|
US3444216A
(en)
|
1966-11-16 |
1969-05-13 |
Upjohn Co |
Process for the oxidation of primary and secondary alcohols
|
|
NZ207394A
(en)
|
1983-03-08 |
1987-03-06 |
Commw Serum Lab Commission |
Detecting or determining sequence of amino acids
|
|
US5128448A
(en)
|
1990-01-10 |
1992-07-07 |
Hoffman-La Roche Inc. |
CCK analogs with appetite regulating activity
|
|
US5374623A
(en)
|
1992-08-20 |
1994-12-20 |
Prototek, Inc. |
Cysteine protease inhibitors effective for in vivo use
|
|
CA2111930A1
(en)
|
1992-12-25 |
1994-06-26 |
Ryoichi Ando |
Aminoketone derivatives
|
|
DZ2285A1
(fr)
|
1996-08-08 |
2002-12-25 |
Smithkline Beecham Corp |
Inhibiteurs de protéase de la cystéine.
|
|
US6043218A
(en)
|
1996-10-22 |
2000-03-28 |
Medical University Of South Carolina |
Positively charged non-natural amino acids, methods of making thereof, and use thereof in peptides
|
|
AR013079A1
(es)
|
1997-05-06 |
2000-12-13 |
Smithkline Beecham Corp |
Derivados sustituidos de tetrahidrofurano-3-onas, de tetrahidropirano-3- onas y tetrahidrotiofen-3-onas, un procedimiento para su preparacion unacomposicion farmaceutica de un medicamento util como inhibidores de proteasas e intermediarios
|
|
HUP0004400A3
(en)
|
1997-11-05 |
2002-10-28 |
Novartis Ag |
Dipeptide nitriles, process for their preparation, pharmaceutical compositions comprising thereof and their use
|
|
GB9806287D0
(en)
|
1998-03-24 |
1998-05-20 |
Synphar Lab Inc |
Monobactam enzyme inhibitors
|
|
MA26618A1
(fr)
|
1998-04-09 |
2004-12-20 |
Smithkline Beecham Corp |
Composes et compositions pharmaceutiques pour le traitement du paludisme
|
|
DZ2815A1
(fr)
|
1998-06-12 |
2003-12-01 |
Smithkline Beecham Corp |
Inhibiteurs de protéase.
|
|
CA2301201A1
(en)
|
1998-08-14 |
2000-02-24 |
Smithkline Beecham Corporation |
Method of inhibiting cathepsin k
|
|
ES2142773B1
(es)
|
1998-10-07 |
2001-01-01 |
Lacer Sa |
Derivados de mononitrato de isosorbida y su empleo como agentes vasodilatadores con tolerancia desminuida.
|
|
CO5150165A1
(es)
|
1998-11-13 |
2002-04-29 |
Smithkline Beecham Plc |
Inhibidores de proteasa: tipo catepsina k
|
|
GB9903861D0
(en)
|
1999-02-20 |
1999-04-14 |
Zeneca Ltd |
Chemical compounds
|
|
AU2560300A
(en)
|
1999-02-20 |
2000-09-04 |
Astrazeneca Ab |
Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsins
|
|
JP2002537294A
(ja)
|
1999-02-20 |
2002-11-05 |
アストラゼネカ アクチボラグ |
カテプシンl及びカテプシンsの阻害剤としてのジ−及びトリペプチドニトリル誘導体
|
|
CA2360740A1
(en)
|
1999-03-02 |
2000-09-08 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Compounds useful as reversible inhibitors of cathepsin s
|
|
HK1039110A1
(zh)
|
1999-03-15 |
2002-04-12 |
Axys Pharmaceuticals, Inc. |
以新颖的合成物及组分作为蛋白酶抑制剂
|
|
TW200404789A
(en)
|
1999-03-15 |
2004-04-01 |
Axys Pharm Inc |
Novel compounds and compositions as protease inhibitors
|
|
EA200100972A1
(ru)
|
1999-03-15 |
2002-02-28 |
Аксис Фармасьютикалз, Инк. |
Новые соединения и композиции как ингибиторы протеаз
|
|
GB9907683D0
(en)
|
1999-04-06 |
1999-05-26 |
Synphar Lab Inc |
Substituted azetidin-2-ones as cysteine protease inhibitors
|
|
GB9911417D0
(en)
|
1999-05-18 |
1999-07-14 |
Peptide Therapeutics Ltd |
Furanone derivatives as inhibitors of cathepsin s
|
|
GB9917909D0
(en)
|
1999-07-31 |
1999-09-29 |
Synphar Lab Inc |
Cysteine protease inhibitors
|
|
DE50003927D1
(de)
|
1999-08-03 |
2003-11-06 |
Siemens Ag |
Ausschaltverzögerungsschaltung für ein elektromechanisches schaltgerät
|
|
US6420364B1
(en)
|
1999-09-13 |
2002-07-16 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Compound useful as reversible inhibitors of cysteine proteases
|
|
HUP0302380A2
(hu)
|
1999-09-13 |
2004-03-01 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Cisztein-proteázok reverzibilis inhibitoraiként alkalmazható új spiroheterociklusos vegyületek, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények
|
|
WO2001019808A1
(en)
|
1999-09-16 |
2001-03-22 |
Axys Pharmaceuticals, Inc. |
Chemical compounds and compositions and their use as cathepsin s inhibitors
|
|
GB9925264D0
(en)
|
1999-10-26 |
1999-12-29 |
Zeneca Ltd |
Chemical compounds
|
|
JP2003513928A
(ja)
|
1999-11-10 |
2003-04-15 |
スミスクライン・ビーチャム・コーポレイション |
プロテアーゼ阻害剤
|
|
WO2001034153A1
(en)
|
1999-11-10 |
2001-05-17 |
Smithkline Beecham Corporation |
Protease inhibitors
|
|
ATE339404T1
(de)
|
1999-12-24 |
2006-10-15 |
Hoffmann La Roche |
Nitrilderivate als cathepsin k hemmer
|
|
DE60132975T2
(de)
|
2000-01-06 |
2009-02-26 |
Merck Frosst Canada Inc., Kirkland |
Neue substanzen und verbindungen als protease-inhibitoren
|
|
GB0003111D0
(en)
|
2000-02-10 |
2000-03-29 |
Novartis Ag |
Organic compounds
|
|
WO2001068645A2
(en)
|
2000-03-15 |
2001-09-20 |
Axys Pharmaceuticals, Inc. |
N-cyanomethylcarboxamides and their use as protease inhibitors
|
|
OA12323A
(en)
|
2000-03-21 |
2006-05-15 |
Smithkline Beecham Corp |
Protease inhibitors.
