JP2010537988A - 紅斑を治療するための改良ブリモニジン組成物 - Google Patents
紅斑を治療するための改良ブリモニジン組成物 Download PDFInfo
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- JP2010537988A JP2010537988A JP2010522973A JP2010522973A JP2010537988A JP 2010537988 A JP2010537988 A JP 2010537988A JP 2010522973 A JP2010522973 A JP 2010522973A JP 2010522973 A JP2010522973 A JP 2010522973A JP 2010537988 A JP2010537988 A JP 2010537988A
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
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- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US96719107P | 2007-08-31 | 2007-08-31 | |
| PCT/US2008/010290 WO2009032223A1 (en) | 2007-08-31 | 2008-08-29 | Improved brimonidine compositions for treating erythema |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010537988A true JP2010537988A (ja) | 2010-12-09 |
| JP2010537988A5 JP2010537988A5 (enExample) | 2011-10-13 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2010522973A Abandoned JP2010537988A (ja) | 2007-08-31 | 2008-08-29 | 紅斑を治療するための改良ブリモニジン組成物 |
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| US (3) | US20090061020A1 (enExample) |
| EP (1) | EP2200617A4 (enExample) |
| JP (1) | JP2010537988A (enExample) |
| KR (1) | KR20100055453A (enExample) |
| CN (2) | CN101808645A (enExample) |
| AR (1) | AR068816A1 (enExample) |
| AU (1) | AU2008296948A1 (enExample) |
| BR (1) | BRPI0816097A2 (enExample) |
| CA (1) | CA2698680A1 (enExample) |
| MX (1) | MX2010002392A (enExample) |
| NO (1) | NO20100301L (enExample) |
| WO (1) | WO2009032223A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014533271A (ja) * | 2011-11-10 | 2014-12-11 | アラーガン インコーポレイテッドAllergan,Incorporated | 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物 |
| US10201535B2 (en) | 2011-11-10 | 2019-02-12 | Allergan, Inc. | Pharmaceutical compositions comprising 7-(1H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7439241B2 (en) * | 2003-05-27 | 2008-10-21 | Galderma Laboratories, Inc. | Compounds, formulations, and methods for treating or preventing rosacea |
| US8410102B2 (en) | 2003-05-27 | 2013-04-02 | Galderma Laboratories Inc. | Methods and compositions for treating or preventing erythema |
| US7812049B2 (en) | 2004-01-22 | 2010-10-12 | Vicept Therapeutics, Inc. | Method and therapeutic/cosmetic topical compositions for the treatment of rosacea and skin erythema using α1-adrenoceptor agonists |
| WO2010136594A2 (en) * | 2009-05-29 | 2010-12-02 | Symatese | Injectable combination of adrenergic receptor agonists with fillers, for decreasing skin reactions due to injection |
| EP2493309A4 (en) * | 2009-10-26 | 2013-05-01 | Galderma Pharma Sa | METHODS OF TREATING OR PREVENTING ACUTE ERYTHEMA |
| EP2329849B1 (en) * | 2009-11-18 | 2015-04-29 | Galderma Research & Development | Combination of alpha-2 adrenergic receptor agonist and non-steroidal anti-inflammatory agent for treating or preventing an inflammatory skin disorder |
| US8394800B2 (en) * | 2009-11-19 | 2013-03-12 | Galderma Laboratories, L.P. | Method for treating psoriasis |
| RU2535008C2 (ru) | 2010-03-26 | 2014-12-10 | Галдерма Ресерч Энд Девелопмент | Улучшенные способы и композиции для безопасного и эффективного лечения телеангиэктазии |
| MX2012010824A (es) * | 2010-03-26 | 2012-10-10 | Galderma Res & Dev | Metodos y composiciones mejoradas para tratamiento seguro y efectivo del eritema. |
| SG189896A1 (en) | 2010-10-21 | 2013-06-28 | Galderma Sa | Brimonidine gel compositions and methods of use |
| FR2966366B1 (fr) * | 2010-10-21 | 2012-11-09 | Galderma Sa | Composition de gel de brimonidine |
| US8053427B1 (en) | 2010-10-21 | 2011-11-08 | Galderma R&D SNC | Brimonidine gel composition |
| FR2966365B1 (fr) * | 2010-10-21 | 2012-11-09 | Galderma Sa | Composition de gel topique |
| CA2814975A1 (en) * | 2010-10-21 | 2012-04-26 | Galderma S.A. | Topical gel composition |
| AU2012217858A1 (en) | 2011-02-15 | 2013-09-05 | Allergan, Inc. | Pharmaceutical cream compositions of oxymetazoline for treating symptoms of rosacea |
| BR112014009210A2 (pt) | 2011-10-19 | 2017-04-18 | Galderma Sa | método para a redução da vermelhidão facial cutânea |
| FR3000397A1 (fr) | 2012-12-31 | 2014-07-04 | Galderma Res & Dev | Combinaison de laropiprant et d'ivermectine pour le traitement de la rosacee |
