JP2010531293A5 - - Google Patents

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Publication number
JP2010531293A5
JP2010531293A5 JP2009553349A JP2009553349A JP2010531293A5 JP 2010531293 A5 JP2010531293 A5 JP 2010531293A5 JP 2009553349 A JP2009553349 A JP 2009553349A JP 2009553349 A JP2009553349 A JP 2009553349A JP 2010531293 A5 JP2010531293 A5 JP 2010531293A5
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JP
Japan
Prior art keywords
group
glycyl
phenylalanyl
salt
general formula
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Application number
JP2009553349A
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English (en)
Japanese (ja)
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JP5653043B2 (ja
JP2010531293A (ja
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Priority to JP2009553349A priority Critical patent/JP5653043B2/ja
Priority claimed from JP2009553349A external-priority patent/JP5653043B2/ja
Publication of JP2010531293A publication Critical patent/JP2010531293A/ja
Publication of JP2010531293A5 publication Critical patent/JP2010531293A5/ja
Application granted granted Critical
Publication of JP5653043B2 publication Critical patent/JP5653043B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009553349A 2007-06-26 2008-06-26 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体 Expired - Fee Related JP5653043B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2009553349A JP5653043B2 (ja) 2007-06-26 2008-06-26 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2007167207 2007-06-26
JP2007167207 2007-06-26
JP2009553349A JP5653043B2 (ja) 2007-06-26 2008-06-26 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体
PCT/JP2008/062033 WO2009001968A1 (en) 2007-06-26 2008-06-26 Benzazepine derivatives useful as vasopressin antagonists

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2014130326A Division JP5689195B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体
JP2014130327A Division JP5893085B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体

Publications (3)

Publication Number Publication Date
JP2010531293A JP2010531293A (ja) 2010-09-24
JP2010531293A5 true JP2010531293A5 (OSRAM) 2013-02-07
JP5653043B2 JP5653043B2 (ja) 2015-01-14

Family

ID=39773045

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2009553349A Expired - Fee Related JP5653043B2 (ja) 2007-06-26 2008-06-26 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体
JP2014130326A Expired - Fee Related JP5689195B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体
JP2014130327A Expired - Fee Related JP5893085B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014130326A Expired - Fee Related JP5689195B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体
JP2014130327A Expired - Fee Related JP5893085B2 (ja) 2007-06-26 2014-06-25 バソプレシン拮抗剤として使用されるベンゾアゼピン誘導体

Country Status (27)

