 2011536026A JP 2011536026 A JP2011536026 A JP 2011536026A JP 2012508726 A JP2012508726 A JP 2012508726A
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disorder
stereoisomers
pain
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disease
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JP2012508726A5 (https=
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ラルセン、ヤヌス、エス.
アフリング、フィリップ、ケイ.
ニールセン、エルセベト、エステルガード
ミルザ、ナヒード
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ノイロサーチ アクティーゼルスカブ
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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

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  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2011536026A 2008-11-14 2009-11-13 ベンゾイミダゾール誘導体及びgabaaレセプター複合体を調節するためのそれらの使用 Abandoned JP2012508726A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US11496008P 2008-11-14 2008-11-14
DKPA200801584 2008-11-14
US61/114,960 2008-11-14
DKPA200801584 2008-11-14
PCT/EP2009/065121 WO2010055128A1 (en) 2008-11-14 2009-11-13 Benzimidazole derivatives and their use for modulating the gabaa receptor complex

Publications (2)

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JP2012508726A true JP2012508726A (ja) 2012-04-12
JP2012508726A5 JP2012508726A5 (https=) 2012-12-27

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JP2011536026A Abandoned JP2012508726A (ja) 2008-11-14 2009-11-13 ベンゾイミダゾール誘導体及びgabaaレセプター複合体を調節するためのそれらの使用

Country Status (9)

Country Link
US (1) US20110257210A1 (https=)
EP (1) EP2358701A1 (https=)
JP (1) JP2012508726A (https=)
CN (1) CN102388035A (https=)
AR (1) AR074342A1 (https=)
CA (1) CA2743531A1 (https=)
MX (1) MX2011004736A (https=)
TW (1) TW201029989A (https=)
WO (1) WO2010055128A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8519134B2 (en) 2009-11-17 2013-08-27 Novartis Ag Aryl-pyridine derivatives as aldosterone synthase inhibitors
CN114807015B (zh) * 2022-05-20 2022-11-22 呈诺再生医学科技(北京)有限公司 一种促进胰岛α细胞转化为β细胞的诱导方法及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6900215B2 (en) * 2000-12-15 2005-05-31 Merck Sharp & Dohme Ltd. Imidazo-pyrimidine derivatives as ligands for gaba receptors
TWI391381B (zh) * 2006-03-24 2013-04-01 Neurosearch As 新穎的苯并咪唑衍生物、含有其之醫藥組成物、及其於製造藥物之用途

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Publication number Publication date
AR074342A1 (es) 2011-01-12
US20110257210A1 (en) 2011-10-20
CN102388035A (zh) 2012-03-21
EP2358701A1 (en) 2011-08-24
MX2011004736A (es) 2011-10-12
CA2743531A1 (en) 2010-05-20
WO2010055128A1 (en) 2010-05-20
TW201029989A (en) 2010-08-16

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