CN101796034A - 用作烟碱型乙酰胆碱受体的调节剂的新颖的1,2,3-三唑衍生物 - Google Patents

用作烟碱型乙酰胆碱受体的调节剂的新颖的1,2,3-三唑衍生物 Download PDF

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Publication number
CN101796034A
CN101796034A CN200880102108A CN200880102108A CN101796034A CN 101796034 A CN101796034 A CN 101796034A CN 200880102108 A CN200880102108 A CN 200880102108A CN 200880102108 A CN200880102108 A CN 200880102108A CN 101796034 A CN101796034 A CN 101796034A
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phenyl
triazol
trifluoromethyl
ylamine
methoxy
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Chinese (zh)
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A·纳蒂
J·K·克里斯坦森
D·彼德斯
G·M·奥尔森
T·戴赫林
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NTG Nordic Transport Group AS
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Neurosearch AS
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    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
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CN200880102108A 2007-08-08 2008-08-06 用作烟碱型乙酰胆碱受体的调节剂的新颖的1,2,3-三唑衍生物 Pending CN101796034A (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DKPA200701134 2007-08-08
DKPA200701134 2007-08-08
US95508107P 2007-08-10 2007-08-10
US60/955,081 2007-08-10
PCT/EP2008/060307 WO2009019278A1 (en) 2007-08-08 2008-08-06 Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors

Publications (1)

Publication Number Publication Date
CN101796034A true CN101796034A (zh) 2010-08-04

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CN200880102108A Pending CN101796034A (zh) 2007-08-08 2008-08-06 用作烟碱型乙酰胆碱受体的调节剂的新颖的1,2,3-三唑衍生物

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US (1) US8110588B2 (enExample)
EP (1) EP2185529A1 (enExample)
JP (1) JP2010535738A (enExample)
KR (1) KR20100046179A (enExample)
CN (1) CN101796034A (enExample)
AU (1) AU2008285644A1 (enExample)
CA (1) CA2695812A1 (enExample)
MX (1) MX2010001135A (enExample)
NZ (1) NZ582520A (enExample)
RU (1) RU2010102994A (enExample)
WO (1) WO2009019278A1 (enExample)
ZA (1) ZA201000127B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113045507A (zh) * 2021-03-04 2021-06-29 中山大学南方学院 一种3,4-二羟基苯甲酸甲酯衍生物及其制备方法与应用

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US20110060017A1 (en) * 2008-03-11 2011-03-10 Neurosearch A/S Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
AU2009279172A1 (en) * 2008-08-08 2010-02-11 Neurosearch A/S Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
EP2324007B1 (en) * 2008-09-02 2012-08-15 NeuroSearch A/S Triazole derivatives and their use as nicotinic acetylcholine receptor modulators
US8653112B2 (en) 2009-10-07 2014-02-18 Karo Bio Ab Substituted pyrazoles as estrogen receptor ligands
SG192078A1 (en) 2011-02-03 2013-08-30 Lupin Ltd Pyrrole derivatives used as modulators of alpha7 nachr
AP3649A (en) 2011-02-23 2016-03-18 Lupin Ltd Heteroaryl derivatives as alpha7 nachr modulators
BR112013025128A2 (pt) 2011-03-31 2017-02-14 Lupin Ltd derivados de pirrol como moduladores de receptor de acetilcolina nicotínico para uso no tratamento de distúrbios neurodegenenerativos tal como doença de alzheimer e doença de parkinson
FR2974365B1 (fr) * 2011-04-20 2017-08-25 Centre Nat De La Rech Scient (C N R S) 1,2,3-triazoles 1,4-disubstituees, leurs procedes de preparation et leurs utilisations diagnostiques et therapeutiques
US8946432B2 (en) 2011-07-05 2015-02-03 Lupin Limited Biaryl derivatives as nAChR modulators
GB201113538D0 (en) 2011-08-04 2011-09-21 Karobio Ab Novel estrogen receptor ligands
US9388196B2 (en) 2012-03-06 2016-07-12 Lupin Limited Thiazole derivatives as alpha 7 nAChR modulators
EP2945936A1 (en) 2012-11-12 2015-11-25 Lupin Limited Thiazole derivatives as alpha 7 nachr modulators
US9617211B2 (en) 2013-01-16 2017-04-11 Lupin Limited Pyrrole derivatives as alpha 7 nAChR modulators
WO2014141091A1 (en) 2013-03-13 2014-09-18 Lupin Limited Pyrrole derivatives as alpha 7 nachr modulators
TW201446243A (zh) 2013-06-03 2014-12-16 Lupin Ltd 4-(5-(4-氯苯基)-2-(2-環丙基乙醯基)-1,4-二甲基-1氫-吡咯-3-基)苯磺醯胺作為α7尼古丁乙醯膽鹼受體調節劑
CA2913987A1 (en) 2013-06-17 2014-12-24 Lupin Limited Pyrrole derivatives as alpha 7 nachr modulators
US20210163425A1 (en) 2017-12-20 2021-06-03 Gyeonggido Business & Science Accelerator Triazole derivative and use thereof

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DE1242216B (de) 1963-12-27 1967-06-15 Union Carbide Corp Verfahren zur Herstellung von Inaminsalzen
CA2469821C (en) 2001-12-18 2009-10-20 Merck & Co., Inc. Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5
JP4559087B2 (ja) * 2002-04-26 2010-10-06 イーライ リリー アンド カンパニー タキキニン受容体アンタゴニストとしてのトリアゾール誘導体
WO2005108347A2 (en) 2004-05-06 2005-11-17 The Regents Of The University Of California Substituted enaminones, their derivatives and uses thereof
CN101090895A (zh) 2004-12-28 2007-12-19 阿斯利康(瑞典)有限公司 芳基磺酰胺调节剂
US20110060017A1 (en) 2008-03-11 2011-03-10 Neurosearch A/S Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors
AU2009279172A1 (en) 2008-08-08 2010-02-11 Neurosearch A/S Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113045507A (zh) * 2021-03-04 2021-06-29 中山大学南方学院 一种3,4-二羟基苯甲酸甲酯衍生物及其制备方法与应用

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US8110588B2 (en) 2012-02-07
EP2185529A1 (en) 2010-05-19
CA2695812A1 (en) 2009-02-12
MX2010001135A (es) 2010-03-09
WO2009019278A1 (en) 2009-02-12
JP2010535738A (ja) 2010-11-25
AU2008285644A1 (en) 2009-02-12
US20100222398A1 (en) 2010-09-02
RU2010102994A (ru) 2011-09-20
KR20100046179A (ko) 2010-05-06
ZA201000127B (en) 2011-03-30

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