JP2010535738A5 - - Google Patents

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Publication number
JP2010535738A5
JP2010535738A5 JP2010519457A JP2010519457A JP2010535738A5 JP 2010535738 A5 JP2010535738 A5 JP 2010535738A5 JP 2010519457 A JP2010519457 A JP 2010519457A JP 2010519457 A JP2010519457 A JP 2010519457A JP 2010535738 A5 JP2010535738 A5 JP 2010535738A5
Authority
JP
Japan
Prior art keywords
phenyl
triazol
ylamine
trifluoromethyl
methoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2010519457A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010535738A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2008/060307 external-priority patent/WO2009019278A1/en
Publication of JP2010535738A publication Critical patent/JP2010535738A/ja
Publication of JP2010535738A5 publication Critical patent/JP2010535738A5/ja
Abandoned legal-status Critical Current

Links

JP2010519457A 2007-08-08 2008-08-06 ニコチン性アセチルコリン受容体の調節物質として有用な新規1,2,3−トリアゾール誘導体 Abandoned JP2010535738A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200701134 2007-08-08
US95508107P 2007-08-10 2007-08-10
PCT/EP2008/060307 WO2009019278A1 (en) 2007-08-08 2008-08-06 Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors

Publications (2)

Publication Number Publication Date
JP2010535738A JP2010535738A (ja) 2010-11-25
JP2010535738A5 true JP2010535738A5 (enExample) 2011-09-15

Family

ID=39870242

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010519457A Abandoned JP2010535738A (ja) 2007-08-08 2008-08-06 ニコチン性アセチルコリン受容体の調節物質として有用な新規1,2,3−トリアゾール誘導体

Country Status (12)

Country Link
US (1) US8110588B2 (enExample)
EP (1) EP2185529A1 (enExample)
JP (1) JP2010535738A (enExample)
KR (1) KR20100046179A (enExample)
CN (1) CN101796034A (enExample)
AU (1) AU2008285644A1 (enExample)
CA (1) CA2695812A1 (enExample)
MX (1) MX2010001135A (enExample)
NZ (1) NZ582520A (enExample)
RU (1) RU2010102994A (enExample)
WO (1) WO2009019278A1 (enExample)
ZA (1) ZA201000127B (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009112459A1 (en) * 2008-03-11 2009-09-17 Neurosearch A/S Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
US20110201656A1 (en) * 2008-08-08 2011-08-18 Neurosearch A/S Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
BRPI0917693A2 (pt) * 2008-09-02 2016-05-17 Neurosearch As composto derivado de triazol, composição farmacêutica, e, uso de um derivado de triazol
AR078538A1 (es) 2009-10-07 2011-11-16 Karobio Ab Pirroles e imidazoles sustituidos como ligandos del receptor de estrogenos
CA2825519A1 (en) 2011-02-03 2012-09-08 Lupin Limited Pyrrole derivatives used as modulators of alpha7 nachr
RS55433B1 (sr) 2011-02-23 2017-04-28 Lupin Ltd Derivati heteroarila kao modulatori nachr alfa7
AU2012235779B2 (en) 2011-03-31 2017-03-02 Lupin Limited Pyrrole derivatives as nicotinic acetylcholine receptor modulators for use in the treatment of neurodegenerative disorders such as Alzheimer's and Parkinson's disease
FR2974365B1 (fr) * 2011-04-20 2017-08-25 Centre Nat De La Rech Scient (C N R S) 1,2,3-triazoles 1,4-disubstituees, leurs procedes de preparation et leurs utilisations diagnostiques et therapeutiques
US8946432B2 (en) 2011-07-05 2015-02-03 Lupin Limited Biaryl derivatives as nAChR modulators
GB201113538D0 (en) 2011-08-04 2011-09-21 Karobio Ab Novel estrogen receptor ligands
NZ629453A (en) 2012-03-06 2016-04-29 Lupin Ltd Thiazole derivatives as alpha 7 nachr modulators
EP2945936A1 (en) 2012-11-12 2015-11-25 Lupin Limited Thiazole derivatives as alpha 7 nachr modulators
EP2945941B1 (en) 2013-01-16 2016-12-07 Lupin Limited Pyrrole derivatives as alpha 7 nachr modulators
US9617210B2 (en) 2013-03-13 2017-04-11 Lupin Limited Pyrrole derivatives as alpha 7 NACHR modulators
TW201446243A (zh) 2013-06-03 2014-12-16 Lupin Ltd 4-(5-(4-氯苯基)-2-(2-環丙基乙醯基)-1,4-二甲基-1氫-吡咯-3-基)苯磺醯胺作為α7尼古丁乙醯膽鹼受體調節劑
WO2014203150A1 (en) 2013-06-17 2014-12-24 Lupin Limited Pyrrole derivatives as alpha 7 nachr modulators
WO2019124577A1 (ko) 2017-12-20 2019-06-27 재단법인 경기도경제과학진흥원 트리아졸 유도체 및 이의 용도
CN113045507B (zh) * 2021-03-04 2022-10-25 中山大学南方学院 一种3,4-二羟基苯甲酸甲酯衍生物及其制备方法与应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1242216B (de) * 1963-12-27 1967-06-15 Union Carbide Corp Verfahren zur Herstellung von Inaminsalzen
EP1458708B1 (en) * 2001-12-18 2007-09-26 Merck & Co., Inc. Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5
DK1501809T3 (da) * 2002-04-26 2008-05-13 Lilly Co Eli Trizolderivater som tachykininreceptorantagonister
UA85711C2 (ru) 2004-05-06 2009-02-25 Зе Регентс Оф Зе Юниверсити Оф Калифорния Замещенные енаминоны, их производные и их применение
EP1833804A1 (en) 2004-12-28 2007-09-19 AstraZeneca AB Aryl sulphonamide modulators
WO2009112459A1 (en) 2008-03-11 2009-09-17 Neurosearch A/S Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
US20110201656A1 (en) 2008-08-08 2011-08-18 Neurosearch A/S Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors

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