JP2012012417A5 - - Google Patents

Download PDF

Info

Publication number
JP2012012417A5
JP2012012417A5 JP2011227135A JP2011227135A JP2012012417A5 JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5 JP 2011227135 A JP2011227135 A JP 2011227135A JP 2011227135 A JP2011227135 A JP 2011227135A JP 2012012417 A5 JP2012012417 A5 JP 2012012417A5
Authority
JP
Japan
Prior art keywords
compound
independently
occurrence
optionally substituted
nrco
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011227135A
Other languages
English (en)
Japanese (ja)
Other versions
JP2012012417A (ja
Filing date
Publication date
Priority claimed from US11/098,751 external-priority patent/US7514448B2/en
Application filed filed Critical
Publication of JP2012012417A publication Critical patent/JP2012012417A/ja
Publication of JP2012012417A5 publication Critical patent/JP2012012417A5/ja
Pending legal-status Critical Current

Links

JP2011227135A 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール Pending JP2012012417A (ja)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US58438304P 2004-06-30 2004-06-30
US60/584,383 2004-06-30
US58472104P 2004-07-01 2004-07-01
US60/584,721 2004-07-01
US11/098,751 2005-04-04
US11/098,751 US7514448B2 (en) 2004-04-02 2005-04-04 Azaindoles useful as inhibitors of rock and other protein kinases
PCT/US2005/011358 WO2005103050A2 (fr) 2004-04-02 2005-04-04 Azaindoles utiles en tant qu'inhibiteurs de la proteine serine/threonine kinase superhelice de la famille rho (rock) et d'autres proteines kinases
USPCT/US05/11358 2005-04-04

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2007519460A Division JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013001760A Division JP2013064015A (ja) 2004-06-30 2013-01-09 タンパク質キナーゼのインヒビターとして有用なアザインドール

Publications (2)

Publication Number Publication Date
JP2012012417A JP2012012417A (ja) 2012-01-19
JP2012012417A5 true JP2012012417A5 (fr) 2013-02-28

Family

ID=37801682

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール
JP2011227135A Pending JP2012012417A (ja) 2004-06-30 2011-10-14 タンパク質キナーゼのインヒビターとして有用なアザインドール

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2007519460A Expired - Fee Related JP5122280B2 (ja) 2004-06-30 2005-06-29 タンパク質キナーゼのインヒビターとして有用なアザインドール

Country Status (4)

Country Link
JP (2) JP5122280B2 (fr)
IL (1) IL180303A0 (fr)
MX (1) MX2007000092A (fr)
NO (1) NO20070502L (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.
AR050917A1 (es) * 2004-08-13 2006-12-06 Amphora Discovery Corp Compuestos basados en 2-amido-tiazol que presentan actividad inhibidora de enzimas que utilizan atp, y composiciones y usos de los mismos
DE102008038221A1 (de) * 2008-08-18 2010-02-25 Merck Patent Gmbh 7-Azaindolderivate
DE102009058280A1 (de) * 2009-12-14 2011-06-16 Merck Patent Gmbh Thiazolderivate
AU2011239966B2 (en) * 2010-04-16 2014-05-08 Ac Immune S.A. Novel compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
CA2803802A1 (fr) * 2010-06-23 2011-12-29 Vertex Pharmaceuticals Incorporated Derives de pyrrolo-pyrazine utiles en tant qu'inhibiteurs de l'atr kinase
DE102011105469A1 (de) * 2011-06-24 2012-12-27 Merck Patent Gmbh 7-Azaindolderivate
KR101742954B1 (ko) * 2012-05-31 2017-06-02 페넥스 파마슈티컬스 아게 고아 핵 수용체 ror[감마]의 조절제로서의 카복사미드 또는 설폰아미드가 치환된 티아졸 및 관련된 유도체
BR112016017981B1 (pt) 2014-02-04 2023-01-17 Taiho Pharmaceutical Co., Ltd. Compostos derivados de azaindola, inibidor de jak3, composição farmacêutica e agente compreendendo ditos compostos, e uso dos mesmos para tratar uma doença que envolve jak3
WO2023110843A1 (fr) * 2021-12-15 2023-06-22 Almirall, S.A. Dérivés hétérobicycliques utilisés comme inhibiteurs de l'itk

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6265403B1 (en) * 1999-01-20 2001-07-24 Merck & Co., Inc. Angiogenesis inhibitors
ES2317889T3 (es) * 2000-03-01 2009-05-01 Janssen Pharmaceutica Nv Derivados de tiazolilo 2,4-disustituido.
SE0202463D0 (sv) * 2002-08-14 2002-08-14 Astrazeneca Ab Novel compounds
TW200604168A (en) * 2004-04-02 2006-02-01 Vertex Pharma Azaindoles useful as inhibitors of rock and other protein kinases
MX2007000092A (es) * 2004-06-30 2007-03-07 Vertex Pharma Azaindoles utiles como inhibidores de proteinas cinasas.

Similar Documents

Publication Publication Date Title
JP2012012417A5 (fr)
CY1118621T1 (el) Πολυμορφικες μορφες του 2-(5-βρωμο-4-(4-κυκλο προπυλναφθαλιν-1-υλ)-4η-1,2,4-τριαζολ-3-υλθειο) οξικου οξεος και χρησεις αυτων
MX2013006585A (es) Compuestos de anillo indeno fusionados.
CO6561783A2 (es) Inhibidores del virus flaviviridae
WO2012003405A4 (fr) Stimulateurs de sgc
MX2012009186A (es) Pirrolidina-2-carboxamidas sustituidas.
JP2013032389A5 (fr)
MX346746B (es) Compuestos de anillo indeno-fusionados.
JP2011137045A5 (fr)
MX2009009492A (es) Compuestos organicos biciclicos adecuados para el tratamiento de condiciones inflamatorias o alergicas.
MD4521C1 (ro) Compuşi antivirali pe bază de imidazolil-dihidroizocromeno-naftoimidazoli condensaţi
WO2012107706A8 (fr) Sels de diaminium de phénothiazine et leurs applications
EA201690019A1 (ru) Производное аминотриазина и содержащая его фармацевтическая композиция
JP2015537008A5 (fr)
JP2015522650A5 (fr)
AR084011A1 (es) Compuestos nitrogenados heterociclicos utiles para el tratamiento de infecciones por el virus sincitial respiratorio (rsv), proceso para prepararlos y composiciones farmaceuticas que los contienen
CY1117688T1 (el) Ενωσεις τετραϋδροπυρρολοθειαζινης
JP2013532130A5 (fr)
WO2012101011A3 (fr) Nouveaux dérivés d'arylbenzocycloalkylamides
JP2015535847A5 (fr)
EA201301315A1 (ru) Способ получения промежуточных соединений эстетрола
PE20150182A1 (es) Compuestos de fenoxietil piperidina
WO2013152277A3 (fr) Analogues de la moénomycine, procédés de synthèse, et leurs utilisations
EA201391537A1 (ru) ЭТИНИЛЬНЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ ПОЛОЖИТЕЛЬНЫХ АЛЛОСТЕРИЧЕСКИХ МОДУЛЯТОРОВ mGluR5
JP2011190277A5 (fr)