Country Link
US (3) US8669229B2 (OSRAM)
EP (3) EP2374798B1 (OSRAM)
JP (3) JP5653043B2 (OSRAM)
KR (1) KR101487201B1 (OSRAM)
CN (3) CN103342680A (OSRAM)
AR (1) AR067176A1 (OSRAM)
AT (1) ATE545633T1 (OSRAM)
AU (1) AU2008269918B2 (OSRAM)
BR (1) BRPI0813768A2 (OSRAM)
CA (1) CA2690335A1 (OSRAM)
CO (1) CO6160295A2 (OSRAM)
CY (3) CY1113519T1 (OSRAM)
DK (3) DK2374798T3 (OSRAM)
ES (3) ES2431515T3 (OSRAM)
HR (3) HRP20120310T1 (OSRAM)
IL (1) IL202561A0 (OSRAM)
MY (3) MY152805A (OSRAM)
NZ (3) NZ581723A (OSRAM)
PH (2) PH12012501362A1 (OSRAM)
PL (3) PL2170831T3 (OSRAM)
PT (3) PT2374798E (OSRAM)
RU (1) RU2471784C2 (OSRAM)
SG (2) SG182231A1 (OSRAM)
SI (3) SI2374797T1 (OSRAM)
TW (1) TWI459947B (OSRAM)
UA (1) UA98966C2 (OSRAM)
WO (1) WO2009001968A1 (OSRAM)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI459947B (zh) * 2007-06-26 2014-11-11 Otsuka Pharma Co Ltd 苯并氮呯化合物及藥學製劑
JP5656399B2 (ja) * 2008-12-26 2015-01-21 大塚製薬株式会社 医薬及び医薬製剤
CN102030709B (zh) * 2009-09-25 2013-10-16 江苏豪森医药集团有限公司 用作加压素受体拮抗剂的苯并氮杂卓类化合物
CN104829531A (zh) * 2009-10-26 2015-08-12 大塚制药株式会社 苯并氮杂*化合物
GB201105537D0 (en) 2011-03-31 2011-05-18 Vantia Ltd New process
CN102260213B (zh) * 2011-05-31 2013-05-15 重庆福安药业(集团)股份有限公司 一种托伐普坦的制备方法
TWI633887B (zh) 2012-05-31 2018-09-01 大塚製藥股份有限公司 用於預防及／或治療多囊性腎臟病之藥物
JP6265999B2 (ja) 2012-12-28 2018-01-24 大塚製薬株式会社 光学活性のトルバプタンを含む注射用持効性製剤及びその製造方法
US9505737B2 (en) 2013-01-11 2016-11-29 Corsair Pharma, Inc. Treprostinil derivative compounds and methods of using same
TWI660748B (zh) * 2013-03-01 2019-06-01 日商大塚製藥股份有限公司 用於口服投藥之包含非晶型托伐普坦（Ｔｏｌｖａｐｔａｎ）的懸浮液
TW201605488A (zh) 2013-10-15 2016-02-16 大塚製藥股份有限公司 用以預防及／或治療多囊腎病之藥物
US11911369B2 (en) * 2015-03-03 2024-02-27 Biohaven Therapeutics Ltd. Prodrugs of riluzole and their method of use
WO2019003433A1 (ja) * 2017-06-30 2019-01-03 大塚製薬株式会社 ベンゾアゼピン誘導体
CN107540672A (zh) * 2017-10-10 2018-01-05 牡丹江医学院 一种治疗肝硬化的药物及其合成方法
HU231206B1 (hu) 2017-12-15 2021-10-28 Richter Gedeon Nyrt. Triazolobenzazepinek
TW201938171A (zh) 2017-12-15 2019-10-01 匈牙利商羅特格登公司 作為血管升壓素Ｖ１ａ受體拮抗劑之三環化合物
JP2020011957A (ja) * 2019-07-22 2020-01-23 コルセア ファーマ インコーポレイテッド トレプロスチニル誘導体化合物およびその使用方法
CN112851583B (zh) * 2021-01-19 2023-09-08 徐州医科大学 新型苯并氮杂䓬类化合物、组合物及其用途
EP4293032A4 (en) * 2021-02-10 2024-10-23 Shanghai Senhui Medicine Co., Ltd. BENZAZEPINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE
CN113112528A (zh) * 2021-04-26 2021-07-13 中南财经政法大学 异常行为监控方法、装置、设备及存储介质

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5045478A (en) * 1986-03-03 1991-09-03 Becton Dickinson And Company Vesicles and use thereof in an assay
US5258510A (en) * 1989-10-20 1993-11-02 Otsuka Pharma Co Ltd Benzoheterocyclic compounds
AU657424B2 (en) 1992-07-02 1995-03-09 Otsuka Pharmaceutical Co., Ltd. Oxytocin antagonist
TW270927B (OSRAM) * 1992-10-16 1996-02-21 Otsuka Pharma Co Ltd
GB9726695D0 (en) 1997-12-17 1998-02-18 Smithkline Beecham Plc Novel compounds
JP4210355B2 (ja) 1997-07-03 2009-01-14 大塚製薬株式会社 固形製剤組成物
NZ510551A (en) 1998-09-29 2003-03-28 American Cyanamid Co Substituted 3-cyanoquinolines useful as protein tyrosine kinases inhibitors
US6642270B2 (en) 2000-05-15 2003-11-04 Paratek Pharmaceuticals, Inc. 7-substituted fused ring tetracycline compounds
AU2005302162A1 (en) 2004-11-02 2006-05-11 Shire Llc Prodrugs of ribavirin with improved hepatic delivery
CN101346390B (zh) * 2005-12-27 2011-11-09 大塚制药株式会社 水溶性苯并氮杂*化合物及其药物组合物
TWI459947B (zh) * 2007-06-26 2014-11-11 Otsuka Pharma Co Ltd 苯并氮呯化合物及藥學製劑

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