| FR3000398A1 (fr) * | 2012-12-31 | 2014-07-04 | Galderma Res & Dev | Combinaison de laropiprant et de brimonidine pour le traitement de la rosacee |
| FR3015288B1 (fr) | 2013-12-19 | 2016-02-12 | Galderma Res & Dev | Utilsation du naratriptan dans le traitement de la rosacee |
| WO2015191917A1 (en) | 2014-06-11 | 2015-12-17 | Allergan, Inc. | Stabilized oxymetazoline formulations and their uses |
| WO2019014518A1 (en) * | 2017-07-14 | 2019-01-17 | Galderma Research And Development | METHODS AND COMPOSITIONS FOR REDUCING ADVERSE EFFECTS OF CHEMOTHERAPEUTIC TREATMENTS |
| BR112021020962A2 (pt) | 2019-05-01 | 2021-12-14 | Clexio Biosciences Ltd | Métodos de tratamento de prurido |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4285967A (en) * | 1978-06-30 | 1981-08-25 | Estee Lauder Inc. | Cosmetic preparation for reducing redness of blemishes |
| US4256763A (en) * | 1978-09-19 | 1981-03-17 | Mchugh John E | Treatment of herpes simplex infections and acne |
| GB8827968D0 (en) * | 1988-11-30 | 1989-01-05 | Boots Co Plc | Sunscreen compositions |
| US5916574A (en) * | 1996-10-09 | 1999-06-29 | Ideal Ideas, Inc. | Method of treating natural poison skin conditions |
| US6410045B1 (en) * | 1999-02-22 | 2002-06-25 | Clyde Lewis Schultz | Drug delivery system for antiglaucomatous medication |
| US6294553B1 (en) * | 2000-02-15 | 2001-09-25 | Allergan Sales, Inc. | Method for treating ocular pain |
| US20040266776A1 (en) * | 2003-06-25 | 2004-12-30 | Gil Daniel W. | Methods of preventing and reducing the severity of stress-associated conditions |
| US7439241B2 (en) * | 2003-05-27 | 2008-10-21 | Galderma Laboratories, Inc. | Compounds, formulations, and methods for treating or preventing rosacea |
| US20050020600A1 (en) * | 2003-07-23 | 2005-01-27 | Scherer Warren J. | Methods of treating cutaneous flushing using selective alpha-2-adrenergic receptor agonists |
| US20050276765A1 (en) * | 2004-06-10 | 2005-12-15 | Paul Nghiem | Preventing skin damage |
| EP2230910A4 (en) * | 2007-12-21 | 2011-04-13 | Galderma Lab Inc | PRE-SURGICAL TREATMENT |
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2008
- 2008-08-18 US US12/193,098 patent/US20090061020A1/en not_active Abandoned
- 2008-08-29 WO PCT/US2008/010290 patent/WO2009032223A1/en not_active Ceased
- 2008-08-29 KR KR1020107005023A patent/KR20100055453A/ko not_active Ceased
- 2008-08-29 CN CN200880105032A patent/CN101808645A/zh active Pending
- 2008-08-29 MX MX2010002392A patent/MX2010002392A/es not_active Application Discontinuation
- 2008-08-29 CN CN201110321688XA patent/CN102552112A/zh active Pending
- 2008-08-29 EP EP08795728A patent/EP2200617A4/en not_active Withdrawn
- 2008-08-29 JP JP2010522973A patent/JP2010537988A/ja not_active Abandoned
- 2008-08-29 BR BRPI0816097A patent/BRPI0816097A2/pt not_active IP Right Cessation
- 2008-08-29 AU AU2008296948A patent/AU2008296948A1/en not_active Abandoned
- 2008-08-29 CA CA2698680A patent/CA2698680A1/en not_active Abandoned
- 2008-09-01 AR ARP080103804A patent/AR068816A1/es not_active Application Discontinuation
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2010
- 2010-03-04 NO NO20100301A patent/NO20100301L/no not_active Application Discontinuation
-
2011
- 2011-10-21 US US13/278,955 patent/US20120040016A1/en not_active Abandoned
-
2012
- 2012-07-12 US US13/547,531 patent/US20120282346A1/en not_active Abandoned
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014533271A (ja) * | 2011-11-10 | 2014-12-11 | アラーガン インコーポレイテッドAllergan,Incorporated | 7−(1h−イミダゾール−4−イルメチル)−5,6,7,8−テトラヒドロキノリンを含む肌の疾患および状態を治療するための医薬組成物 |
| US10201535B2 (en) | 2011-11-10 | 2019-02-12 | Allergan, Inc. | Pharmaceutical compositions comprising 7-(1H-imidazol-4-ylmethyl)-5,6,7,8-tetrahydro-quinoline for treating skin diseases and conditions |
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0816097A2 (pt) | 2016-11-01 |
| AU2008296948A1 (en) | 2009-03-12 |
| US20120040016A1 (en) | 2012-02-16 |
| CN102552112A (zh) | 2012-07-11 |
| AR068816A1 (es) | 2009-12-09 |
| CN101808645A (zh) | 2010-08-18 |
| KR20100055453A (ko) | 2010-05-26 |
| US20120282346A1 (en) | 2012-11-08 |
| EP2200617A1 (en) | 2010-06-30 |
| NO20100301L (no) | 2010-03-25 |
| WO2009032223A1 (en) | 2009-03-12 |
| MX2010002392A (es) | 2010-07-28 |
| EP2200617A4 (en) | 2011-01-12 |
| US20090061020A1 (en) | 2009-03-05 |
| CA2698680A1 (en) | 2009-03-12 |
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