JP2012012417A5 - - Google Patents
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- JP2012012417A5 JP2012012417A5 JP2011227135A JP2011227135A JP2012012417A5 JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5 JP 2011227135 A JP2011227135 A JP 2011227135A JP 2011227135 A JP2011227135 A JP 2011227135A JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5
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- JP
- Japan
- Prior art keywords
- compound
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- Prior art date
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- 0 *c1c(-c2c[n]c3c2c(*)c(*)cn3)nc(*)[s]1 Chemical compound *c1c(-c2c[n]c3c2c(*)c(*)cn3)nc(*)[s]1 0.000 description 1
Applications Claiming Priority (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US58438304P | 2004-06-30 | 2004-06-30 | |
US60/584,383 | 2004-06-30 | ||
US58472104P | 2004-07-01 | 2004-07-01 | |
US60/584,721 | 2004-07-01 | ||
US11/098,751 | 2005-04-04 | ||
US11/098,751 US7514448B2 (en) | 2004-04-02 | 2005-04-04 | Azaindoles useful as inhibitors of rock and other protein kinases |
PCT/US2005/011358 WO2005103050A2 (fr) | 2004-04-02 | 2005-04-04 | Azaindoles utiles en tant qu'inhibiteurs de la proteine serine/threonine kinase superhelice de la famille rho (rock) et d'autres proteines kinases |
USPCT/US05/11358 | 2005-04-04 |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2007519460A Division JP5122280B2 (ja) | 2004-06-30 | 2005-06-29 | タンパク質キナーゼのインヒビターとして有用なアザインドール |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2013001760A Division JP2013064015A (ja) | 2004-06-30 | 2013-01-09 | タンパク質キナーゼのインヒビターとして有用なアザインドール |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2012012417A JP2012012417A (ja) | 2012-01-19 |
JP2012012417A5 true JP2012012417A5 (fr) | 2013-02-28 |
Family
ID=37801682
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2007519460A Expired - Fee Related JP5122280B2 (ja) | 2004-06-30 | 2005-06-29 | タンパク質キナーゼのインヒビターとして有用なアザインドール |
JP2011227135A Pending JP2012012417A (ja) | 2004-06-30 | 2011-10-14 | タンパク質キナーゼのインヒビターとして有用なアザインドール |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2007519460A Expired - Fee Related JP5122280B2 (ja) | 2004-06-30 | 2005-06-29 | タンパク質キナーゼのインヒビターとして有用なアザインドール |
Country Status (4)
Country | Link |
---|---|
JP (2) | JP5122280B2 (fr) |
IL (1) | IL180303A0 (fr) |
MX (1) | MX2007000092A (fr) |
NO (1) | NO20070502L (fr) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2007000092A (es) * | 2004-06-30 | 2007-03-07 | Vertex Pharma | Azaindoles utiles como inhibidores de proteinas cinasas. |
AR050917A1 (es) * | 2004-08-13 | 2006-12-06 | Amphora Discovery Corp | Compuestos basados en 2-amido-tiazol que presentan actividad inhibidora de enzimas que utilizan atp, y composiciones y usos de los mismos |
DE102008038221A1 (de) * | 2008-08-18 | 2010-02-25 | Merck Patent Gmbh | 7-Azaindolderivate |
DE102009058280A1 (de) * | 2009-12-14 | 2011-06-16 | Merck Patent Gmbh | Thiazolderivate |
AU2011239966B2 (en) * | 2010-04-16 | 2014-05-08 | Ac Immune S.A. | Novel compounds for the treatment of diseases associated with amyloid or amyloid-like proteins |
CA2803802A1 (fr) * | 2010-06-23 | 2011-12-29 | Vertex Pharmaceuticals Incorporated | Derives de pyrrolo-pyrazine utiles en tant qu'inhibiteurs de l'atr kinase |
DE102011105469A1 (de) * | 2011-06-24 | 2012-12-27 | Merck Patent Gmbh | 7-Azaindolderivate |
KR101742954B1 (ko) * | 2012-05-31 | 2017-06-02 | 페넥스 파마슈티컬스 아게 | 고아 핵 수용체 ror[감마]의 조절제로서의 카복사미드 또는 설폰아미드가 치환된 티아졸 및 관련된 유도체 |
BR112016017981B1 (pt) | 2014-02-04 | 2023-01-17 | Taiho Pharmaceutical Co., Ltd. | Compostos derivados de azaindola, inibidor de jak3, composição farmacêutica e agente compreendendo ditos compostos, e uso dos mesmos para tratar uma doença que envolve jak3 |
WO2023110843A1 (fr) * | 2021-12-15 | 2023-06-22 | Almirall, S.A. | Dérivés hétérobicycliques utilisés comme inhibiteurs de l'itk |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6265403B1 (en) * | 1999-01-20 | 2001-07-24 | Merck & Co., Inc. | Angiogenesis inhibitors |
ES2317889T3 (es) * | 2000-03-01 | 2009-05-01 | Janssen Pharmaceutica Nv | Derivados de tiazolilo 2,4-disustituido. |
SE0202463D0 (sv) * | 2002-08-14 | 2002-08-14 | Astrazeneca Ab | Novel compounds |
TW200604168A (en) * | 2004-04-02 | 2006-02-01 | Vertex Pharma | Azaindoles useful as inhibitors of rock and other protein kinases |
MX2007000092A (es) * | 2004-06-30 | 2007-03-07 | Vertex Pharma | Azaindoles utiles como inhibidores de proteinas cinasas. |
-
2005
- 2005-06-29 MX MX2007000092A patent/MX2007000092A/es active IP Right Grant
- 2005-06-29 JP JP2007519460A patent/JP5122280B2/ja not_active Expired - Fee Related
-
2006
- 2006-12-25 IL IL180303A patent/IL180303A0/en unknown
-
2007
- 2007-01-26 NO NO20070502A patent/NO20070502L/no not_active Application Discontinuation
-
2011
- 2011-10-14 JP JP2011227135A patent/JP2012012417A/ja active Pending
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