|
|
JP2003530384A
(ja)
|
2000-04-06 |
2003-10-14 |
メルク フロスト カナダ アンド カンパニー |
カテプシンシステインプロテアーゼ阻害薬
|
|
CO5280093A1
(es)
|
2000-04-18 |
2003-05-30 |
Smithkline Beecham Corp |
Metodos de tratamiento
|
|
HUP0301231A2
(hu)
|
2000-06-14 |
2003-08-28 |
Smithkline Beecham Corp. |
Proteáz inhibitorok, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk
|
|
US6462076B2
(en)
|
2000-06-14 |
2002-10-08 |
Hoffmann-La Roche Inc. |
Beta-amino acid nitrile derivatives as cathepsin K inhibitors
|
|
WO2002017924A1
(en)
|
2000-09-01 |
2002-03-07 |
Smithkline Beecham Corporation |
Method of treatment
|
|
WO2002032879A1
(en)
|
2000-10-19 |
2002-04-25 |
Naeja Pharmaceutical Inc. |
Dihydropyrimidine derivatives as cysteine protease inhibitors
|
|
WO2002051983A2
(en)
|
2000-12-22 |
2002-07-04 |
Axys Pharmaceuticals, Inc. |
Novel compounds and compositions as cathepsin inhibitors
|
|
CA2434068A1
(en)
|
2001-01-17 |
2002-07-25 |
Amura Therapeutics Limited |
Inhibitors of cruzipain and other cysteine proteases
|
|
PT1362052E
(pt)
*
|
2001-01-17 |
2007-04-30 |
Amura Therapeutics Ltd |
Inibidores de cruzipaína e de outras proteases de cisteína
|
|
WO2002080920A1
(en)
|
2001-04-06 |
2002-10-17 |
Axys Pharmaceuticals, Inc. |
Arylacetamido-ketobenzoxazole as cysteine protease inhibitors
|
|
EP1401453A4
(en)
|
2001-05-17 |
2005-04-06 |
Smithkline Beecham Corp |
PROTEASE INHIBITORS
|
|
FR2826572B1
(fr)
|
2001-06-29 |
2005-10-07 |
Oreal |
Compositions contenant un derive d'hydroxydiphenyl ether inhibant le developpement des odeurs corporelles
|
|
WO2003013518A1
(en)
|
2001-08-03 |
2003-02-20 |
Smithkline Beecham Corporation |
Alpha-ketoamide derivatives as cathepsin k inhibitors
|
|
AR036375A1
(es)
|
2001-08-30 |
2004-09-01 |
Novartis Ag |
Compuestos pirrolo [2,3-d] pirimidina -2- carbonitrilo, un proceso para su preparacion, una composicion farmaceutica y el uso de dichos compuestos para la preparacion de medicamentos
|
|
MXPA04002282A
(es)
|
2001-09-14 |
2005-03-07 |
Axis Pharmaceutical Inc |
Nuevos compuestos y preparaciones como inhibidores de la catepsina.
|
|
EP1434769A2
(en)
|
2001-10-02 |
2004-07-07 |
Boehringer Ingelheim Pharmaceuticals Inc. |
Compounds useful as reversible inhibitors of cysteine proteases
|
|
CA2463770A1
(en)
|
2001-10-29 |
2003-05-08 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Compounds useful as reversible inhibitors of cysteine proteases
|
|
DE60225316T2
(de)
|
2001-11-13 |
2009-02-26 |
AXYS Pharmaceuticals, Inc., South San Francisco |
Cyanoalkylamino-derivate als protease-hemmer
|
|
EP1446392A1
(en)
|
2001-11-14 |
2004-08-18 |
Aventis Pharmaceuticals, Inc. |
Oligopeptides and compositions containing them as cathepsin s inhibitors
|
|
CN100354276C
(zh)
|
2002-07-16 |
2007-12-12 |
阿姆拉医疗有限公司 |
生物活性化合物
|
|
DE602005019971D1
(de)
|
2004-01-08 |
2010-04-29 |
Medivir Ab |
Inhibitoren von cysteinprotease
|
|
WO2006064286A1
(en)
|
2004-12-13 |
2006-06-22 |
Medivir Uk Ltd |
Cathepsin s inhibitors
|
|
GB0614044D0
(en)
*
|
2006-07-14 |
2006-08-23 |
Amura Therapeutics Ltd |
Compounds
|
|
GB0614042D0
(en)
*
|
2006-07-14 |
2006-08-23 |
Amura Therapeutics Ltd |
Compounds
|