MX2011004736A - Derivados de benzimidazol y su uso para modular el complejo del receptor gaba a. - Google Patents
Derivados de benzimidazol y su uso para modular el complejo del receptor gaba a.Info
- Publication number
- MX2011004736A MX2011004736A MX2011004736A MX2011004736A MX2011004736A MX 2011004736 A MX2011004736 A MX 2011004736A MX 2011004736 A MX2011004736 A MX 2011004736A MX 2011004736 A MX2011004736 A MX 2011004736A MX 2011004736 A MX2011004736 A MX 2011004736A
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- Mexico
- Prior art keywords
- disorder
- pain
- stereoisomers
- fluoro
- disease
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- KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 description 1
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- CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical compound FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Engineering & Computer Science (AREA)
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- Public Health (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
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- Heart & Thoracic Surgery (AREA)
- Transplantation (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11496008P | 2008-11-14 | 2008-11-14 | |
| DKPA200801584 | 2008-11-14 | ||
| PCT/EP2009/065121 WO2010055128A1 (en) | 2008-11-14 | 2009-11-13 | Benzimidazole derivatives and their use for modulating the gabaa receptor complex |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2011004736A true MX2011004736A (es) | 2011-10-12 |
Family
ID=41563731
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2011004736A MX2011004736A (es) | 2008-11-14 | 2009-11-13 | Derivados de benzimidazol y su uso para modular el complejo del receptor gaba a. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20110257210A1 (https=) |
| EP (1) | EP2358701A1 (https=) |
| JP (1) | JP2012508726A (https=) |
| CN (1) | CN102388035A (https=) |
| AR (1) | AR074342A1 (https=) |
| CA (1) | CA2743531A1 (https=) |
| MX (1) | MX2011004736A (https=) |
| TW (1) | TW201029989A (https=) |
| WO (1) | WO2010055128A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8519134B2 (en) | 2009-11-17 | 2013-08-27 | Novartis Ag | Aryl-pyridine derivatives as aldosterone synthase inhibitors |
| CN114807015B (zh) * | 2022-05-20 | 2022-11-22 | 呈诺再生医学科技(北京)有限公司 | 一种促进胰岛α细胞转化为β细胞的诱导方法及其应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6900215B2 (en) * | 2000-12-15 | 2005-05-31 | Merck Sharp & Dohme Ltd. | Imidazo-pyrimidine derivatives as ligands for gaba receptors |
| TWI391381B (zh) * | 2006-03-24 | 2013-04-01 | Neurosearch As | 新穎的苯并咪唑衍生物、含有其之醫藥組成物、及其於製造藥物之用途 |
-
2009
- 2009-11-05 TW TW098137558A patent/TW201029989A/zh unknown
- 2009-11-13 MX MX2011004736A patent/MX2011004736A/es not_active Application Discontinuation
- 2009-11-13 EP EP09756151A patent/EP2358701A1/en not_active Withdrawn
- 2009-11-13 CN CN2009801454691A patent/CN102388035A/zh active Pending
- 2009-11-13 AR ARP090104401A patent/AR074342A1/es unknown
- 2009-11-13 CA CA2743531A patent/CA2743531A1/en not_active Abandoned
- 2009-11-13 US US13/129,186 patent/US20110257210A1/en not_active Abandoned
- 2009-11-13 WO PCT/EP2009/065121 patent/WO2010055128A1/en not_active Ceased
- 2009-11-13 JP JP2011536026A patent/JP2012508726A/ja not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AR074342A1 (es) | 2011-01-12 |
| US20110257210A1 (en) | 2011-10-20 |
| CN102388035A (zh) | 2012-03-21 |
| EP2358701A1 (en) | 2011-08-24 |
| JP2012508726A (ja) | 2012-04-12 |
| CA2743531A1 (en) | 2010-05-20 |
| WO2010055128A1 (en) | 2010-05-20 |
| TW201029989A (en) | 2010-08-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |